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N-ethyl-N-[(2E)-3-phenylprop-2-en-1-yl]-2-(1,2,3,6-tetrahydropyridin-4-yl)acetamide
3-{[2-(2-butyl-1H-imidazol-4-yl)-1H-imidazol-1-yl]methyl}-5-(2-methylpropyl)-1,2,4-oxadiazole
9-[2-(1H-imidazol-2-yl)benzoyl]-2-(prop-2-en-1-yl)-2,9-diazaspiro[5.5]undecan-3-one
1-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}-4-(1,3-thiazol-2-yl)piperazine
N-[(5-chlorothiophen-2-yl)methyl]-2-ethylpyrimidine-5-carboxamide
2-cyclopentyl-9-(5-propylpyrimidin-4-yl)-2,9-diazaspiro[5.5]undecan-3-one
3-(3-fluorophenyl)-N-{[4-(4-methoxyphenyl)-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}benzamide
2-[(3,5-difluorophenyl)methyl]-8-(6-methylpyrimidin-4-yl)-2,8-diazaspiro[4.5]decan-3-one
N-{[3-(2H-1,3-benzodioxol-5-ylmethoxy)phenyl]methyl}-4-(2-oxopyrrolidin-1-yl)-N-(pyridin-2-ylmethyl)benzamide
N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]-1-(propan-2-yl)-1H-pyrazole-4-carboxamide
N-{[2-(2,4-difluorophenoxy)pyridin-3-yl]methyl}-5-(hydroxymethyl)furan-2-carboxamide
N-(2-methoxyethyl)-2-[(2S)-2-(methylamino)propanoyl]-1,2,3,4-tetrahydroisoquinoline-6-sulfonamide
(1-{[3-(2-chlorophenyl)-1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}piperidin-3-yl)methanol
N-[(1R,2S)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]-2-(3-methyl-5-oxo-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-1-yl)acetamide
N-[(1-ethylpyrrolidin-2-yl)methyl]-N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-3-methylthiophene-2-carboxamide
(1R,5R)-N-(3-chloro-4-fluorophenyl)-6-propyl-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
3-(5-{[3-(2-phenylpyridin-4-yl)pyrrolidin-1-yl]methyl}thiophen-3-yl)prop-2-yn-1-ol
(2E)-N-[2-(2-ethyl-7-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethyl]-3-(thiophen-2-yl)prop-2-enamide
4-[2-(2-{8-oxatricyclo[7.4.0.02,7]trideca-1(9),2(7),3,5,10,12-hexaen-6-yl}-1H-imidazol-1-yl)ethyl]-4H-1,2,4-triazole
(1S,6R)-9-[3-(5-methylfuran-2-yl)-1H-pyrazole-5-carbonyl]-3,9-diazabicyclo[4.2.1]nonan-4-one
5-(pyrrolidin-1-ylmethyl)-N-{2-[(trifluoromethyl)sulfanyl]ethyl}furan-2-carboxamide
1-(5-methyl-2-phenylfuran-3-carbonyl)-1,4-diazepan-6-ol
4-{8-chloro-1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}-N-cyclopropylpyridine-2-carboxamide
1-[(2-methoxyphenyl)methyl]-5-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]piperidin-2-one
6,7-dimethoxy-2-[3-(1H-pyrazol-4-yl)benzoyl]-1,2,3,4-tetrahydroisoquinoline
{[1-benzyl-2-(2-methoxyethanesulfonyl)-1H-imidazol-5-yl]methyl}(methyl)(thiophen-2-ylmethyl)amine
ethyl 4-{[5-methyl-2-(naphthalen-1-yl)-1,3-oxazol-4-yl]methyl}piperazine-1-carboxylate
1-methyl-N-{1-oxaspiro[4.5]decan-3-yl}-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-cyclopropyl-3-{5-[(5-methoxy-1,3,4-thiadiazol-2-yl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanamide
4-[4-(1-benzothiophen-2-yl)-1H-imidazol-2-yl]-1-(propan-2-yl)pyrrolidin-2-one
(3R,9aR)-3-[(benzylsulfanyl)methyl]-8-(4-fluorobenzoyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
3-methyl-N-{1-[1-(1,2,5-thiadiazole-3-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}butanamide
N-(3-{4-[(1,3-benzothiazol-2-ylmethyl)amino]piperidin-1-yl}phenyl)cyclopropanecarboxamide
3-(2-oxo-2-{4H,5H,6H,7H-thieno[3,2-c]pyridin-5-yl}ethyl)-4-(2-phenylethyl)piperazin-2-one
1-cyclohexyl-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
N,N,4,5-tetramethyl-6-[4-(1-propylpiperidin-4-yl)piperazin-1-yl]pyrimidin-2-amine
N,N-diethyl-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
2-(4-methylpiperazine-1-carbonyl)-6-[3-(1H-pyrazol-3-yl)phenyl]pyrazine
2-(1,3-dimethyl-2,5-dioxoimidazolidin-4-yl)-N-methyl-N-{[2-(trifluoromethyl)phenyl]methyl}acetamide
3-(3-chloro-1,2-oxazol-5-yl)-1-(4-cyclopentyl-1,4-diazepan-1-yl)propan-1-one
1-[(3,4-difluorophenyl)methyl]-3-hydroxy-3-{[(pentan-3-yl)amino]methyl}piperidin-2-one
1-{2-[(1S,6R)-3,9-diazabicyclo[4.2.1]nonan-9-yl]-2-oxoethyl}azepan-2-one
N-(2,1,3-benzoxadiazol-5-ylmethyl)-N-methyl-1,9-dioxaspiro[5.5]undecan-4-amine
1-(4-chlorophenyl)-N-({1-[3-(1,2-oxazolidin-2-yl)propanoyl]piperidin-3-yl}methyl)cyclopropane-1-carboxamide
1-[(5-methylfuran-2-yl)methyl]-5-(2,4,5-trimethoxyphenyl)-1H,4H-pyrazolo[3,4-d]imidazole
2-[1-(1-{[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}piperidin-4-yl)-1H-1,2,3-triazol-4-yl]propan-2-amine
{[4-(3-methoxybenzenesulfonyl)-1,4-oxazepan-6-yl]methyl}dimethylamine
9-ethyl-1-methyl-4-[(3-methyl-1-benzofuran-2-yl)methyl]-1,4,9-triazaspiro[5.6]dodecan-10-one
4-(4-methylphenyl)-N-[3-(sulfamoylmethyl)phenyl]piperazine-1-carboxamide
1-(3-methoxypropyl)-8-methyl-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione