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3-cyclopropyl-N-(pyridin-3-yl)-1H-pyrazole-5-carboxamide
1-{3-[5-(hydroxymethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-(methylsulfanyl)ethan-1-one
N-(2-{4H,5H,6H-cyclopenta[d][1,3]thiazol-2-yl}ethyl)-3-(trimethyl-1H-pyrazol-4-yl)propanamide
[(1R,2R,4R)-bicyclo[2.2.1]hept-5-en-2-ylmethyl](methyl){[3-(1H-1,2,3,4-tetrazol-5-yl)phenyl]methyl}amine
2-ethyl-4-[1-methyl-3-(trifluoromethyl)-1H-pyrazole-5-carbonyl]-1-(propan-2-yl)piperazine
2-(4-chlorophenyl)-5-{1-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-1H-imidazol-2-yl}pyrimidine
N,1,3-trimethyl-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-6-(pyridin-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
6-[(3S,4S)-3-(dimethylamino)-4-hydroxypyrrolidin-1-yl]-N-[(4-ethyl-1,3-thiazol-2-yl)methyl]pyridine-3-carboxamide
3-[4-(5-cyanopyridin-2-yl)piperazine-1-carbonyl]piperidine-1-carboxamide
2-methoxy-2-methyl-1-{3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}propan-1-one
N-[2-(cyclohex-1-en-1-yl)ethyl]-2-(3-oxo-1-{[2-(trifluoromethyl)phenyl]methyl}piperazin-2-yl)acetamide
1-{4-[4-ethyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-4-methylpentan-1-one
2-{[3-ethyl-4-(propan-2-yl)piperazin-1-yl]methyl}-3,5-dimethoxybenzoic acid
1-methyl-8-{[4-(2-methylphenyl)phenyl]methyl}-3-[3-(pyridin-4-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-(isoquinolin-5-ylmethyl)-N-methyl-4-(pyridin-3-yl)pyrimidin-2-amine
8-methyl-3-(2-methylpropyl)-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[2-(2-chlorophenyl)-2-(dimethylamino)ethyl]-3-(3,5-dimethyl-1H-pyrazol-4-yl)propanamide
N-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-N-methyl-4-(4H-1,2,4-triazol-4-yl)benzamide
N-[(3S,4R)-1-({4-[(dimethylamino)methyl]thiophen-2-yl}methyl)-4-(4-methylphenyl)pyrrolidin-3-yl]acetamide
4-{4-[(3,3-dimethylpyrrolidin-1-yl)methyl]-1H-1,2,3-triazol-1-yl}-1-[(2E)-2-methylpent-2-en-1-yl]piperidine
4-(3,5-dimethyl-1H-pyrazol-1-yl)-N-[1-(4-methyl-1H-imidazol-2-yl)propyl]benzamide
4-[1-({3-methoxy-2-[(2-methylprop-2-en-1-yl)oxy]phenyl}methyl)pyrrolidin-2-yl]-3,5-dimethyl-1,2-oxazole
N-(cyclohex-1-en-1-ylmethyl)-4-(pyrrolidin-1-ylmethyl)benzamide
2,3-dimethyl-N-[2-(3-{[methyl(thiophen-3-ylmethyl)amino]methyl}phenoxy)propyl]-1H-indole-5-carboxamide
1-cyclobutanecarbonyl-4-[1-methyl-3-(trifluoromethyl)-1H-pyrazole-5-carbonyl]-1,4-diazepane
(2S)-N-ethyl-1-[3-(3-hydroxy-3-methylbutyl)benzoyl]pyrrolidine-2-carboxamide
4-[(4-{6-oxo-4-[2-(1H-pyrazol-1-yl)ethyl]-1,6-dihydropyrimidin-2-yl}phenyl)methyl]-1,4-diazepan-2-one
(2R)-2-amino-3-methyl-1-{4-[2-methyl-6-(morpholin-4-yl)pyrimidin-4-yl]piperidin-1-yl}butan-1-one
N-[cyclopropyl(4-methylpyridin-2-yl)methyl]pyrazolo[1,5-a]pyridine-7-carboxamide
N-[(2S)-2-aminopropyl]-1-methyl-2-oxo-6-(propan-2-yl)-1,2-dihydropyridine-3-carboxamide
(1S,6R)-9-({3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)-3,9-diazabicyclo[4.2.1]nonan-4-one
3-[(2,4-difluorophenyl)methyl]-5-(1-methyl-1H-imidazol-2-yl)-1,2,4-oxadiazole
5-(dimethylamino)-1-methyl-N-(thiophen-2-ylmethyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
2-(cyclopropylmethyl)-8-[4-(4-fluorophenyl)-4-oxobutyl]-2,8-diazaspiro[5.5]undecan-3-one
(4aS,8aR)-6-(furan-2-carbonyl)-1-[2-(1H-imidazol-4-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
1-[2-(azepan-1-yl)ethyl]-3-(3-cyano-4-methoxyphenyl)-1-methylurea
3,5-dimethyl-N-{[1-(pyridin-2-yl)piperidin-3-yl]methyl}-1H-indole-2-carboxamide
{2-[({1-[(2-methoxyphenyl)methyl]piperidin-3-yl}methyl)(1,3-thiazol-2-ylmethyl)amino]ethyl}dimethylamine
6-ethyl-2-methyl-N-{[1-methyl-2-(methylsulfanyl)-1H-imidazol-5-yl]methyl}quinoline-4-carboxamide
N5-(2,6-dimethoxypyridin-3-yl)-1-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3,5-dicarboxamide
1-{3-[5-(2-methoxy-4-methylphenyl)-4-phenyl-1H-imidazol-1-yl]piperidin-1-yl}ethan-1-one
N-ethyl-4-methyl-5-[3-(2-phenylethyl)piperidine-1-carbonyl]-1,3-thiazol-2-amine
1-(2-methoxyethyl)-4-[3-(5-methylfuran-2-yl)benzoyl]piperazine
(1-{1-[1-(2-ethoxyethyl)-3-methyl-1H-pyrazole-5-carbonyl]piperidin-4-yl}ethyl)dimethylamine
1-tert-butyl-3-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}-1H-pyrrole
5-(but-3-en-1-yl)-3-cyclopropyl-1-phenyl-1H-1,2,4-triazole
3-[(3R,4S)-1-(1H-1,3-benzodiazol-2-ylmethyl)-4-(morpholin-4-yl)piperidin-3-yl]propanoic acid
3-(2-oxoazepan-3-yl)-3,4-dihydroquinazolin-4-one
4-ethyl-1-(2-phenylpropyl)-1,4-diazepan-5-one
(2-methoxyethyl)[(1-methyl-1H-pyrazol-4-yl)methyl]{[1-(propan-2-yl)piperidin-4-yl]methyl}amine