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N-[(dimethyl-1,2-oxazol-4-yl)methyl]-4-hydroxy-N-methyl-2-(phenoxymethyl)pyrimidine-5-carboxamide
2-methoxy-N-[3-(1-{[(2-methyl-2H-1,2,3-triazol-4-yl)carbamoyl]methyl}-1H-pyrazol-4-yl)phenyl]acetamide
(3S,4S)-N-[3-(dimethylamino)phenyl]-3,4-bis(hydroxymethyl)pyrrolidine-1-carboxamide
1-[2-(1-{pyrazolo[1,5-a]pyrimidin-3-ylmethyl}piperidin-4-yl)ethyl]pyrrolidin-2-one
N-methyl-N'-(4-methylphenyl)-N-[(3-methylthiophen-2-yl)methyl]propanediamide
3-[(3R,4S)-4-(morpholin-4-yl)-1-(quinoline-4-carbonyl)piperidin-3-yl]propan-1-ol
2-methyl-4-[4-(piperidine-1-carbonyl)piperidin-1-yl]pyridine
2-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-N-[(2E)-3-phenylprop-2-en-1-yl]-N-propylacetamide
2-cyclohexyl-6-[4-(morpholine-4-carbonyl)piperidine-1-carbonyl]-1,3-benzoxazole
1-[2-(1H-imidazol-2-yl)benzoyl]-4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine
2,5-dimethyl-3-{3-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyrazine
[(2S,4R)-4-(dimethylamino)-1-{[5-(2-methylpropyl)thiophen-2-yl]methyl}pyrrolidin-2-yl]methanol
N-cyclopropyl-4-methoxy-3-{[1-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)piperidin-4-yl]oxy}benzamide
1-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-(2-methylpropyl)-5-(oxolan-3-yl)-1H-1,2,4-triazole
2-{1-[(1-ethyl-1H-imidazol-2-yl)methyl]-1H-imidazol-2-yl}-1-(4-methoxyphenyl)-1H-imidazole
2-{4-[(4-ethylpiperazin-1-yl)methyl]phenyl}-6-(oxolan-2-yl)-3,4-dihydropyrimidin-4-one
(2R,3R,6R)-3-(4-methoxyphenyl)-5-(1,3-thiazol-2-yl)-1,5-diazatricyclo[5.2.2.02,6]undecane
2-methyl-N-{3-[3-(6-methylpyridazin-3-yl)-1,2,4-oxadiazol-5-yl]phenyl}propanamide
3-{1-[(4,6-dimethylpyrimidin-2-yl)amino]ethyl}adamantan-1-ol
{[5,8-dimethoxy-2-(3-methoxyphenyl)quinolin-3-yl]methyl}(2-phenylethyl)amine
3-[(1-ethyl-1H-indazol-3-yl)methyl]-1-(2-methyl-2,3-dihydro-1-benzofuran-5-yl)urea
1-(2-aminoethyl)-4-(naphthalen-2-yloxy)piperidine-4-carboxylic acid
N-({2-[3-(4-methoxybenzenesulfonamido)phenyl]-5-methyl-1,3-oxazol-4-yl}methyl)oxane-4-carboxamide
prop-2-en-1-yl 2-(5-fluoro-1H-1,3-benzodiazol-2-yl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carboxylate
2-{[4-(2,4-difluorophenyl)-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
N-({1-[ethyl(methyl)amino]cyclopentyl}methyl)-3-(3-fluorophenyl)-1H-pyrazole-4-carboxamide
4-{4,6-dimethyl-11-oxo-3,7,8,10-tetraazatricyclo[7.4.0.02,7]trideca-1,3,5,8-tetraen-13-yl}-1H-pyrazole-3-carboxylic acid
N-(furan-2-ylmethyl)-8-methoxy-N-(prop-2-en-1-yl)-3,4-dihydro-2H-1-benzopyran-3-carboxamide
[(4-ethyl-5-{1-[(4-methoxyphenyl)methyl]piperidin-4-yl}-4H-1,2,4-triazol-3-yl)methyl]dimethylamine
8-(dimethyl-1,2-oxazole-4-carbonyl)-3-(pentan-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
5-{1-[(4-chlorophenyl)methyl]-4-hydroxypiperidin-4-yl}-N-(1,4-dioxan-2-ylmethyl)-1-benzofuran-2-carboxamide
ethyl 1-[(dimethyl-1,2-oxazol-4-yl)sulfonyl]-4-{[3-(trifluoromethyl)phenyl]methyl}piperidine-4-carboxylate
(3S,4R)-N,N-dimethyl-1-[(3-methyl-1-phenyl-1H-pyrazol-4-yl)methyl]-4-(propan-2-yl)pyrrolidin-3-amine
4-(4-fluorophenyl)-N-[5-(3-methylphenyl)-4H-1,2,4-triazol-3-yl]-1,2,3,6-tetrahydropyridine-1-carboxamide
1-[4-(2-fluoro-4-methoxyphenyl)-1H-1,2,3-triazol-1-yl]-3-(pyrrolidin-1-yl)propan-2-ol
(3R,5S)-1-benzyl-N3-(4-fluorophenyl)-N5-(2-phenylethyl)piperidine-3,5-dicarboxamide
1-{4-[(1-benzyl-1H-imidazol-5-yl)methyl]-6-hydroxy-1,4-diazepan-1-yl}ethan-1-one
N-({3-[2-(2-fluorophenyl)ethoxy]phenyl}methyl)-N-(oxolan-2-ylmethyl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
(5-{[({1-[2-(3-fluorophenyl)ethyl]piperidin-4-yl}methyl)(methyl)amino]methyl}furan-2-yl)methanol
N-methyl-N-(1,3-thiazol-2-ylmethyl)-1-{[3-(trifluoromethyl)phenyl]methyl}-1H-1,2,3-triazole-4-carboxamide
5-{4-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidine-1-carbonyl}-2-(pyridin-2-yl)pyrimidin-4-ol
2-amino-N-{imidazo[1,2-a]pyrazin-3-ylmethyl}-4-methyl-1,3-thiazole-5-carboxamide
4-(2,5-dihydro-1H-pyrrole-1-carbonyl)-1,2,3,4-tetrahydroquinolin-2-one
1-(5-{[(2R,6R)-6-methyl-2-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridin-1-yl]methyl}imidazo[2,1-b][1,3]thiazole-6-carbonyl)azocane
N-({5-[(2-fluoro-5-methylphenyl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-methoxyacetamide
1-(benzyloxy)-8-{2-[3-(trifluoromethyl)phenyl]acetyl}-1,8-diazaspiro[4.5]decan-2-one
4-(4-methanesulfonylphenyl)-8-(trifluoromethyl)quinoline
(3S,5R)-1-[(2,4-difluorophenyl)methyl]-5-[(pyridin-4-ylmethyl)carbamoyl]piperidine-3-carboxylic acid
2-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-N-ethyl-N-[(4-fluorophenyl)methyl]acetamide
N-(2,2,6,6-tetramethylpiperidin-4-yl)-4-(trimethyl-1H-pyrazol-4-yl)pyrimidin-2-amine