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N-(1-{[4-(2-methylpropyl)phenyl]methyl}piperidin-3-yl)-3-(1H-1,2,4-triazol-1-yl)propanamide
1-(1H-imidazol-2-ylmethyl)-4-[4-(methylamino)pyrimidin-2-yl]-1,4-diazepan-6-ol
9-{[2-(4-methoxyphenyl)pyrimidin-5-yl]methyl}-6-oxa-9-azaspiro[4.5]decane
N-(4,6-dimethyl-2-oxo-1,2-dihydropyridin-1-yl)-3-(5-phenyl-2H-1,2,3,4-tetrazol-2-yl)propanamide
1-[2-(4-methylpentyl)morpholine-4-carbonyl]cyclopropane-1-carboxamide
ethyl 4-[(4-chlorophenyl)methyl]-1-(2,6-dimethylpyrimidine-4-carbonyl)piperidine-4-carboxylate
3,3,3-trifluoro-1-{4-hydroxy-4-[3-(trifluoromethyl)phenyl]piperidin-1-yl}propan-1-one
N-({1-[2-(2-methoxyphenyl)ethyl]piperidin-4-yl}methyl)-N-methyl-3-(1,2-oxazolidin-2-yl)propanamide
(3S,4R)-4-(3-methoxyphenyl)-1-(pyridine-3-carbonyl)pyrrolidine-3-carboxylic acid
N-[(5-chlorothiophen-2-yl)methyl]-1-(2-hydroxyethyl)-1H-1,3-benzodiazole-5-carboxamide
5-methyl-1-({4-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]phenyl}methyl)-1H-1,2,3,4-tetrazole
3-methyl-N-(1-{1-[(1-phenyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)butanamide
(1S,5R)-6-(cyclobutylmethyl)-N-[(3-fluorophenyl)methyl]-7-oxo-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
9-[(2,5-difluorophenyl)methyl]-2-[2-(dimethylamino)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
2-(5-{[methyl(propan-2-yl)amino]methyl}-1H-1,2,3,4-tetrazol-1-yl)-N-[1-(5,6,7,8-tetrahydronaphthalen-2-yl)ethyl]acetamide
1-[3-(1,4-oxazepan-4-ylmethyl)phenoxy]-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-ol
6-(4-fluorophenyl)-N-[2-(propane-2-sulfonyl)ethyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
(2S,4R)-4-amino-N,N-diethyl-1-[6-oxo-2-(propan-2-yl)-1,6-dihydropyrimidine-5-carbonyl]pyrrolidine-2-carboxamide
2-(cyclopropylmethyl)-8-(3-hydroxy-4-methylbenzoyl)-2,8-diazaspiro[5.5]undecan-3-one
2-{5-methanesulfonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}ethan-1-amine
{[4-(butan-2-yloxy)-3-ethoxyphenyl]methyl}[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]amine
5-(ethoxymethyl)-1-[(3-methylphenyl)methyl]-3-(1H-1,2,4-triazol-1-ylmethyl)-1H-1,2,4-triazole
1-methyl-N-[(3-methyloxetan-3-yl)methyl]-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
1-(2-methoxyethyl)-5-[3-(oxan-4-yl)-1H-1,2,4-triazol-5-yl]piperidin-2-one
(3R,4R)-1-[3-chloro-4-(pyrrolidin-1-yl)benzoyl]-4-ethylpiperidine-3,4-diol
2-(2,3-difluorophenoxymethyl)-N-methyl-N-[2-(1H-pyrazol-4-yl)ethyl]-1,3-oxazole-4-carboxamide
2-methoxy-4-{2-[3-oxo-3-(pyrrolidin-1-yl)propyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl}pyridine-3-carbonitrile
(2,3-dihydro-1-benzofuran-2-ylmethyl)({[2-(4-methoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl})methylamine
(4aS,7aR)-1-(4-ethoxybenzoyl)-4-propyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[2-(4-chlorophenyl)-2-hydroxyethyl]-2-methyl-1,3-thiazole-4-carboxamide
(2S,4S,5R)-5-(2-chlorophenyl)-4-(4-hydroxypiperidine-1-carbonyl)-1,2-dimethylpyrrolidine-2-carboxylic acid
1-[2-chloro-5-(morpholin-4-yl)phenyl]-3-[3-(1H-imidazol-1-yl)propyl]urea
N-[(3-cyclohexyl-1,2,4-oxadiazol-5-yl)methyl]-5,7-dimethylpyrido[2,3-d]pyrimidin-4-amine
4-(3,6-dimethylpyrazin-2-yl)-N-{3-[(methylcarbamoyl)methyl]phenyl}piperazine-1-carboxamide
4-(4-methanesulfonylphenoxymethyl)-5-methyl-2-(2-methylphenyl)-1,3-oxazole
2-(5-{1H-pyrazolo[1,5-a]imidazole-7-carbonyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl)-1H-1,3-benzodiazole
2-methyl-4-[3-(2-phenylethyl)-5-[1-(1H-pyrazol-1-yl)propyl]-1H-1,2,4-triazol-1-yl]pyridine
N-methyl-4-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}-N-(1H-pyrazol-5-ylmethyl)butanamide
N-[3-(ethylcarbamoyl)phenyl]-3-[(4-fluorophenyl)methyl]piperidine-1-carboxamide
6,6-dimethyl-N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}-5-oxothiomorpholine-3-carboxamide
1-[(2R,6R)-6-methyl-2-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridin-1-yl]-2-(piperazin-1-yl)ethan-1-one
1-(2-methylphenyl)-3-[1-(1-{[4-(propan-2-yloxy)phenyl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]urea
N-[2-(adamantan-1-yl)propan-2-yl]-3-[5-(5-methyl-1,2-oxazol-3-yl)-1,3,4-oxadiazol-2-yl]propanamide
N-{1-[1-(5-methyl-1,2-oxazole-3-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}-3-phenylpropanamide
N-{2-[cyclopentyl(methyl)amino]ethyl}-N,5,6-trimethylpyrimidin-4-amine
3-[(2-methoxyphenyl)methyl]-5-(oxan-2-yl)-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazole
2-(3-methoxypropyl)-8-[2-(phenylsulfanyl)ethyl]-2,8-diazaspiro[4.5]decan-3-one
1-{[5-(1-cyclohexyl-1H-1,2,4-triazol-5-yl)furan-2-yl]methyl}-4-methylpiperazine
(3R,4R)-1-[(3-chloro-1-benzothiophen-2-yl)methyl]-4-[4-(pyridin-2-yl)piperazin-1-yl]piperidin-3-ol
8-{[4-chloro-2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl}-1,3-dioxa-8-azaspiro[4.5]decan-2-one