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2-(1-benzofuran-2-yl)-2-[methyl(oxan-4-ylmethyl)amino]acetic acid
N-[(3S,4R)-1-(4-fluoro-2-methylbenzenesulfonyl)-4-propylpyrrolidin-3-yl]acetamide
1-[(3aS,6aS)-3a-(hydroxymethyl)-octahydrocyclopenta[c]pyrrol-2-yl]-2-(2-phenyl-1H-imidazol-1-yl)ethan-1-one
N-(2-fluorophenyl)-5-[4-(2-hydroxyethyl)-1H-pyrazol-1-yl]furan-2-carboxamide
2-(4-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}piperazin-1-yl)pyridine-3-carboxamide
2-{1-[5-(4-fluorophenyl)-1,2,4-triazin-3-yl]piperidin-3-yl}-1,3-benzoxazole
5-(2-{2-[(2-ethyl-6-methylpyrimidin-4-yl)amino]ethyl}morpholin-4-yl)-2-methyl-2,3-dihydropyridazin-3-one
1-(2,6-dimethylpyrimidine-4-carbonyl)-4-(3-methylpyridin-4-yl)-1,4-diazepane
2-(1H-indol-3-yl)-N-[(5-methylpyrazin-2-yl)methyl]-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-amine
N-[2-(morpholin-4-yl)-2-(pyridin-4-yl)ethyl]-1-[2-(piperidin-1-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
4-(1-benzyl-1H-imidazol-2-yl)-1-(5-ethyl-1,3-oxazole-4-carbonyl)piperidine
2-{[4-hydroxy-4-(5-methylpyridin-2-yl)piperidin-1-yl]methyl}-5-methoxy-4H-pyran-4-one
4-{1-[1-(4-methoxyphenyl)cyclopentanecarbonyl]piperidin-4-yl}pyrimidine
2-{3-[1-(2-ethoxyethyl)-1H-pyrazol-3-yl]phenyl}pyrazine
3-(4-methyl-1,3-thiazol-5-yl)-N-(pyridin-3-ylmethyl)-N-(thiophen-3-ylmethyl)propanamide
4-{3-[1-(pyrrolidin-1-yl)ethyl]phenyl}-1H-pyrazole-3-carbonitrile
N-({5-[(2-fluoro-5-methylphenyl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)methanesulfonamide
N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-1-benzoxepine-4-carboxamide
{[1-(cyclohexylmethyl)-2-cyclopropylmethanesulfonyl-1H-imidazol-5-yl]methyl}(methyl)(thiophen-2-ylmethyl)amine
2-[2-(propan-2-yl)-1H-imidazol-1-yl]-N-[3-(1,2,3,4-tetrahydroquinolin-1-yl)propyl]propanamide
2-(4-{[2-(4-fluoro-3-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazin-1-yl)pyrimidine
1-{1-[1-(4-chloro-3-fluorobenzoyl)piperidin-4-yl]ethyl}-4-methylpiperazine
N-[(1-{[3-(3-methoxyphenyl)phenyl]methyl}piperidin-4-yl)methyl]acetamide
2-{5-[2-(2-phenylethyl)piperidine-1-carbonyl]-1H-pyrazol-3-yl}phenol
N-[2-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-5-(morpholin-4-ylmethyl)furan-3-carboxamide
N-(1-{imidazo[2,1-b][1,3,4]thiadiazol-6-yl}ethyl)-3-(2-methyl-1H-indol-1-yl)propanamide
6-(3,4-dihydro-2H-1-benzopyran-3-carbonyl)-1-[2-(piperidin-1-yl)ethyl]-3-(pyridin-4-yl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
[3-ethyl-1-(3-fluoropyridin-4-yl)piperidin-3-yl]methanol
N-cyclohexyl-2-ethyl-N-(pyridin-2-ylmethyl)pyrimidine-5-carboxamide
N-[(2-methoxy-4,6-dimethylpyridin-3-yl)methyl]-2-[1-(2-methylpropyl)-3-oxopiperazin-2-yl]acetamide
3-fluoro-N-{1-[1-(3-phenylpropyl)piperidin-4-yl]-1H-pyrazol-5-yl}benzamide
[(5-chlorofuran-2-yl)methyl]({1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl})methylamine
4-{5-[4-(morpholin-4-yl)piperidine-1-carbonyl]pyridin-2-yl}benzamide
3-{[1-(3-methylpyridin-4-yl)-3-(propan-2-yl)-1H-1,2,4-triazol-5-yl]methyl}-3,4-dihydro-1,2,3-benzotriazin-4-one
4-{5-methyl-6-[(2-methylpyridin-3-yl)oxy]pyrimidin-4-yl}-1H-pyrrolo[2,3-b]pyridin-6-amine
2-[4-(2-methoxypyridine-3-carbonyl)-1-[(6-methylpyridin-2-yl)methyl]piperazin-2-yl]ethan-1-ol
3-[3-(propan-2-yloxy)benzoyl]-1-(propane-2-sulfonyl)piperidine
1-{1-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]piperidin-4-yl}piperidine-3-carboxylic acid
(1R,3S)-3-(2-aminoethoxy)-7-[(2,3-difluoro-6-methoxyphenyl)methyl]-7-azaspiro[3.5]nonan-1-ol
3-{ethyl[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]sulfamoyl}-N,N-dimethylbenzamide
2-[3-(3-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-N,6-dimethylpyrimidin-4-amine
(3R,5R)-N-{3-[(furan-2-ylmethyl)sulfanyl]propyl}-5-(pyrrolidine-1-carbonyl)piperidine-3-carboxamide
2-(2-{9-oxa-2-azaspiro[5.5]undecan-2-ylmethyl}phenoxy)acetic acid
5-methyl-N-[2-(3-phenylpiperidin-1-yl)ethyl]-1,3,4-oxadiazol-2-amine
11-[4-(2-fluorophenyl)piperazin-1-yl]-4-[3-(propan-2-yloxy)propyl]-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
(2R,3R,6R)-5-{7-methyl-[1,2,4]triazolo[4,3-a]pyrimidine-3-carbonyl}-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecane
1-[4-(5-{[(2-hydroxyethyl)(methyl)amino]methyl}-4-methyl-4H-1,2,4-triazol-3-yl)piperidin-1-yl]ethan-1-one
1-[(4aR,8aR)-7-[2-(4-chloro-1H-pyrazol-1-yl)ethyl]-4a-hydroxy-decahydro-2,7-naphthyridin-2-yl]-2-methoxyethan-1-one
N4-[3-(2-methoxyphenoxy)propyl]-N4,6-dimethylpyrimidine-2,4-diamine
1-cyclopentyl-N-[2-(4,5-dimethyl-1H-1,3-benzodiazol-2-yl)ethyl]-6-oxopiperidine-3-carboxamide