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{2-[4-(1-hydroxy-3-phenylpropyl)piperidin-1-yl]-2-oxoethyl}urea
1-{2-[(2-methylprop-2-en-1-yl)oxy]phenyl}-3-{[2-(morpholin-4-yl)-1,3-thiazol-4-yl]methyl}urea
[(3R,4R)-4-[(dimethylamino)methyl]-1-{[2-(5-methylfuran-2-yl)phenyl]methyl}pyrrolidin-3-yl]methanol
2-methoxy-N,N-dimethyl-5-({methyl[2-(phenylsulfanyl)ethyl]carbamoyl}amino)benzamide
[(3S,4S)-4-(hydroxymethyl)-1-{[4-(methylsulfanyl)phenyl]methyl}pyrrolidin-3-yl]methanol
1-[3-chloro-2-(propan-2-yloxy)phenyl]-3-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)ethyl]urea
6-(diethylamino)-N-[2-(1-methylpiperidin-2-yl)ethyl]pyridine-3-carboxamide
N-cyclopropyl-2-[4-({[(3R,4R)-4-(pyrrolidin-1-yl)oxolan-3-yl]carbamoyl}amino)phenyl]acetamide
6-methyl-2-({2-[5-(oxolan-3-yl)-4-phenyl-1H-imidazol-1-yl]ethyl}amino)-3,4-dihydropyrimidin-4-one
N-(1-{1-[3-(2H-1,3-benzodioxol-5-yl)-2-methylpropyl]piperidin-4-yl}-1H-pyrazol-5-yl)-2,2-dimethylpropanamide
3-{5-oxo-3-[(trimethyl-1H-pyrazol-1-yl)methyl]-4,5-dihydro-1H-1,2,4-triazol-4-yl}propanoic acid
methyl (2S,4R)-4-(2,2-diphenylacetamido)-1-[(4-hydroxyphenyl)methyl]pyrrolidine-2-carboxylate
{1-methyl-5-[2-methyl-2-(morpholin-4-yl)propyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl}methanol
N-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-2-{1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-3-oxopiperazin-2-yl}acetamide
4-phenyl-1-[4-(1H-pyrazol-3-yl)benzoyl]piperidine-4-carbonitrile
N-{5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl}-3-[5-(thiophen-2-yl)furan-2-yl]propanamide
N-[(1S,3aS,6aS)-octahydropentalen-1-yl]-3-(3-methoxyphenyl)-1H-pyrazole-4-carboxamide
2-(2-methoxyphenoxy)-N-[(1-{[2-(5-methylfuran-2-yl)phenyl]methyl}piperidin-3-yl)methyl]acetamide
N-{4-[(3S)-3-acetamidopyrrolidine-1-carbonyl]phenyl}cyclobutanecarboxamide
N4,N4-diethyl-N2-[(5-methylpyrazin-2-yl)methyl]morpholine-2,4-dicarboxamide
N-(2-{imidazo[1,2-a]pyrimidin-2-yl}ethyl)-2-{1-[(5-methylfuran-2-yl)methyl]-3-oxopiperazin-2-yl}acetamide
2-(2-fluorophenoxymethyl)-N-methyl-N-[(1-methylpiperidin-2-yl)methyl]-1,3-oxazole-4-carboxamide
dimethyl(1-{3-[5-(2-methylpropyl)-1H-1,2,4-triazol-3-yl]phenyl}ethyl)amine
N-ethyl-2-methyl-N-[2-(4-methylbenzenesulfonyl)ethyl]-1-benzofuran-5-carboxamide
1-{1-[2-(4-chlorophenoxy)acetyl]piperidin-4-yl}-N-cyclopropylpiperidine-4-carboxamide
N-[(1-methylpiperidin-3-yl)methyl]-4-propylbenzamide
1-{1-[1-(1-ethyl-1H-pyrazole-5-carbonyl)piperidin-4-yl]ethyl}-4-methylpiperazine
1-(cyclohexylmethyl)-N-[3-(pyridin-3-yl)propyl]-1H-1,2,3-triazole-4-carboxamide
8-acetyl-2-(4-chloro-2-methylbenzoyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-5-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-1,2-oxazole-3-carboxamide
1-(2H-1,3-benzodioxol-4-ylmethyl)-3-(2,5-dimethoxyphenyl)pyrrolidine
1-(carbamoylmethyl)-N-({2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}methyl)piperidine-3-carboxamide
N-cyclopropyl-2-[3-(6-methoxynaphthalene-2-carbonyl)piperidin-1-yl]acetamide
4-[1-(propan-2-yl)-1H-imidazol-2-yl]-1-(5-propyl-1,3,4-thiadiazol-2-yl)piperidine
(1R,3S)-3-methoxy-7-(4-methyl-1,3-oxazole-5-carbonyl)-7-azaspiro[3.5]nonan-1-ol
5-(2-ethylpiperidine-1-carbonyl)-N-[(4-methylphenyl)methyl]-4-oxo-1-[2-(pyridin-2-yl)ethyl]-1,4-dihydropyridine-3-carboxamide
5-[(diethylcarbamoyl)methyl]-N-(2-methoxyethyl)-1-(3-methylbutyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
6-[4-(4-hydroxypiperidin-1-yl)piperidine-1-carbonyl]-4-methyl-1H,2H,3H-pyrazolo[3,4-b]pyridin-3-one
phenyl (7R,9aR)-7-[(benzylsulfanyl)methyl]-6,9-dioxo-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxylate
3-(2-methoxyphenyl)-1-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl}propan-1-one
3-ethyl-4-[3-(4-phenylphenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl]-1H-pyrazole
6-methyl-5-phenyl-2-[4-(thiomorpholin-4-ylmethyl)phenyl]-3,4-dihydropyrimidin-4-one
N-[(3S,4R)-4-(4-methylphenyl)-1-(4-propyl-1,2,3-thiadiazole-5-carbonyl)pyrrolidin-3-yl]acetamide
N-[(3-methyl-1-benzofuran-2-yl)methyl]-2-[2-(propan-2-yl)-1H-imidazol-1-yl]propanamide
3-({3-azaspiro[5.5]undecan-9-yl}amino)-N-(1,3-thiazol-2-yl)propanamide
(3S,4R)-3-ethyl-1-(5-ethyl-2-methylpyrimidin-4-yl)-4-methylpiperidin-4-ol
N-[(4-ethyl-1,3-thiazol-2-yl)methyl]-6-{[1-(1-methyl-1H-pyrazol-4-yl)ethyl]amino}pyridine-3-carboxamide
{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}(methyl){[1-(propan-2-yl)-1H-imidazol-2-yl]methyl}amine
1-(6-methoxy-2,3-dihydro-1H-indene-5-carbonyl)-3-(2-methoxyphenoxy)azetidine
1-({1-ethyl-3-[(2-methoxyphenyl)methyl]-1H-1,2,4-triazol-5-yl}methyl)-4,6-dimethyl-1,2-dihydropyrimidin-2-one