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N-(2-acetamidophenyl)-2-[2-(3-methoxyphenyl)pyrrolidin-1-yl]acetamide
6-methoxy-N,3-dimethyl-N-[2-(5-methyl-1,2,4-oxadiazol-3-yl)ethyl]-1-benzofuran-2-carboxamide
N-(2-methylphenyl)-4-(4-phenyl-1H-1,2,3-triazol-1-yl)piperidine-1-carboxamide
N-(6,6-dimethyl-1-phenyl-4,5,6,7-tetrahydro-1H-indazol-4-yl)butanamide
2-(2,3-dihydro-1H-inden-1-yl)-N-[2-(pyrrolidine-1-sulfonyl)ethyl]acetamide
1-[2-(2-ethyl-1H-imidazol-1-yl)ethyl]-2-oxo-3-(pentan-3-yl)-1H,2H,3H-imidazo[4,5-b]pyridine-6-carboxylic acid
N-(1-{[5-(oxan-2-yl)furan-2-yl]methyl}piperidin-4-yl)methanesulfonamide
N-methyl-N-{[5-oxo-4-(3-phenoxyphenyl)-4,5-dihydro-1H-1,2,4-triazol-3-yl]methyl}methanesulfonamide
N-cyclobutyl-2-phenyl-5,6,7,8-tetrahydroquinazolin-5-amine
5-methyl-N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}pyrazolo[1,5-a]pyrimidin-7-amine
5-(dimethyl-1,2-oxazol-4-yl)-2,3-difluorophenol
5-(3-{[(1,3-benzothiazol-2-yl)amino]methyl}pyrrolidin-1-yl)-2-methyl-2,3-dihydropyridazin-3-one
N-[(4-fluorophenyl)methyl]-N-(1-hydroxybutan-2-yl)-5-methylthiophene-2-carboxamide
1-(3,4-diethoxyphenyl)-2-[2-(3-methyl-1,2,4-oxadiazol-5-yl)piperidin-1-yl]ethan-1-one
5-{[3-(2-hydroxyethyl)-4-[1-(propan-2-yl)piperidin-4-yl]piperazin-1-yl]methyl}-2-methoxyphenol
2-[4-(1H-imidazol-1-yl)phenyl]-1-[1-(thiophen-3-yl)propan-2-yl]-1H-imidazole
3-(1-{[4-(difluoromethoxy)phenyl]methyl}piperidin-4-yl)-N-[(4-fluorophenyl)methyl]propanamide
3-amino-1-{[5-methoxy-2-(1H-pyrazol-1-yl)phenyl]methyl}pyrrolidine-3-carboxylic acid
2-amino-6-(4-{1,3-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}piperazin-1-yl)-3,4-dihydropyrimidin-4-one
2-[4-fluoro-3-(hydroxymethyl)phenyl]-2-[4-(2-methylphenyl)-1,4-diazepan-1-yl]acetic acid
3-[4-(4-ethoxyphenyl)-1H-imidazol-2-yl]-1-ethylpiperidine
3-(3-methoxyphenyl)-N-methyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-1H-pyrazole-4-carboxamide
5-methyl-N-[2-methyl-1-(pyrrolidin-1-yl)propan-2-yl]-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
N-[2-(1H-1,3-benzodiazole-1-carbonyl)phenyl]piperidine-4-carboxamide
1-{4-[(2-hydroxy-3-methoxypropyl)amino]-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl}ethan-1-one
2-(4-acetylpiperazin-1-yl)-2-{4-[(butylcarbamoyl)amino]phenyl}acetic acid
6-{1-[2-(piperidin-2-yl)ethyl]-1H-1,2,3-triazole-4-carbonyl}-1H,2H,3H,4H,5H,6H,7H,8H-pyrazolo[3,4-d]azepin-3-one
3-(3-hydroxy-3-methylbutyl)-N-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]benzamide
2-(3-methoxyphenyl)-1,3-thiazole
3-[2-(3,5-dimethylpiperidin-1-yl)ethyl]-8-methyl-3,4-dihydroquinazolin-4-one
[(8-methoxyquinolin-5-yl)methyl](methyl){[5-methyl-2-(5-methylfuran-2-yl)-1,3-oxazol-4-yl]methyl}amine
N-methyl-N-[2-(1,2,4-oxadiazol-3-yl)ethyl]-3-phenoxypropanamide
N-ethyl-N-(2-methylprop-2-en-1-yl)-1-(2-methylpropyl)-5-oxopyrrolidine-3-carboxamide
N5-[(3-fluoro-4-methylphenyl)methyl]-N3-methyl-N3-(2-methylpropyl)-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
3-(5-methyl-4H-1,2,4-triazol-3-yl)-N-[(trimethylpyrazin-2-yl)methyl]aniline
N-[(1S,3aS,6aS)-octahydropentalen-1-yl]-3-(4-chloro-1H-pyrazol-1-yl)propanamide
N-[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl]-4-hydroxy-2-(pyridin-3-yl)pyrimidine-5-carboxamide
N-methyl-2-{5-propanoyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}pyridine-3-carboxamide
N-{[2-(1H-imidazol-1-yl)pyridin-3-yl]methyl}-2,2-dimethyl-4-oxo-3,4-dihydro-2H-pyran-6-carboxamide
ethyl 1-[5-(2,4-difluorophenoxymethyl)-1,2-oxazole-3-carbonyl]piperidine-4-carboxylate
4-[(2-{1-[(2S)-1-(prop-2-en-1-yl)pyrrolidine-2-carbonyl]piperidin-4-yl}-1H-imidazol-1-yl)methyl]pyridine
N-(2,1,3-benzothiadiazol-5-ylmethyl)-N-methyl-5-[(4H-1,2,4-triazol-3-ylsulfanyl)methyl]furan-2-carboxamide
4-chloro-2-{[3-(2-hydroxyethyl)-4-[(3-methoxyphenyl)methyl]piperazin-1-yl]methyl}phenol
N-({3-[2-(4-fluorophenyl)ethoxy]phenyl}methyl)-N-(pyridin-4-ylmethyl)oxolane-2-carboxamide
N-(2-methoxyethyl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]isoquinoline-1-carboxamide
(1R)-3-{[4-methyl-5-(piperidin-4-ylmethyl)-4H-1,2,4-triazol-3-yl]sulfanyl}-1-phenylpropan-1-ol
2-(furan-2-yl)-2-oxo-N-(2-phenyl-5,6,7,8-tetrahydroquinazolin-5-yl)acetamide
3-(2-ethylbutyl)-8-(1H-pyrrole-2-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
3-(2,3-dihydro-1,4-benzodioxin-6-ylsulfanyl)-N-[(2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)methyl]propanamide
3-[5-({4-[2-(methylsulfanyl)ethyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}methyl)furan-2-yl]-1H-pyrazole