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1-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-4-(2-methyl-1H-imidazol-1-yl)butan-1-one
1-[3-(2-ethylphenoxy)azetidin-1-yl]-2-(1H-pyrazol-1-yl)butan-1-one
5-(methoxymethyl)-N-[2-(3-phenyl-1,2,4-oxadiazol-5-yl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine
(3S,4R)-4-(pyridin-4-yl)-1-[3-(trifluoromethyl)-1H-pyrazole-5-carbonyl]pyrrolidine-3-carboxylic acid
methyl({[2-(morpholin-4-yl)pyrimidin-5-yl]methyl})[1-(pyridin-2-yl)ethyl]amine
4-{1-[4-(1H-1,2,3,4-tetrazol-1-ylmethyl)benzoyl]piperidin-4-yl}thiomorpholine
1-cyclohexanecarbonyl-N-{1-[(3-fluorophenyl)methyl]-4-methyl-1H-pyrazol-5-yl}pyrrolidine-2-carboxamide
4-[(2-ethoxyphenyl)methyl]-3-[2-(1,4-oxazepan-4-yl)-2-oxoethyl]piperazin-2-one
3-[2-(dimethylamino)ethyl]-8-[4-(pyrrolidin-1-yl)benzoyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
(3aR,6aR)-2-methanesulfonyl-5-{thieno[3,2-d]pyrimidin-4-yl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-butyl-5-{1-[3-(1,2-oxazinan-2-yl)propanoyl]pyrrolidin-2-yl}thiophene-2-carboxamide
1-{4-[3-(3-methoxyphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]phenyl}ethan-1-one
N-{[3-(3-methoxyphenyl)-1,2-oxazol-5-yl]methyl}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
(3R,4S)-4-(propan-2-yl)-1-{[2-(propan-2-yl)-1,3-oxazol-4-yl]methyl}pyrrolidin-3-amine
N-cyclohexyl-3-{[4-(3-hydroxy-3-methylbutyl)phenyl]formamido}propanamide
N,1,3,5-tetramethyl-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-1H-pyrazole-4-carboxamide
1-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-3-[5-(4-methylphenyl)-1,3,4-thiadiazol-2-yl]urea
2-{1-[(2-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[(2-methyl-1,3-thiazol-4-yl)methyl]acetamide
N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]-5-(pyridin-4-yl)pyrazolo[1,5-a]pyrimidin-7-amine
2-cyclopropyl-4-hydroxy-N-[(2-methoxy-4,6-dimethylpyridin-3-yl)methyl]pyrimidine-5-carboxamide
2-[(3-methoxyphenyl)methyl]-8-(3-methyl-1,2-oxazole-5-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
(3S)-1-(8-fluoroquinoline-2-carbonyl)piperidin-3-amine
1-[(1R,3S)-1-hydroxy-3-methoxy-7-azaspiro[3.5]nonan-7-yl]-3-{imidazo[1,2-a]pyridin-2-yl}propan-1-one
2-chloro-5-[2-(hydroxymethyl)phenyl]-N-methylbenzamide
2-(2,5-dioxoimidazolidin-1-yl)-N-[(1-ethyl-1H-1,3-benzodiazol-2-yl)methyl]acetamide
5-{[3-(diphenylmethyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}-1,3-oxazolidin-2-one
(3S,4R)-1-[2-(dimethyl-1,2-oxazol-4-yl)ethyl]-4-(4-methoxyphenyl)-N,N-dimethylpyrrolidin-3-amine
N-methyl-2-[1-(3,3,3-trifluoropropyl)piperidin-4-yl]acetamide
4-[4-(2,5-dihydro-1H-pyrrol-1-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-7-carbonyl]-N-methyl-1,3-thiazol-2-amine
(3aR,6aR)-2-acetyl-5-[(4-acetyl-1-methyl-1H-pyrrol-2-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
(3S,4S)-N-(4-fluoro-3-methoxyphenyl)-3-hydroxy-4-(piperidin-1-yl)pyrrolidine-1-carboxamide
1-(4-fluorophenyl)-5-(2-methoxyethyl)-3-phenyl-1H-1,2,4-triazole
(4aR,7aS)-1-(2-methoxyacetyl)-4-(2-methoxypyridine-4-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(4aR,7aS)-1-(cyclopropylmethyl)-4-{2-[4-(hydroxymethyl)phenyl]acetyl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(2R,4R)-4-hydroxy-N-(2-{[(3-methylphenyl)methyl]carbamoyl}phenyl)pyrrolidine-2-carboxamide
1-(azepan-1-yl)-3-(3-{[methyl(pyridin-2-ylmethyl)amino]methyl}phenoxy)propan-2-ol
3-(1-methoxypropan-2-yl)-6-methyl-3H,4H-thieno[2,3-d]pyrimidin-4-one
N-[(5-phenyl-1,2-oxazol-3-yl)methyl]-1-(prop-2-en-1-yl)-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-{6-[(2-hydroxyethyl)amino]pyrimidin-4-yl}-4-(1H-pyrazol-1-yl)piperidine-4-carboxylic acid
(2R,3S,6R)-3-(3,5-difluorophenyl)-5-(1H-pyrazole-3-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
2-[4-(3-benzyl-1H-1,2,4-triazol-5-yl)piperidin-1-yl]pyrimidine
2-(pyridin-4-yl)-N-[2-(1,3-thiazol-2-yl)ethyl]quinoline-4-carboxamide
N-(pyrimidin-4-ylmethyl)-6-[3-(trifluoromethyl)phenyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
N-{[7-chloro-2-(4-methoxyphenyl)quinolin-3-yl]methyl}-2-(dimethyl-1H-1,2,4-triazol-1-yl)-N-(oxolan-2-ylmethyl)acetamide
N-benzyl-1-{2-[(3-methylthiophen-2-yl)formamido]ethyl}-1H-1,2,3-triazole-4-carboxamide
N,N-dimethyl-4-(3-methyl-1-propyl-1H-pyrazole-4-carbonyl)piperazine-1-sulfonamide
1-[(2E)-3-phenylprop-2-en-1-yl]-4-(pyrrolidine-3-carbonyl)piperazine
N-[(dimethyl-1,3-thiazol-2-yl)methyl]-5-{[2-(propan-2-yl)-1H-imidazol-1-yl]methyl}-1H-pyrazole-3-carboxamide
N-[3-(2-ethyl-1H-imidazol-1-yl)propyl]-3,3-dimethylcyclohexan-1-amine
4-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-3-[2-(morpholin-4-yl)-2-oxoethyl]piperazin-2-one