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2-[4-hydroxy-4-(5-methylpyridin-2-yl)piperidin-1-yl]-1,3-thiazole-4-carboxamide
1'-[(5-chlorothiophen-2-yl)methyl]-5-(2-methylpropyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
3-[3-(dimethylamino)propyl]-1-(2-phenylethyl)-8-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[3-(dimethylamino)propyl]-1-(7-fluoro-2-methylquinoline-4-carbonyl)-N-methylpiperidin-3-amine
3-phenyl-6-{4-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}pyridazine
N-benzyl-N-methyl-3-({methyl[1-(1,2-oxazol-3-yl)ethyl]amino}methyl)imidazo[1,2-a]pyridine-2-carboxamide
N-methyl-2-(5-methyl-3-oxo-2,3-dihydro-1H-pyrazol-4-yl)-N-[1-(3-methylpyridin-2-yl)propan-2-yl]acetamide
ethyl 4-[3-(piperidin-3-yl)benzamido]piperidine-1-carboxylate
5-[2-(2,4-difluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]-2-ethylpyrimidine
3,3-dimethyl-1-{4-[4-(morpholin-4-yl)phenyl]phenyl}urea
2-({[(3S,4R)-1-[(2-chloro-4-fluorophenyl)methyl]-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}(ethyl)amino)ethan-1-ol
2-{4-[(3,5-dimethoxyphenyl)methyl]-1-[(4-fluorophenyl)methyl]piperazin-2-yl}ethan-1-ol
1-[3-(butan-2-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-2-[2-(propan-2-yl)-1H-1,3-benzodiazol-1-yl]ethan-1-one
N-cyclopropyl-1-[5-(1H-pyrazol-1-ylmethyl)furan-2-carbonyl]piperazine-2-carboxamide
N-{[(2S,4S)-4-fluoropyrrolidin-2-yl]methyl}-2-[4-(trifluoromethyl)phenyl]-1,3-thiazole-4-carboxamide
2-[3-(3,4-difluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]ethan-1-ol
1-(6-chloropyridin-3-yl)-3-(3-methoxypropyl)urea
4-(3-fluorophenyl)-N-(oxolan-3-yl)benzamide
4-(3,5-dimethyl-1H-pyrazol-1-yl)-1-[3-(1-methyl-1H-imidazole-2-carbonyl)piperidin-1-yl]butan-1-one
2-(3-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)-N-(2,3,4,9-tetrahydro-1H-carbazol-6-ylmethyl)acetamide
N,2-dimethyl-N-[2-(phenylsulfanyl)ethyl]-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
N-(2-{5-[(cyclohexylmethyl)sulfanyl]-4-(4-methoxyphenyl)-4H-1,2,4-triazol-3-yl}ethyl)cyclobutanecarboxamide
3-cyclobutyl-N-[5-methyl-2-(1H-1,2,3,4-tetrazol-1-yl)phenyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carboxamide
N-benzyl-3-{1-[(2-butyl-1H-imidazol-4-yl)methyl]piperidin-4-yl}-N-methylpropanamide
N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-3-oxo-3,4-dihydroquinoxaline-2-carboxamide
4-[(3R,4R)-3-(azepan-1-ylmethyl)-4-(hydroxymethyl)pyrrolidine-1-carbonyl]-1-methyl-1,2-dihydropyridin-2-one
3-[1-(2-phenoxybenzoyl)azetidin-3-yl]pyridine
2-(2-hydroxyethyl)-8-[(4-phenoxyphenyl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
5-chloro-2-[4-(1-ethyl-1H-imidazol-2-yl)piperidine-1-carbonyl]phenol
8-(6,8-difluoroquinolin-4-yl)-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
N-[4-(2-{2,7-diazaspiro[4.5]decan-7-yl}-2-oxoethoxy)phenyl]propanamide
N-{[2-(2,4-difluorophenoxy)pyridin-3-yl]methyl}-3-methylpiperidine-3-carboxamide
N-[1-(cyclopropylmethyl)-1H-indazol-3-yl]-2-(1H-1,2,4-triazol-1-yl)acetamide
6-ethyl-2-methyl-4-[3-(propoxymethyl)pyrrolidine-1-carbonyl]quinoline
N-(3-methylphenyl)-3-[1-(oxane-4-carbonyl)piperidin-4-yl]propanamide
1-(5-{[4-(2-hydroxyethyl)piperidin-1-yl]methyl}-2-methoxyphenoxy)-3-(4-methylpiperazin-1-yl)propan-2-ol
7-{[2-fluoro-4-(trifluoromethyl)phenyl]methyl}-2,7-diazaspiro[4.4]nonane-1,3-dione
8-[(3-methylpyridin-2-yl)methyl]-2-(3-phenylpropyl)-2,8-diazaspiro[4.5]decan-3-one
(4aS,8aR)-6-[(4-methyl-1,3-thiazol-5-yl)methyl]-1-[2-(methylamino)ethyl]-decahydro-1,6-naphthyridin-2-one
N-(2,3-dihydro-1H-inden-2-yl)-2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
(1R,5S)-N-[1-methyl-3-(pyridin-2-yl)-1H-pyrazol-5-yl]-7-oxo-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
5-{3-[3-(2-fluorophenoxymethyl)piperidin-1-yl]-3-oxopropyl}-5-[(4-methoxyphenyl)methyl]pyrrolidin-2-one
2-(2-amino-4,6-dimethylpyrimidin-5-yl)-1-[4-(dimethylamino)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]ethan-1-one
N-[1-(pyridin-4-yl)propyl]-5-[(quinolin-6-yloxy)methyl]-1,2-oxazole-3-carboxamide
(1R,5R)-6-[(2-chloro-4-fluorophenyl)methyl]-3-(pyridine-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
1-(1H-imidazol-4-ylmethyl)-4-(3-phenylpropyl)-1,4-diazepane
2-{1-[(8-methoxy-3,4-dihydro-2H-1,5-benzodioxepin-7-yl)methyl]piperidin-2-yl}pyridine
N-ethyl-2-{1-[(2-fluoro-4-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-(2-methylprop-2-en-1-yl)acetamide
1-methyl-N-(propan-2-yl)-N-[(2,4,5-trimethoxyphenyl)methyl]piperidine-2-carboxamide
(3R,4R)-1-[(2-ethoxyphenyl)methyl]-4-(4-hydroxypiperidin-1-yl)piperidin-3-ol