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N-methyl-N-{[2-(methylamino)pyrimidin-5-yl]methyl}-5-oxo-1-[4-(propan-2-yl)phenyl]pyrrolidine-3-carboxamide
(7R,9aR)-6,9-dioxo-N-phenyl-7-(propan-2-yl)-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxamide
ethyl 4-{[2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl]amino}piperidine-1-carboxylate
2-(1-benzyl-1H-pyrazol-4-yl)-2-[methyl(pyridin-2-ylmethyl)amino]acetic acid
7-fluoro-2-oxo-N-[1-(thiophen-3-yl)propan-2-yl]-1,2-dihydroquinoline-4-carboxamide
4-[4-(1H-imidazol-1-ylmethyl)phenyl]-N,N-dimethylbenzamide
3-[2-(dimethylamino)-2-(5-methylfuran-2-yl)ethyl]-1-(2-ethyl-1H-1,3-benzodiazol-6-yl)urea
1-{4-[(oxolan-2-ylmethyl)amino]-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl}ethan-1-one
N-[(4-hydroxyphenyl)methyl]-1-(oxan-4-yl)piperidine-4-carboxamide
ethyl 2-{3-[2-(quinolin-3-yl)pyridin-4-yl]pyrrolidin-1-yl}acetate
2-{2-[4-(2-hydroxyethyl)piperazin-1-yl]-4-(morpholin-4-yl)pyrimidin-5-yl}-2-methylpropanoic acid
4-({5-[(5-propylfuran-2-yl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-1,4-oxazepane
1-(2-{[5-(3-benzyl-1,2,4-oxadiazol-5-yl)pyridin-2-yl]amino}ethyl)piperidin-2-one
(2S,4S)-1-(2,3-dihydro-1H-inden-2-yl)-4-[(naphthalen-2-ylmethyl)amino]-N-(pyridin-3-ylmethyl)pyrrolidine-2-carboxamide
(1-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)({2-[2-(1H-imidazol-1-yl)ethoxy]-3-methoxyphenyl}methyl)amine
N-(2-methoxy-5-methylphenyl)-2-[2-(oxolan-3-yl)-1H-imidazol-1-yl]acetamide
2-{[({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)(2-methoxyethyl)amino]methyl}-4-methoxyphenol
3-[2-(2,6-difluorophenyl)ethyl]-1-(1H-pyrrole-2-carbonyl)piperidine
4-{[(4aS,8aR)-1-[2-(methylamino)ethyl]-2-oxo-decahydro-1,6-naphthyridin-6-yl]methyl}benzonitrile
3-(2-methylphenyl)-1-{[(1s,4s)-4-aminocyclohexyl]methyl}pyrrolidin-3-ol
3-({[2-(4-chloro-1H-pyrazol-1-yl)ethyl]amino}methyl)piperidin-3-ol
2-{[3-(hydroxymethyl)-3-(prop-2-en-1-yl)piperidin-1-yl]methyl}benzoic acid
2-[1-butyl-5-(5-fluoro-1,3-dimethyl-1H-indol-2-yl)-1H-1,2,4-triazol-3-yl]acetamide
1-{4-[(2-ethoxybutyl)amino]-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl}ethan-1-one
N-(1H-imidazol-2-ylmethyl)-3-[3-(2-methoxyphenyl)-1,2,4-oxadiazol-5-yl]propanamide
2-(4-chloro-2-methylphenoxy)-1-{5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepin-8-yl}propan-1-one
(3R,4S)-1-(1-tert-butyl-1H-pyrrole-3-carbonyl)-3,4-dimethylpiperidin-4-ol
(3R)-3,4,4-trimethyl-1-[2-(methylamino)-1,3-thiazole-4-carbonyl]pyrrolidin-3-ol
7-(2-methylphenyl)-4-(thiophen-3-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-[2-(3-fluorophenyl)ethyl]-1-(naphthalen-1-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
2-[(2-methoxyethyl)(methyl)amino]-2-(6-methoxypyridin-3-yl)acetic acid
N-[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl]-N-ethyl-2-(thiophen-2-yl)-1,3-thiazole-4-carboxamide
N,N-diethyl-1-[7-(pyridine-3-carbonyl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl]pyrrolidin-3-amine
3-[2-(4-fluorophenyl)ethyl]-1-[5-(methoxymethyl)furan-2-carbonyl]piperidine
{3-[4-(3,6-dimethylpyrazin-2-yl)piperazin-1-yl]propyl}diethylamine
2-[(4-methyl-1,3-thiazol-2-yl)sulfanyl]-1-{5-methyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}ethan-1-one
1,4,6-trimethyl-3-(4-phenyl-1,2,3,6-tetrahydropyridine-1-carbonyl)-1,2-dihydropyridin-2-one
2-methyl-5-phenyl-N-(pyrimidin-4-ylmethyl)pyrazolo[1,5-a]pyrimidin-7-amine
2-cyclohexyl-N-(2-methanesulfonamidoethyl)-1,3-benzoxazole-6-carboxamide
N-[2-(4-chloro-3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-2,3-dimethylquinoxaline-6-carboxamide
N-[(4-ethylphenyl)methyl]-5-(methoxymethyl)-N-methylpyrazolo[1,5-a]pyrimidin-7-amine
1-{[2-(3,4-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(2-methoxyphenoxy)piperidine
1-(6-ethyl-4-methylquinolin-2-yl)azetidin-3-ol
2-(2-methoxyphenyl)-1-{2-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidin-1-yl}ethan-1-one
2-[2-chloro-4-({5-hydroxy-1-oxa-9-azaspiro[5.5]undecan-9-yl}methyl)phenoxy]acetamide
(3aR,6aR)-2-(propylcarbamoyl)-5-(pyridin-4-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-(3-{3-[3-(morpholin-4-yl)-3-oxopropyl]piperidine-1-carbonyl}phenyl)acetamide
N-ethyl-1-methyl-N-[2-(5-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-1H-imidazole-2-carboxamide
9-[(4-methanesulfonylphenyl)methyl]-2-(prop-2-en-1-yl)-2,9-diazaspiro[5.5]undecan-3-one
N-{2-[7-(cyclohex-3-en-1-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}-2-(4-fluorophenyl)acetamide