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N,N-dimethyl-2-{2-methyl-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}acetamide
N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-3-(1H-pyrazol-1-yl)propanamide
8-(2-amino-4-ethyl-1,3-thiazole-5-carbonyl)-2-cyclopentyl-2,8-diazaspiro[5.5]undecan-3-one
7-methyl-2-[2-(pyridin-3-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
3-{6-hydroxy-4-[(3-phenyl-1H-pyrazol-4-yl)methyl]-1,4-diazepan-1-yl}propanoic acid
N-[2-hydroxy-3-(3-methoxyphenoxy)propyl]-5-(propan-2-yl)-1,3-oxazole-4-carboxamide
N-methyl-N-{[2-(methylamino)pyrimidin-5-yl]methyl}-2-oxo-6-phenyl-1,2-dihydropyridine-3-carboxamide
2-(2-methoxyethyl)-8-[5-(methoxymethyl)thiophene-2-carbonyl]-2,8-diazaspiro[5.5]undecan-3-one
1-[(4-phenyl-1,3-thiazol-2-yl)methyl]-3-(pyrrolidin-1-yl)piperidine
4-({1-[3-(5-methylfuran-2-yl)benzoyl]piperidin-4-yl}methyl)morpholine
5-{3-[2-(2,4-difluorophenyl)ethyl]piperidine-1-carbonyl}-2-methylphenol
1-[4-(cyclopropylamino)-2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl]-3-(1H-1,2,3,4-tetrazol-1-yl)propan-1-one
3-(3-hydroxyquinoxalin-2-yl)-1-(4-methanesulfonylpiperazin-1-yl)propan-1-one
{[2-(naphthalen-2-yl)pyrimidin-5-yl]methyl}[2-(4,5,6,7-tetrahydro-2H-indazol-3-yl)ethyl]amine
N-[(8-methoxyquinolin-5-yl)methyl]-N-methyl-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide
2-(5-fluoro-2-methylphenyl)-4,6-dimethoxy-1,3,5-triazine
ethyl (2S)-2-[(3-propanamidophenyl)formamido]propanoate
N3-(1-benzylpiperidin-4-yl)-1-(cyclohexylmethyl)-4-oxo-N5-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
2-(4-methoxyphenyl)-1-{4-[2-methyl-5-(trifluoromethyl)-1H-1,3-benzodiazol-1-yl]piperidin-1-yl}ethan-1-one
1-{4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-(1-methyl-1H-indol-3-yl)ethan-1-one
4-{[2-(4-fluorophenyl)pyrrolidin-1-yl]methyl}-5-methyl-2-(3-methylthiophen-2-yl)-1,3-oxazole
1-{4-[2-(1H-pyrazol-1-ylmethyl)-1,4-oxazepane-4-carbonyl]piperidin-1-yl}ethan-1-one
7-cyclopentyl-2-(2-methyl-1H-pyrrole-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
2,5-dimethyl-N-[(3R,5S)-1-methyl-5-(methylcarbamoyl)pyrrolidin-3-yl]-1-phenyl-1H-pyrrole-3-carboxamide
4-chloro-1-ethyl-N-[(5-methylthiophen-2-yl)methyl]-N-(prop-2-en-1-yl)-1H-pyrazole-5-carboxamide
methyl 2-[(3-carbamoyl-1,2,4-oxadiazol-5-yl)methyl]-1-oxo-1,2-dihydroisoquinoline-7-carboxylate
N-(butan-2-yl)-1-ethyl-N-(thiophen-3-ylmethyl)-1H-pyrazole-4-carboxamide
4-[(2-fluoro-4-methoxyphenyl)methyl]-7-(thiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
(2S,4R)-N-(1,1-dioxo-1λ6-thiolan-3-yl)-4-[(4-methoxyphenyl)sulfanyl]-1-{[2-(trifluoromethyl)phenyl]methyl}pyrrolidine-2-carboxamide
5-{[3-(2,5-dimethoxyphenyl)pyrrolidin-1-yl]methyl}-2-propylpyrimidine
2-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}-2,8-diazaspiro[4.5]decane-3-carboxylic acid
4-(2-butoxyacetyl)-5-methyl-1-(4-methylphenyl)piperazin-2-one
2-[4-(4-cyclohexylpiperazine-1-carbonyl)-5-(methoxymethyl)-1H-pyrazol-1-yl]-5-methyl-4-(thiophen-2-yl)pyrimidine
N-({1-[2-(4-chlorophenyl)ethyl]piperidin-3-yl}methyl)-2-acetamido-N-methylacetamide
(1S,5R)-3-[3-(3-methoxyphenyl)propanoyl]-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonan-7-one
2-[3-(3-methoxyphenoxy)azetidine-1-carbonyl]-N,N-dimethylaniline
N-(2-ethylphenyl)-1-methyl-10-oxo-1,4,9-triazaspiro[5.6]dodecane-4-carboxamide
(1R,5R)-6-benzyl-3-{imidazo[1,2-a]pyrimidine-2-carbonyl}-3,6-diazabicyclo[3.2.2]nonane
N-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)ethyl]-3-phenyl-1H-pyrazole-4-carboxamide
2-amino-3-ethyl-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-3H-imidazo[4,5-b]pyridine-6-carboxamide
2-(2,3-dihydro-1H-inden-1-yl)-1-(thiomorpholin-4-yl)ethan-1-one
N-cyclooctyl-5-(4-methylpiperidine-1-carbonyl)-4-oxo-1-(pyridin-2-ylmethyl)-1,4-dihydropyridine-3-carboxamide
2-{5-[5-(methoxymethyl)thiophen-2-yl]-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-1-yl}pyridine
4-benzyl-3-ethyl-1-[5-(propan-2-yl)pyrimidin-4-yl]-1,4-diazepan-5-one
N-{[2-(dimethylamino)-5,8-dimethoxyquinolin-3-yl]methyl}-N-(furan-2-ylmethyl)-1,3-thiazole-5-carboxamide
2-ethoxy-6-[(3-{4-[3-(trifluoromethyl)phenyl]-1H-pyrazol-5-yl}piperidin-1-yl)methyl]phenol
2-({5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)-N-methylethane-1-sulfonamide
2-(2-methoxyphenyl)-5-[(3-phenyl-1H-pyrazol-4-yl)methyl]-2,3,4,5-tetrahydro-1,5-benzothiazepin-4-one
2-[(3-ethyl-1H-1,2,4-triazol-5-yl)sulfanyl]-N-methyl-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}acetamide
5-{2-[4-(acetamidomethyl)piperidin-1-yl]pyrimidin-4-yl}-2-ethoxybenzoic acid