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(2-phenylpropyl)[(5,6,7-trimethoxy-2-phenylquinolin-3-yl)methyl]amine
1-(4-methanesulfonylphenyl)-3-[1-(pyrimidin-2-yl)piperidin-3-yl]urea
3-[1-(4-methylphenyl)cyclopentyl]-5-(oxolan-3-yl)-1,2,4-oxadiazole
methyl 1-(cyclopropylmethyl)-2-oxo-3-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}-2,3-dihydro-1H-1,3-benzodiazole-5-carboxylate
N-(2-methoxyethyl)-N-(1,3-thiazol-2-ylmethyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-(oxolan-2-ylmethyl)-3-[5-(3-phenylpropyl)-1,3,4-oxadiazol-2-yl]propanamide
3-[(2-methylprop-2-en-1-yl)oxy]-N-[(1-methylpyrrolidin-3-yl)methyl]benzamide
3-[3-(4-phenoxybenzoyl)piperidine-1-carbonyl]pyridin-1-ium-1-olate
2-methyl-5-{2-oxo-2-[(1S,5R)-3-(pyridin-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethyl}-3,4-dihydropyrimidin-4-one
N-[(5-cyclopropyl-1,2-oxazol-3-yl)methyl]-6-(4-fluorophenyl)-N-methylimidazo[2,1-b][1,3]thiazole-3-carboxamide
N-{[2-(dimethylamino)-5,8-dimethoxyquinolin-3-yl]methyl}-N-(furan-2-ylmethyl)-3-(3-methyl-1H-pyrazol-1-yl)propanamide
(1R,5R)-6-(cyclopropylmethyl)-3-[3-(thiophen-3-yl)-1H-pyrazole-5-carbonyl]-3,6-diazabicyclo[3.2.2]nonane
3-[(3R,4S)-1-[2-(benzyloxy)acetyl]-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propanoic acid
1-(2-ethylpyrimidine-5-carbonyl)-N-(3-fluorophenyl)piperidin-3-amine
N-[3-(furan-2-yl)phenyl]-1-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]piperidine-4-carboxamide
N-(2-chloro-4-{2-[2-(dimethylamino)pyrimidin-5-yl]-1H-imidazol-1-yl}phenyl)propanamide
2,4-dimethoxy-6-{4-[(3-methylpyridin-2-yl)methyl]piperazine-1-carbonyl}pyrimidine
1-(azepan-1-yl)-3-[3-({[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]amino}methyl)phenoxy]propan-2-ol
5-{3-[5-(5-ethylfuran-2-yl)-4-phenyl-1H-imidazol-1-yl]propyl}-1H-1,2,3,4-tetrazole
2-{2-[(4-methoxyphenyl)methyl]pyrimidin-4-yl}pyridine-4-carboxylic acid
N-methyl-3-(3-{4-[3-(trifluoromethyl)phenyl]piperazin-1-yl}piperidin-1-yl)propanamide
ethyl 4-[4-(4-{[1-(1,3-thiazol-2-yl)ethyl]amino}piperidin-1-yl)benzoyl]piperazine-1-carboxylate
2-chloro-4-[2-(pyrrolidine-1-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carbonyl]pyridine
N-methyl-5-(propan-2-yl)-N-{[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}-1,2-oxazole-3-carboxamide
1-{5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}-4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazine
2-[(1S,5R)-6-[(4-ethylphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-3-yl]-N,N-dimethylacetamide
2-(4-{[(1R,5R)-3-(pyridine-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}phenoxy)ethan-1-ol
2-[(3S,4R)-3-(propan-2-yl)-4-{2-[(propan-2-yl)amino]pyrimidine-5-amido}pyrrolidin-1-yl]acetic acid
9-ethyl-1-methyl-4-[2-(thiophen-3-yl)acetyl]-1,4,9-triazaspiro[5.6]dodecan-10-one
7-(3-chlorophenyl)-4-(2-methyl-1,3-thiazole-4-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
(3R,4R)-4-cyclopropyl-3-methyl-1-{[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}piperidin-4-ol
4-{2-[1-(4-chloro-3-methylbenzoyl)piperidin-2-yl]ethyl}morpholine
(4aS,7aR)-1-[2-(benzyloxy)ethyl]-4-(2-hydroxyethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-{1-azabicyclo[2.2.2]octan-3-yl}-2-(propan-2-yl)pyrimidine-5-carboxamide
(3R,4S)-4-(4-{[2-(trifluoromethyl)phenyl]methyl}-1,4-diazepan-1-yl)oxolan-3-ol
2-methoxyethyl 3-(4,4,4-trifluorobutanamido)azepane-1-carboxylate
3-(1-methyl-1H-imidazol-2-yl)-6-[4-(4-phenyl-1H-pyrazol-5-yl)piperidin-1-yl]pyridazine
2-{2-[(3R,4R)-3-(hydroxymethyl)-4-(morpholin-4-ylmethyl)pyrrolidin-1-yl]-2-oxoethyl}-6-methyl-2,3-dihydropyridazin-3-one
3-{[4-(4-benzyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)piperidin-1-yl]methyl}benzonitrile
7-(cyclopropylmethyl)-2-[6-(4H-1,2,4-triazol-4-yl)pyridine-3-carbonyl]-2,7-diazaspiro[4.5]decan-6-one
N-[(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)methyl]-1H-pyrrolo[2,3-b]pyridin-6-amine
(1R,3S)-7-{2-[(dimethylamino)methyl]-1,3-thiazole-4-carbonyl}-7-azaspiro[3.5]nonane-1,3-diol
6-ethoxy-4-methyl-2-(3-{4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazine-1-carbonyl}piperidin-1-yl)quinazoline
3-[1-(cyclohexylmethyl)-1H-pyrazol-5-yl]-1-[3-(4-methylpiperazin-1-yl)propyl]urea
(3S)-3-methyl-4-{[6-(4-methyl-1,4-diazepane-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}-1-(2-methylpropyl)piperazin-2-one
4-{4-[2-(2-hydroxyethyl)piperidine-1-carbonyl]phenyl}-2-methylbutan-2-ol
N-({5-methanesulfonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-5-methylthiophene-2-carboxamide
(1S,5R)-6-methyl-3-[(5-phenylthiophen-2-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
1-{[2-(4-methoxy-2,3-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidine-4-carbonitrile
3-{6-amino-1H-pyrrolo[2,3-b]pyridin-4-yl}-4-methoxy-N-methylbenzamide