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N-[(2-methoxyphenyl)methyl]-N-(prop-2-en-1-yl)-1H-1,3-benzodiazole-2-carboxamide
N5-cyclopentyl-N6-[2-(methylsulfanyl)ethyl]-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
5-cyclohexaneamido-1-(2-methoxyethyl)-N-methyl-N-[1-(4-methyl-1,3-thiazol-2-yl)ethyl]-1H-1,3-benzodiazole-7-carboxamide
N-[3-hydroxy-1-(4-methylphenyl)propyl]-3-(3-hydroxy-3-methylbutyl)benzamide
2-amino-4-(1H-imidazol-4-yl)-5H,6H,7H-pyrrolo[2,3-h]quinoline-3-carbonitrile
5-(furan-3-yl)-1-(thiophen-2-ylmethyl)-1H,4H-pyrazolo[3,4-d]imidazole
N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-3,4-dihydro-2H-1-benzopyran-2-carboxamide
1-(2,3-dihydro-1H-inden-2-yl)-4-(1,2-oxazole-3-carbonyl)-1,4-diazepan-6-ol
N-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
N-cyclopropyl-3-{[(1-ethyl-1H-pyrazol-4-yl)methyl](methyl)sulfamoyl}benzamide
(3R,5S)-N3-(2,3-dihydro-1H-inden-5-yl)-1-[(4-hydroxyphenyl)methyl]-N5-(2-phenylethyl)piperidine-3,5-dicarboxamide
N-cyclobutyl-5-{1-[3-(thiophen-3-yl)propanoyl]pyrrolidin-2-yl}thiophene-2-carboxamide
5-(2-chloro-4-fluorophenoxymethyl)-N-[(1-methyl-2,3-dihydro-1H-indol-5-yl)methyl]-1,2-oxazole-3-carboxamide
methyl 5-[2-(quinazolin-4-yloxy)acetyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylate
N-{[6-chloro-4-(pyrrolidin-1-yl)quinazolin-2-yl]methyl}-4-methylbenzene-1-sulfonamide
2-(4-acetylphenoxy)-N-[1-(4-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]acetamide
2-{2-[(dimethylamino)methyl]-4-phenylphenoxy}-N-(1,3-thiazol-2-ylmethyl)acetamide
N-(1,1-dioxo-1λ6-thiolan-3-yl)-N-ethyl-3-(4-methylphenyl)-1H-pyrazole-5-carboxamide
N-[4-({1-[(3-methoxyphenyl)methyl]-2-oxo-3-phenyl-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-6-yl}methyl)phenyl]acetamide
7-[(6-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-2,3-dimethyl-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
3-[4-(4-chlorophenyl)-4-hydroxypiperidine-1-carbonyl]piperidine-1-carboxamide
4-[(3-chloro-4-propoxyphenyl)methyl]morpholine-2-carboxamide
1-{2-[({3-[1-(dimethylamino)ethyl]phenyl}methyl)(methyl)amino]ethyl}piperidin-2-one
2-(3-methyl-1,2-oxazol-5-yl)-1-{2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl}ethan-1-one
1-(4-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}piperidin-1-yl)-2-(2-methyl-1,3-thiazol-4-yl)ethan-1-one
(2,1,3-benzoxadiazol-5-ylmethyl)(methyl){[2-(propan-2-yl)pyrimidin-4-yl]methyl}amine
3-(5-methylfuran-2-yl)-N-{[(2S)-5-oxopyrrolidin-2-yl]methyl}-N-(pyridin-2-ylmethyl)-1H-pyrazole-5-carboxamide
({1-[2-(4-chlorophenyl)ethyl]piperidin-3-yl}methyl)[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl]methylamine
N-[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]-2-(3-fluorophenoxymethyl)-1,3-oxazole-4-carboxamide
1-{4-[4-(6-amino-2-methylpyrimidin-4-yl)piperazin-1-yl]phenyl}ethan-1-one
4-(5-oxo-3-propyl-4,5-dihydro-1H-1,2,4-triazol-4-yl)benzoic acid
2-{2-[4-(6-methylpyridin-2-yl)piperazin-1-yl]-2-oxoethyl}-2-azaspiro[4.5]decan-3-one
({4-[(dimethylamino)methyl]thiophen-2-yl}methyl)(1,4-dioxan-2-ylmethyl)methylamine
2-{[(2,3-difluorophenyl)formamido]methyl}-N,N-dimethyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide
({2,3-dimethylimidazo[2,1-b][1,3]thiazol-6-yl}methyl)({[4-ethoxy-3-(prop-2-en-1-yl)phenyl]methyl})amine
2-methyl-4-{4-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}phenol
2-{4-[3-(morpholin-4-ylmethyl)phenyl]phenyl}acetamide
methyl 6-{[4-(methoxycarbonyl)phenyl]methyl}-2-(piperidine-1-sulfonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
N-(pyridin-2-ylmethyl)-4-(3,3,3-trifluoropropyl)pyrimidin-2-amine
2-ethyl-4-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]pyridine
(3S,4R)-4-(2,3-dimethoxyphenyl)-1-{[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}pyrrolidine-3-carboxylic acid
methyl 4-[4-ethyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carboxylate
9-[(2-aminopyridin-3-yl)methyl]-2-(3-hydroxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
3-methyl-1-[4-(4-methylphenyl)phenyl]-3-[2-(2-oxopiperidin-1-yl)ethyl]urea
2-amino-N-[2-(4-fluoro-2-methoxyphenyl)phenyl]acetamide
3-[5-(2,3-dihydro-1H-inden-2-yl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]propanoic acid
1-[(1R,3S)-1,3-dihydroxy-7-azaspiro[3.5]nonan-7-yl]-4-(3,5-dimethyl-1H-pyrazol-1-yl)butan-1-one
4-[4-cyclopropyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-[(4-fluorophenyl)methyl]piperidine
2-oxo-N-[(5-phenyl-1,2-oxazol-3-yl)methyl]-1-oxaspiro[4.5]decane-4-carboxamide
N-(2-methoxyethyl)-4-methyl-3-{[(pyridin-4-ylmethyl)carbamoyl]methyl}-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide