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N-benzyl-4-(4-phenyl-1H-1,2,3-triazol-1-yl)piperidine-1-carboxamide
1-[(4aR,8aR)-7-{[3-fluoro-4-(trifluoromethyl)phenyl]methyl}-4a-hydroxy-decahydro-2,7-naphthyridin-2-yl]ethan-1-one
1-[1-(2-aminopyridine-4-carbonyl)piperidin-4-yl]piperidin-4-ol
4-[(2,4-difluorophenyl)methyl]-9-methoxy-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
4-(1-{[1-butyl-2-(ethanesulfonyl)-1H-imidazol-5-yl]methyl}piperidin-4-yl)pyridine
1-(2-methyl-1,3-thiazole-4-carbonyl)-3-{2-[2-(trifluoromethyl)phenyl]ethyl}piperidine
N-{[2-(2,6-dimethylphenoxy)pyridin-3-yl]methyl}-1,2,3-thiadiazole-4-carboxamide
1-(1-methylpiperidine-2-carbonyl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
2-(1-benzyl-3-oxopiperazin-2-yl)-N-(1-methanesulfonylpiperidin-4-yl)acetamide
[4-(3-methyl-1-propyl-1H-pyrazole-4-carbonyl)morpholin-3-yl]methanol
N-[(3R,4R)-3-hydroxy-1-[3-(hydroxymethyl)quinolin-2-yl]piperidin-4-yl]pyrazine-2-carboxamide
N'-[2-(4-cyclopentylmorpholin-2-yl)ethyl]-N-(propan-2-yl)ethanediamide
N-(4-{3-methyl-1-[(3-methylphenyl)methyl]-6-oxo-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-4-yl}phenyl)acetamide
6-[1-tert-butyl-3-(oxan-4-yl)-1H-1,2,4-triazol-5-yl]pyridin-2-amine
2-(2,5-dimethoxyphenyl)-N-{[4-(4-fluorophenyl)-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}acetamide
(3R,5S)-N-(2-hydroxyethyl)-1-(pyridin-4-ylmethyl)-5-[3-(trifluoromethyl)phenoxymethyl]piperidine-3-carboxamide
2-(2-aminoethyl)-N-[3,3-dimethyl-1-(pyridin-3-yl)butyl]quinazolin-4-amine
[(3R,4R)-4-[(dimethylamino)methyl]-1-[(2-ethoxynaphthalen-1-yl)methyl]pyrrolidin-3-yl]methanol
3-(3,5-dimethoxyphenyl)-4-methylpyridine
N-(6-chloropyridin-3-yl)-4-(2-methylpyrimidin-4-yl)piperidine-1-carboxamide
2-phenyl-1-{1-[4-(pyridin-2-yl)pyrimidin-2-yl]piperidin-4-yl}ethan-1-ol
1-methyl-3-{[1-(5-methyl-1,3-oxazole-4-carbonyl)piperidin-4-yl]methyl}-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
2-({1-[1-(2-fluorophenyl)-2,2-dimethylcyclopropanecarbonyl]piperidin-4-yl}oxy)pyrimidine
5-[4-(cyclopropylmethyl)-3-(propan-2-yl)-1,4-diazepane-1-carbonyl]quinoxaline
N,N-dimethyl-1-{6-[3-(trifluoromethyl)phenyl]imidazo[2,1-b][1,3]thiazole-3-carbonyl}pyrrolidin-3-amine
N-(1-benzylpyrrolidin-3-yl)-3-{1-[(3,4-difluorophenyl)methyl]piperidin-4-yl}propanamide
1-{4-[(4-chloro-3-fluorophenyl)methyl]-6-hydroxy-1,4-diazepan-1-yl}ethan-1-one
(1R,3R,5S)-8-(1-ethyl-5-methyl-1H-pyrazole-3-carbonyl)-3-(4-methoxyphenyl)-8-azabicyclo[3.2.1]octane
N-cyclopropyl-1-(2-ethoxyethyl)-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
[1-(dimethyl-1,3-thiazol-4-yl)ethyl]({4-[2-(1H-imidazol-1-yl)ethoxy]phenyl}methyl)methylamine
3-[2-methoxy-1-(1-methyl-1H-pyrazol-5-yl)ethyl]-1-(5-methyl-2,1,3-benzothiadiazol-4-yl)urea
1-[2-ethoxy-5-(trifluoromethyl)phenyl]-3-[(3S,4R)-4-hydroxyoxolan-3-yl]-3-methylurea
{1-[1-(1,2-oxazol-3-ylmethyl)piperidin-3-yl]piperidin-4-yl}methanol
2-{1-[(4-ethoxyphenyl)methyl]-4-[(1-methyl-1H-indol-3-yl)methyl]piperazin-2-yl}ethan-1-ol
2-(8-methoxyquinolin-2-yl)benzonitrile
1-[3-chloro-4-(1H-1,2,4-triazol-1-yl)phenyl]-3-{3-[2-(propan-2-yl)-1H-imidazol-1-yl]propyl}urea
4-[4-(4,4-difluoropiperidin-1-yl)piperidin-1-yl]-6-ethyl-2-(pyrrolidin-1-yl)pyrimidine
2-(ethylamino)-N-[(3-phenyl-1H-1,2,4-triazol-5-yl)methyl]pyrimidine-5-carboxamide
4-[4-(4-fluorophenyl)-1H-1,2,3-triazol-1-yl]-1-(1,3-thiazole-4-carbonyl)piperidine
6-(2-fluoro-4-methoxyphenyl)-N,N-dimethyl-7-(3-methylbut-2-en-1-yl)-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
(3aS,6aS)-2-cyclobutanecarbonyl-5-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-[(2-fluoro-5-methoxyphenyl)methyl]-3-hydroxy-3-({[2-(pyridin-4-yl)ethyl]amino}methyl)piperidin-2-one
(1S,5R)-3-methyl-6-[(6-methyl-2H-1,3-benzodioxol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
N-ethyl-5-{4-[(3-fluorophenyl)methyl]piperazine-1-carbonyl}pyrimidin-2-amine
2-[6-(cyclopentylamino)-1H-pyrrolo[2,3-b]pyridin-4-yl]benzamide
1-{3,6-dimethyl-[1,2]oxazolo[5,4-b]pyridine-4-carbonyl}-3-[(dimethylamino)methyl]pyrrolidin-3-ol
(2S,4S)-4-amino-1-[(4Z)-hept-4-en-1-yl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
3-({cyclopropyl[(1-methyl-1H-pyrazol-4-yl)methyl]amino}methyl)-7-(methylsulfanyl)-1,2-dihydroquinolin-2-one
N-ethyl-4-[(5-methyl-1H-1,2,3,4-tetrazol-1-yl)methyl]-N-[2-(4-methyl-1H-1,3-benzodiazol-2-yl)ethyl]benzamide
7-(3-methoxyphenyl)-2-(1-methyl-1H-1,3-benzodiazol-2-yl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one