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2-(2-chloro-6-fluorobenzamido)-N-methyl-N-[(2-methyl-1,3-thiazol-4-yl)methyl]-7-oxo-4,5,6,7-tetrahydro-1,3-benzothiazole-5-carboxamide
2-[4-(3-acetamidophenyl)-1H-pyrazol-1-yl]-N-(2-methyl-2H-1,2,3-triazol-4-yl)acetamide
N-methyl-2-(methylsulfanyl)-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}pyrimidine-5-carboxamide
(2R,3R,6R)-3-(4-methoxyphenyl)-5-(6-methylpyridine-3-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
2-amino-1-[(2R,3S,6R)-3-(3,5-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]ethan-1-one
2-ethyl-8-{2-[4-(1H-1,2,3,4-tetrazol-1-yl)phenyl]acetyl}-2,8-diazaspiro[4.5]decan-3-one
4-[(1-methoxybutan-2-yl)amino]-N,5-dimethyl-N-(propan-2-yl)thieno[2,3-d]pyrimidine-6-carboxamide
(4aR,8aR)-4a-hydroxy-N,N-dimethyl-7-(quinoline-6-carbonyl)-decahydro-2,7-naphthyridine-2-carboxamide
N-[2-({4-oxo-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3(8),6,12,14-pentaen-6-yl}amino)ethyl]pyridine-3-carboxamide
{1-[4-(2-chlorophenyl)-3-oxopiperazin-1-yl]-3-methyl-1-oxobutan-2-yl}urea
3-(2H-1,3-benzodioxol-5-yl)-N-methyl-N-[(3-methylpyridin-4-yl)methyl]-3-phenylpropanamide
4-methoxy-6-(1-methyl-1H-pyrazol-4-yl)quinazoline
N-{[2-(2,4-difluorophenoxy)pyridin-3-yl]methyl}-2-(2-oxopiperidin-1-yl)acetamide
5-(2-methoxyethyl)-1-(4-methoxyphenyl)-3-(2-methylpropyl)-1H-1,2,4-triazole
3-(2-fluoro-4-methoxyphenyl)-4-{[(2R)-2-(methoxymethyl)pyrrolidin-1-yl]methyl}-1-phenyl-1H-pyrazole
5-cyclohexaneamido-N-[(5-fluoro-2-methylphenyl)methyl]-1-(2-methoxyethyl)-1H-1,3-benzodiazole-7-carboxamide
1-[2-(3-chlorophenyl)acetyl]-4-(cyclopropylmethyl)-1,4-diazepan-5-one
(3S,4S)-1-[1-methyl-6-(pyridin-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]-4-(propan-2-yloxy)pyrrolidin-3-ol
3-benzyl-4-{[1-(2-hydroxyethyl)-3-methyl-1H-pyrazol-4-yl]methyl}piperazin-2-one
4-{[4-(5-methyl-1,2,4-oxadiazol-3-yl)piperidin-1-yl]methyl}-2,1,3-benzoxadiazole
7-[2-(3-methoxyphenyl)ethyl]-2-oxa-7-azaspiro[4.5]decan-8-one
(4aR,8aR)-2-[2-(1H-1,3-benzodiazol-1-yl)ethyl]-7-methanesulfonyl-decahydro-2,7-naphthyridin-4a-ol
2-(dimethylamino)-N-methyl-2-(3-methylphenyl)-N-(1,2-oxazol-3-ylmethyl)acetamide
4,4-difluoro-1-({3-methoxy-4-[(3-methylbut-2-en-1-yl)oxy]phenyl}methyl)piperidine
4-{4-[4-(3-ethenylphenyl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}-1λ6-thiane-1,1-dione
N-[(3-ethyl-1,2-oxazol-5-yl)methyl]-N-methyl-1,2,5-oxadiazole-3-carboxamide
(2R,3R,6R)-5-(5-ethyl-1,2-oxazole-3-carbonyl)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
6,7-dimethoxy-3-{[2-(4-methyl-1,2,5-oxadiazol-3-yl)pyrrolidin-1-yl]methyl}-1,2-dihydroquinolin-2-one
(3aS,6aR)-3-[3-(4-fluorophenyl)propyl]-5-(1,3-thiazol-2-ylmethyl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
N-(3-ethylphenyl)-N'-(2-hydroxy-2-phenylethyl)butanediamide
(3S,4R)-1-[(2,5-dimethylthiophen-3-yl)sulfonyl]-N,N-dimethyl-4-(propan-2-yl)pyrrolidin-3-amine
1-[4-(1-benzofuran-2-yl)pyrimidin-2-yl]-5-cyclopropyl-N-ethyl-N-(pyridin-4-ylmethyl)-1H-pyrazole-4-carboxamide
5-[3-(3,4-difluorophenyl)propanoyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
(3S,4R)-1-(2,6-difluorobenzoyl)-4-(4-fluorophenyl)pyrrolidine-3-carboxylic acid
N-ethyl-2-{8-[(5-methylpyrazin-2-yl)methyl]-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl}acetamide
N,N-diethyl-1-[1-(furan-2-ylmethyl)piperidin-3-yl]-1H-1,2,3-triazole-4-carboxamide
1-{5-propyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-2-(1H-pyrazol-1-yl)butan-1-one
1-(4,7-dimethyl-2-oxo-2H-chromen-6-yl)-3-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}urea
4-(2-methylphenoxy)-1-[2-(1H-1,2,4-triazol-1-yl)acetyl]piperidine-4-carboxylic acid
N-{[5-(4-methylphenyl)-1,2-oxazol-3-yl]methyl}-5-(morpholin-4-ylmethyl)furan-3-carboxamide
N-[2-(2-hydroxyethoxy)ethyl]-2-[(3S)-3-hydroxypyrrolidin-1-yl]-1-methyl-1H-1,3-benzodiazole-5-carboxamide
N-methyl-N-{2-[1-(3-methylpyridin-4-yl)-3-(propan-2-yl)-1H-1,2,4-triazol-5-yl]ethyl}methanesulfonamide
2-{imidazo[1,2-a]pyridine-6-carbonyl}-1-(propan-2-yl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole
1-(3-methylcinnolin-5-yl)-3-[2-(2-oxoimidazolidin-1-yl)ethyl]urea
3-fluoro-5-[4-(1,2,3,4-tetrahydroisoquinolin-2-yl)piperidine-1-carbonyl]benzonitrile
2-[(2R,3R,6R)-3-(4-fluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]benzonitrile
2-cyclopropyl-9-[(4-fluoro-3-methylphenyl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
1-[(4-ethylphenyl)methyl]-4-(pyridin-4-ylmethyl)-1,4-diazepan-5-one
5-(2-{[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]amino}ethyl)-1-(3-phenylpropyl)pyrrolidin-2-one
N-[(1-ethylpyrrolidin-2-yl)methyl]-N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}cyclohex-1-ene-1-carboxamide