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5-chloro-2-{4-[2-methyl-2-(piperidin-1-yl)propyl]piperazin-1-yl}pyrimidine
N-[(1S,2R)-2-aminocyclobutyl]-4-tert-butylbenzene-1-sulfonamide
N-[3-ethyl-4-(4-fluorophenyl)-1-methyl-1H-pyrazol-5-yl]morpholine-4-carboxamide
N-(3-methyl-2-oxo-2,3-dihydro-1,3-benzoxazol-5-yl)-2-(pyridin-3-yl)piperidine-1-carboxamide
N3-methyl-N3-(2-methylpropyl)-4-oxo-1-(propan-2-yl)-N5-[2-(thiophen-2-yl)ethyl]-1,4-dihydropyridine-3,5-dicarboxamide
N-(3-hydroxy-3-phenylpropyl)-N-methyl-2-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
4-({5-[1-(4-fluorophenyl)-2,2-dimethylcyclopropyl]-1,2,4-oxadiazol-3-yl}methyl)morpholine
1-(2-chlorophenyl)-5-(1H-imidazol-1-ylmethyl)-3-(2-methylpropyl)-1H-1,2,4-triazole
methyl 9-[(1-methyl-5-oxopyrrolidin-3-yl)methoxy]-3-[2-(3-methylphenyl)acetyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
3-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-1-(4-ethoxy-2-fluorophenyl)-3-methylurea
1-(azepan-1-yl)-4-[3-(1-methoxypropan-2-yl)-3H-imidazo[4,5-b]pyridin-2-yl]butan-1-one
N,3-dimethyl-4-oxo-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-3,4-dihydroquinazoline-7-carboxamide
1-(2-oxo-2,3-dihydro-1H-indol-5-yl)-3-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}urea
5-ethyl-N-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-amine
2-{4-[(3,5-dimethyl-1H-indol-2-yl)methyl]-1-(1-methylpiperidin-4-yl)piperazin-2-yl}ethan-1-ol
4-[2-(5-ethyl-1-benzofuran-3-yl)acetyl]-1λ6-thiomorpholine-1,1-dione
(1R,5R)-N,N-dimethyl-6-({6-methylimidazo[1,2-a]pyridin-2-yl}methyl)-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
2-chloro-N-{[5-(3,6-dimethylpyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-6-fluorobenzamide
2-(2-{1,2-dihydrospiro[indole-3,4'-piperidine]-1'-ylmethyl}phenoxy)acetic acid
[1-(4,6-dimethylpyridine-3-carbonyl)-3-(2-methoxyethyl)piperidin-3-yl]methanol
({5-[1-benzyl-3-(1H-1,2,4-triazol-1-ylmethyl)-1H-1,2,4-triazol-5-yl]furan-2-yl}methyl)dimethylamine
4-(4-chlorophenyl)-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]butanamide
N-{1,9-dioxaspiro[5.5]undecan-4-yl}-1H-1,2,3-benzotriazole-5-carboxamide
3-(4-benzoylpiperazine-1-carbonyl)-2-methyl-4,5,6,7-tetrahydro-1H-indol-4-one
N-[5-(2-chloro-4-fluorophenyl)pyridin-2-yl]acetamide
2-[(3,5-difluorophenyl)methyl]-8-(3-fluoropropyl)-2,8-diazaspiro[4.5]decan-3-one
2-methoxy-5-oxo-6-[4-(pyridin-2-yl)butyl]-5,6-dihydro-1,6-naphthyridine-3-carbonitrile
3-(1-{[2-(2,4-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-2-yl)propan-1-ol
3,5-dimethyl-4-[5-(thiophene-2-sulfonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl]-1,2-oxazole
(3S,4S)-4-cyclopropyl-1-{5-[(methylsulfanyl)methyl]furan-2-carbonyl}pyrrolidine-3-carboxylic acid
1-{1-[2-(3,4-dihydro-2H-1,4-benzoxazin-4-yl)-2-oxoethyl]piperidin-4-yl}pyrrolidin-2-one
2-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-N-(3-hydroxy-2,2-dimethylpropyl)-2,3-dihydro-1H-indene-2-carboxamide
5-{4-[(2-methylphenyl)methyl]piperazine-1-carbonyl}-4-phenylpyrimidin-2-amine
N-[(3-ethyl-4,5-dihydro-1,2-oxazol-5-yl)methyl]-4-{[1-(2-methoxyacetyl)piperidin-4-yl]oxy}benzamide
N-[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2,4,6-tetraen-3-amine
8-{6-methyl-2H-[1,3]dioxolo[4,5-g]quinolin-8-yl}-2,8-diazaspiro[4.5]decan-3-one
N-[3-(3-methoxyphenyl)phenyl]-1-[2-(1H-1,2,4-triazol-1-yl)acetyl]piperidine-2-carboxamide
3-{[1-benzyl-3-(5-methylfuran-2-yl)-1H-1,2,4-triazol-5-yl]methyl}-1λ6-thiolane-1,1-dione
2-(1-{1-[(6-chloro-2H-chromen-3-yl)methyl]piperidin-4-yl}-1H-1,2,3-triazol-4-yl)ethan-1-ol
1-{2-[2-(3-chlorophenyl)ethyl]-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl}-N-(pyridin-4-ylmethyl)piperidine-4-carboxamide
(3aR,6aR)-2-[2-(3-chlorophenyl)acetyl]-5-methanesulfonyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-{5-cyclopropyl-1-[4-(thiophen-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carbonyl}-N,N-dimethylpyrrolidin-3-amine
1-({[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl](methyl)carbamoyl}methyl)piperidine-4-carboxamide
N-[1-(2,3-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3-methylbut-2-enamide
(3R,4R)-1-{[2-(methoxymethyl)pyrimidin-5-yl]methyl}-3-methyl-4-(oxan-4-yl)piperidin-4-ol
(3S,4S)-4-(morpholin-4-yl)-1-(4-phenyl-1H-imidazole-5-carbonyl)pyrrolidin-3-ol
N-[(2-ethoxypyridin-3-yl)methyl]-2-(phenylamino)pyrimidine-5-carboxamide
1-(1-ethyl-1H-pyrazole-5-carbonyl)spiro[azepane-4,2'-chromene]
2-(morpholin-3-yl)-N-[2-(6-oxo-3-phenyl-1,6-dihydropyridazin-1-yl)ethyl]acetamide
2-[4-(2,6-dimethoxy-4-methylphenyl)phenyl]-N,N-dimethylacetamide