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1-[2-(4-methoxyphenyl)ethyl]-3-(3-methyl-1,2,4-thiadiazol-5-yl)urea
4-({1-[6-(thiomorpholin-4-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl]piperidin-4-yl}methyl)morpholine
N-[(1-methanesulfonylpiperidin-3-yl)methyl]-2-(2-methoxyphenoxy)acetamide
1-(1,3-dioxo-2-{spiro[bicyclo[2.2.1]heptane-7,1'-cyclopropan]-2-en-5-ylmethyl}-2,3-dihydro-1H-isoindol-4-yl)-N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]piperidine-3-carboxamide
2-{2-[(1R,2R,6S,7S)-4-azatricyclo[5.2.1.02,6]decan-4-yl]-2-oxoethyl}-1,2-dihydroisoquinolin-1-one
8-(2,1,3-benzothiadiazol-5-ylmethyl)-3-(2,3-dihydro-1H-inden-2-yl)-1-ethyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-methyl-4-[4-(pyrrolidine-1-carbonyl)piperidine-1-carbonyl]pyridin-2-amine
4-(5-{3-[3-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl}pyridin-2-yl)piperazine-1-carboxamide
N-(oxolan-2-ylmethyl)-N-(thiophen-3-ylmethyl)-1,2,3-thiadiazole-4-carboxamide
3-({4-[(3-methylpyridin-2-yl)methyl]piperazin-1-yl}methyl)pyrrolidin-3-ol
2-{2-[(3S,4S)-3-(dimethylamino)-4-hydroxypyrrolidin-1-yl]-4-(morpholin-4-yl)pyrimidin-5-yl}-2-methylpropanoic acid
2-[1-(2,3-dihydro-1H-inden-4-yl)-5-[2-(methylamino)-1,3-thiazol-4-yl]-1H-1,2,4-triazol-3-yl]acetamide
4-{[4-(difluoromethoxy)phenyl]methyl}-1,3λ6,4-oxathiazinane-3,3-dione
1,1,1-trifluoro-3-({5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}amino)propan-2-ol
N-[2-(cyclohex-1-en-1-yl)ethyl]-1-ethyl-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-(4,7-dimethyl-2-oxo-2H-chromen-6-yl)-4-methylpyridine-3-carboxamide
9-(2,1,3-benzoxadiazol-5-yl)-1-ethyl-1H,2H,3H,6H,7H,8H,9H-[1,4]oxazino[3,2-g]quinoline-2,7-dione
3-chloro-4-hydroxy-N-(1-propylpyrrolidin-3-yl)benzamide
4-(1H-imidazol-2-yl)-1-(1-phenyl-1H-1,2,3-triazole-4-carbonyl)piperidine
3-[1-(2-benzyl-1,3-thiazole-4-carbonyl)piperidin-2-yl]pyridine
4-(4-methyl-3-phenyl-1H-pyrazole-5-carbonyl)-2-(trifluoromethyl)morpholine
4-({4-[(4-fluorophenyl)methyl]-1,4-diazepan-1-yl}methyl)-1,5-dimethyl-1H-pyrrole-2-carbonitrile
4-(6-aminopyridine-3-carbonyl)-9-(cyclopropylmethyl)-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
2-(dimethyl-1,2-oxazol-4-yl)-1-{9-[2-(4-methyl-1,3-thiazol-5-yl)ethoxy]-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl}ethan-1-one
N-(1H-imidazol-2-ylmethyl)-3-(4-methoxypiperidine-1-carbonyl)benzene-1-sulfonamide
({5-[1-(1-benzofuran-2-ylmethyl)piperidin-4-yl]-4-ethyl-4H-1,2,4-triazol-3-yl}methyl)dimethylamine
N-(1-carbamoylcyclopentyl)-2-methyl-1H-1,3-benzodiazole-5-carboxamide
4-[(2R)-2-amino-3-methoxypropanoyl]-1-(4-methylphenyl)piperazin-2-one
8-methyl-N-[(3-methylpyridin-4-yl)methyl]-2-propyl-2,8-diazaspiro[4.5]decane-3-carboxamide
N-(2-{3-[benzyl(methyl)amino]piperidine-1-carbonyl}thiophen-3-yl)acetamide
1-(2-chloro-4-fluorophenyl)-3-{[1-(3-methoxypropyl)pyrrolidin-3-yl]methyl}urea
1-{9-methoxy-5H,6H-benzo[h]quinazolin-2-yl}-5-methyl-N-[2-methyl-2-(morpholin-4-yl)propyl]-1H-pyrazole-4-carboxamide
3-{3-[(dimethylamino)methyl]-3-hydroxypyrrolidine-1-carbonyl}-6-ethyl-1,5-dimethyl-1,2-dihydropyridin-2-one
1-(2-{[cyclohexyl(methyl)amino]methyl}phenyl)-3-{[(2S,4S)-4-fluoropyrrolidin-2-yl]methyl}urea
1-cyclopentyl-3-methyl-4-{2-[(propan-2-yl)amino]pyrimidin-5-yl}-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
N-[3-(5-cyclopropyl-1H-pyrazol-1-yl)propyl]-5,7-dimethylpyrido[2,3-d]pyrimidin-4-amine
3-chloro-6-[3-(4-methoxy-3,5-dimethylbenzoyl)piperidin-1-yl]pyridazine
1-cyclopentyl-4-[(4-fluoro-3-methylphenyl)methyl]-1,4-diazepane
1-(furan-3-carbonyl)-3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine
4-(3-tert-butyl-1H-pyrazol-1-yl)-1-(9H-purin-6-yl)piperidine-4-carboxylic acid
2-(4-ethylphenyl)-1-[3-(1H-imidazol-1-yl)propyl]-1H-imidazole
2-[4-({methyl[2-(pyridin-2-yl)ethyl]amino}methyl)phenyl]-6-(pyridin-3-yl)-3,4-dihydropyrimidin-4-one
3-(3-hydroxy-1,2-oxazol-5-yl)-1-[3-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]propan-1-one
ethyl 1-(4-methyl-1,3-oxazole-5-carbonyl)-3-(2-phenylethyl)piperidine-3-carboxylate
1-{4H-thieno[3,2-b]pyrrole-5-carbonyl}-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
4-{[(1R,3S)-1,3-dihydroxy-7-azaspiro[3.5]nonan-7-yl]methyl}-N-methylbenzene-1-sulfonamide
4-(1,3-dimethyl-1H-pyrazole-5-carbonyl)-1-[(4-fluorophenyl)methyl]-2-(propan-2-yl)-1,4-diazepane
N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-3-(2-methylphenyl)-3-phenylpropanamide
N-{[4-(3-fluorophenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}-5-oxo-2,5-dihydro-1H-pyrazole-3-carboxamide
N-{[2-(dimethylamino)-7-methylquinolin-3-yl]methyl}-N-[2-(4-fluorophenyl)ethyl]pent-4-enamide