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1-(6-methoxy-3-methyl-1-benzofuran-2-carbonyl)-4-(1-methyl-1H-imidazol-2-yl)piperidine
3-{1-[1-(2-hydroxybutyl)piperidin-4-yl]-1H-pyrazol-5-yl}-1-(2-methoxyphenyl)urea
8-[(1-methyl-1H-pyrazol-4-yl)methyl]-1-(2-phenylethyl)-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
7-methoxy-6-methyl-4-[2-(morpholin-4-yl)-1,3-thiazol-5-yl]-1,2,3,4-tetrahydroquinolin-2-one
5-[(2-methylphenyl)methyl]-4-(thiophen-2-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
(5S,9aS,9bS)-5-(4-methoxy-2,3-dimethylphenyl)-2-methyl-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
N-{[4-(oxolan-3-yloxy)phenyl]methyl}-N-(pyridin-2-ylmethyl)cyclohexanecarboxamide
(3S,4R)-3-benzyl-4-methyl-1-{2-methylimidazo[1,2-a]pyridine-3-carbonyl}piperidin-4-ol
2-methoxy-N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
N,3-dimethyl-4-oxo-N-[1-(pyridin-3-yl)pentyl]-3,4-dihydroquinazoline-7-carboxamide
{[2-(2,5-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(ethyl)(2-methylprop-2-en-1-yl)amine
5-cyclopropanecarbonyl-1'-[(2E)-3,7-dimethylocta-2,6-dien-1-yl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
2-[(3R,4S)-3-[4-(2-methyl-1H-imidazol-1-yl)butanamido]-4-propylpyrrolidin-1-yl]acetic acid
6-ethyl-N-methyl-2-(morpholin-4-yl)-N-[2-(1H-pyrazol-4-yl)ethyl]pyrimidin-4-amine
[(1S,3R,3aS,6aR)-5-methyl-1-phenyl-3-[1-(propan-2-yl)piperidin-4-yl]-octahydropyrrolo[3,4-c]pyrrol-1-yl]methanol
(1-{[2-(2,4-dimethoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-4-yl)methanol
2-ethoxy-5-[2-(4-ethylpiperazin-1-yl)pyrimidin-4-yl]benzoic acid
N-[(1-butyl-1H-1,2,4-triazol-5-yl)methyl]-N-methylaniline
2-[1-(2-methyloxane-2-carbonyl)azetidin-3-yl]pyridine
N-{[5-(dimethylcarbamoyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
2-[4-(2,6-dimethylpyridin-4-yl)piperazin-1-yl]-5-methoxypyrimidine
1-[2-(3-ethoxyphenoxy)ethyl]-N-methylpyrrolidine-3-carboxamide
N-[2-(pyrrolidine-1-sulfonyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]pyridine-4-carboxamide
3-(3-methoxyphenyl)-N-methyl-N-[3-(oxolan-2-yl)propyl]-1H-pyrazole-4-carboxamide
5-[(3R,4S)-3-amino-4-(5-methylfuran-2-yl)pyrrolidine-1-carbonyl]-N-ethyl-4-methyl-1,3-thiazol-2-amine
(3aR,5S,6S,7aS)-2-{[1-(5-chloropyridin-2-yl)-1H-pyrrol-2-yl]methyl}-octahydro-1H-isoindole-5,6-diol
1-methyl-2-(2-phenylpyrrolidine-1-carbonyl)piperidine
3-[(3R,4S)-1-[6-methyl-2-(methylamino)pyrimidin-4-yl]-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propanoic acid
N-(5-ethyl-1-methyl-1H-1,2,4-triazol-3-yl)-4-[(3-methylpiperidin-1-yl)methyl]benzamide
2-methyl-5-(3-{[(1-phenylpiperidin-4-yl)amino]methyl}pyrrolidin-1-yl)-2,3-dihydropyridazin-3-one
[(4aS,8aR)-6-[2-(4-chloro-1H-pyrazol-1-yl)ethyl]-decahydro-1,6-naphthyridin-4a-yl]methanol
7-[(4-fluorophenyl)methyl]-2-(pent-4-enoyl)-2,7-diazaspiro[4.5]decan-6-one
3-hexyl-8-(6-oxo-1,6-dihydropyridine-3-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
ethyl 4-(4-{4-[methyl(1H-pyrazol-5-ylmethyl)amino]piperidin-1-yl}benzoyl)piperazine-1-carboxylate
4-(3-chloro-4-methylphenyl)-3-[(methylamino)methyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
2-(4-benzyl-3-ethyl-5-oxo-1,4-diazepan-1-yl)acetamide
(3S,5R)-N3-(4-methylphenyl)-N5-[2-(4-methylphenyl)ethyl]piperidine-3,5-dicarboxamide
N-{[7-methoxy-2-(morpholin-4-yl)quinolin-3-yl]methyl}-5,6-dimethyl-2-oxo-N-(oxolan-2-ylmethyl)-1,2-dihydropyridine-3-carboxamide
2-{[(3-benzyl-1,2,4-oxadiazol-5-yl)methyl]amino}pyridine-3-carboxamide
methyl({[1-(2-methylpropyl)-2-phenylmethanesulfonyl-1H-imidazol-5-yl]methyl})(1,2-oxazol-3-ylmethyl)amine
1-(1-{[2,4-dimethyl-6-(1H-pyrazol-1-yl)phenyl]methyl}azetidin-3-yl)piperidine
1-[2-(4-chlorophenyl)ethyl]-N-cyclobutyl-6-oxopiperidine-3-carboxamide
2-(2-ethyl-1H-1,3-benzodiazol-1-yl)-N-[2-(6-hydroxy-2-methylpyrimidin-4-yl)ethyl]butanamide
4-(4-{5-propylpyrazolo[1,5-a]pyrimidin-7-yl}piperazin-1-yl)phenol
1-(4-{[3-(2-hydroxyethyl)-4-(propan-2-yl)piperazin-1-yl]methyl}phenyl)imidazolidin-2-one
(3R,9aR)-3-methyl-8-[(4-methylphenyl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
1-[1-(2,4-difluorobenzoyl)piperidin-4-yl]-3-phenylpropan-1-ol
2-(5-chloro-2-methoxypyridin-4-yl)-6-(piperidine-1-carbonyl)pyrazine
N-({2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}methyl)-2-(1,2,3,4-tetrahydroisoquinolin-2-yl)propanamide
3-propyl-1-[4-(1H-pyrazol-4-yl)butanoyl]piperidine-3-carboxylic acid