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3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]-1-(5-propyl-1,2-oxazole-3-carbonyl)piperidine
2-{2-[1-(1-phenylethyl)-1H-1,3-benzodiazol-2-yl]-1H-imidazol-1-yl}ethan-1-ol
(3aS,6aR)-3-[2-(4-fluorophenyl)ethyl]-5-{[5-(hydroxymethyl)furan-2-yl]methyl}-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
N-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]-3-(1H-pyrazol-1-ylmethyl)benzamide
1-(6-chloro-1,3-benzothiazol-2-yl)-N-[2-(pyridin-4-yl)ethyl]piperidin-4-amine
1-cyclohexyl-3-(cyclopropylmethyl)-N-ethyl-N-methyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
N-(3-chloro-4-propanamidophenyl)-3-(2-ethyl-1H-imidazol-1-yl)propanamide
N-(5-methyl-1,2-oxazol-3-yl)-2-(pyridazine-3-carbonyl)-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
5-(2-chlorophenyl)-N-[2-(3-methyl-1H-pyrazol-1-yl)ethyl]furan-2-carboxamide
5-methanesulfonyl-N-(6-methoxy-1,2,3,4-tetrahydronaphthalen-1-yl)-2-methylpyrimidin-4-amine
4-[2-(2H-1,3-benzodioxol-5-yloxy)acetyl]-5-methyl-1-phenylpiperazin-2-one
5-{2-[(3S,4R)-3-(dimethylamino)-4-(4-methylphenyl)pyrrolidin-1-yl]-2-oxoethyl}-2,6-dimethyl-3,4-dihydropyrimidin-4-one
(4aS,8aR)-1-[3-(1H-imidazol-1-yl)propyl]-6-(1,3-oxazole-4-carbonyl)-decahydro-1,6-naphthyridin-2-one
2-(2H-1,3-benzodioxol-5-yl)-N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]acetamide
N-{[2-fluoro-4-(trifluoromethyl)phenyl]methyl}-3-(1-methyl-1H-pyrazol-4-yl)propanamide
4-(3-methoxybenzenesulfonyl)-2-(trifluoromethyl)morpholine
2,6-dimethyl-4-({[(4-oxo-3,4-dihydroquinazolin-2-yl)methyl]amino}methyl)phenyl acetate
2-[(1S,5R)-6-{[2-(cyclopentyloxy)phenyl]methyl}-3,6-diazabicyclo[3.2.2]nonan-3-yl]-N,N-dimethylacetamide
1-(1-benzylpyrrolidine-2-carbonyl)-4-[(3-fluorophenyl)methyl]piperazine
N-[2-(dimethylamino)ethyl]-N-(oxolan-2-ylmethyl)-3-phenyl-1H-pyrazole-4-carboxamide
N-(3,4-dihydro-2H-1,5-benzodioxepin-7-ylmethyl)-1-(propan-2-yl)-1H-pyrazole-4-carboxamide
N-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-2,8-dimethyl-N-(propan-2-yl)quinoline-4-carboxamide
2-[4-(dimethylamino)-6-oxo-1,6-dihydropyridazin-1-yl]-N-[2-(furan-2-yl)-2-(pyrrolidin-1-yl)ethyl]acetamide
{1-[1-(3,6-dimethylpyrazin-2-yl)piperidin-4-yl]ethyl}dimethylamine
2-[1-(propan-2-yl)-1H-imidazol-2-yl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
{[2-(1H-imidazol-1-yl)pyridin-3-yl]methyl}({[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl})amine
3-(1,2-oxazinan-2-yl)-1-[3-(pyridin-2-ylmethoxy)piperidin-1-yl]propan-1-one
4,4,4-trifluoro-1-[4-(naphthalen-2-yl)piperazin-1-yl]butan-1-one
3-(3-methylphenyl)-N-[(4-sulfamoylphenyl)methyl]-1H-pyrazole-4-carboxamide
N-{[1-(ethoxymethyl)cyclopropyl]methyl}-3-(4-hydroxyphenyl)benzamide
(2S,4R)-4-amino-N,N-diethyl-1-[1-methyl-3-(thiophen-2-yl)-1H-pyrazole-5-carbonyl]pyrrolidine-2-carboxamide
(1S,5R)-6-[(5-ethylpyridin-2-yl)methyl]-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
N-{[1-(1H-imidazol-1-ylmethyl)cyclopropyl]methyl}-4-(4-oxo-3,4-dihydroquinazolin-3-yl)butanamide
N-[(2-fluorophenyl)methyl]-2-[8-(2-methoxyethyl)-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl]acetamide
1-methyl-3-[4-(2-methylphenyl)-1,4-diazepane-1-carbonyl]-1H-indole
(1R,5R)-3-[3-(3-methoxyphenyl)-1H-pyrazole-5-carbonyl]-6-propyl-3,6-diazabicyclo[3.2.2]nonane
N-methyl-2-(2-{1-[(4-methylphenyl)methyl]-3-oxopiperazin-2-yl}acetamido)acetamide
3-[(3R,4S)-1-[(1-methyl-1H-indol-4-yl)methyl]-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propanoic acid
1-[5-(2-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-yl]-4-(2-methoxyethyl)piperazine
ethyl 2-{[3-(3-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl]amino}acetate
1-(cyclopropylmethyl)-3-hydroxy-3-({[(4-methyl-1,3-thiazol-2-yl)methyl]amino}methyl)piperidin-2-one
4-ethyl-5-[3-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidine-1-carbonyl]-1,3-thiazol-2-amine
4-[3-(4-ethyl-1-methyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)piperidine-1-carbonyl]-1,2-dihydrophthalazin-1-one
2-(4-{[3-(cyclopentyloxy)phenyl]methyl}-1-(thiophen-2-ylmethyl)piperazin-2-yl)ethan-1-ol
{1-[(2,3-difluoro-4-methoxyphenyl)methyl]-3-ethylpiperidin-3-yl}methanol
4-(1H-indol-3-yl)-1-[(1R,5R)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]butan-1-one
1-(2H-1,3-benzodioxol-5-ylmethyl)-3-(2-oxo-2-{4H,5H,6H,7H-thieno[3,2-c]pyridin-5-yl}ethyl)-3-phenylpyrrolidine-2,5-dione
5-(1-methyl-1H-pyrazol-4-yl)-3-[3-(pyridin-2-ylmethoxy)piperidin-1-yl]pyrazin-2-amine
2-{4-[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl]-1-[(5-methylfuran-2-yl)methyl]piperazin-2-yl}ethan-1-ol
N-{[3-(benzyloxy)phenyl]methyl}-4-hydroxy-2-methylpyrimidine-5-carboxamide