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1-{[3-(2-chlorophenyl)-1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-4-methylpiperazine
8-(1-methyl-1H-pyrazole-3-carbonyl)-2-(3-methylbut-2-en-1-yl)-2,8-diazaspiro[4.5]decan-3-one
3-(3,5-dimethyl-1H-pyrazol-1-yl)-1-[3-(morpholine-4-carbonyl)-1-(2-phenylethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]propan-1-one
(4aS,7aR)-1-(1H-pyrazole-3-carbonyl)-4-(pyridin-3-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-(2H-1,3-benzodioxol-5-yl)-3-phenyl-N-[2-(1H-1,2,4-triazol-5-ylsulfanyl)ethyl]propanamide
2-cyclopropyl-N-(2-methoxyethyl)-4-methyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]pyrimidine-5-carboxamide
(3S,4R)-1-[(5-carboxyfuran-2-yl)methyl]-4-(3-fluorophenyl)pyrrolidine-3-carboxylic acid
N-[(5-tert-butyl-1,3-benzoxazol-2-yl)methyl]-4,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
N-(3,4-dihydro-2H-1,5-benzodioxepin-7-ylmethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
(3aR,6aR)-2-methyl-N-{[2-(trifluoromethyl)phenyl]methyl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
4-(4-cyclopropyl-1H-1,2,3-triazol-1-yl)-1-[(2-ethylphenyl)methyl]piperidine
1-(2,3-dihydro-1,4-benzodioxine-6-carbonyl)-4-[(dimethylamino)methyl]azepan-4-ol
(4aR,6R,8aS)-8a-(methoxymethyl)-2-[(1-methyl-1H-imidazol-2-yl)methyl]-6-(morpholin-4-yl)-decahydroisoquinoline
3-(4-methylphenoxymethyl)-1-(trimethyl-1H-pyrazole-4-carbonyl)piperidine
2,4-dimethoxy-5-[4-(1H-pyrazol-5-yl)phenyl]pyrimidine
3-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-(2-hydroxyethyl)propanamide
(3S,4S)-4-cyclopropyl-1-[4-(3,5-dimethyl-1H-pyrazol-1-yl)butanoyl]pyrrolidine-3-carboxylic acid
(1R,5R)-N,N-dimethyl-6-[2-(1-methyl-1H-indol-3-yl)acetyl]-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
2-[(isoquinolin-5-yloxy)methyl]-N-methyl-N-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]-1,3-oxazole-4-carboxamide
N-(1-{5H,6H,7H,8H,9H-[1,2,3,4]tetrazolo[1,5-a]azepine-9-carbonyl}piperidin-4-yl)benzamide
1-(butan-2-yl)-1-(pyridin-4-ylmethyl)-3-[3-(1H-1,2,4-triazol-1-ylmethyl)phenyl]urea
N-cyclopropyl-1-{1-[(4-hydroxy-5-methoxypyridin-2-yl)methyl]piperidin-4-yl}piperidine-3-carboxamide
3-(2-fluorophenoxymethyl)-1-[3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-carbonyl]piperidine
2-(furan-2-yl)-2-oxo-N-[(2E)-3-phenylprop-2-en-1-yl]-N-propylacetamide
2-{2-[(1R,9aR)-octahydro-1H-quinolizin-1-ylmethoxy]phenoxy}acetamide
2-[(2R,3R,6R)-3-(3-hydroxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]acetic acid
6-{[1-(ethoxymethyl)cyclopropyl]methyl}-2-methoxy-5-oxo-5,6-dihydro-1,6-naphthyridine-3-carbonitrile
2-amino-7-(2-methyl-4,5,6,7-tetrahydro-2H-indazole-3-carbonyl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
2-cyclopropyl-8-(2-methoxypyridine-4-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
N-benzyl-N-ethyl-5-(phenoxymethyl)-1H-pyrazole-3-carboxamide
3-ethyl-1-[2-methyl-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]piperidin-3-ol
4-chloro-N-[2-(ethanesulfonyl)ethyl]-1-methyl-1H-pyrazole-3-carboxamide
3-chloro-4-{[1-(2-hydroxypropanoyl)piperidin-4-yl]oxy}-N-(2-methoxyethyl)benzamide
4-[(2-chlorophenyl)methyl]-11-[(1,2-oxazol-3-ylmethyl)amino]-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
2-(2,4-dichlorophenoxy)-N-[2-(5-methyl-1,3,4-thiadiazol-2-yl)ethyl]acetamide
4-{4-phenyl-5-[2-(1H-pyrazol-1-ylmethyl)phenyl]-1H-imidazol-1-yl}piperidine
2-{[(4-methyl-2-propyl-1,3-thiazol-5-yl)methyl]amino}propan-1-ol
2-[2-(3-cyclopentyl-1,2,4-oxadiazol-5-yl)ethyl]pyrazine
3-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}-1-(1-methyl-1H-indazol-6-yl)urea
2-{1-[(4-methoxy-3-methylphenyl)methyl]-4-(1H-pyrazol-3-ylmethyl)piperazin-2-yl}ethan-1-ol
1-(2-chloro-6-methylbenzenesulfonyl)-4-hydroxypiperidine-4-carboxylic acid
(2R)-2-methyl-N-(5,6,7,8-tetrahydronaphthalen-2-ylmethyl)pyrrolidine-2-carboxamide
2-[3-(2-methoxyethyl)-5-(3-phenyl-1H-pyrazol-4-yl)-1H-1,2,4-triazol-1-yl]acetic acid
ethyl 1-[(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)methyl]-4-oxo-5-phenoxy-1,4-dihydropyridine-3-carboxylate
3-[1-(1H-imidazole-5-carbonyl)piperidin-3-yl]-N-[(3-methoxyphenyl)methyl]propanamide
5-acetyl-N-(furan-2-ylmethyl)-2,4-dimethyl-1H-pyrrole-3-carboxamide
4-({1-[(2,3-difluorophenyl)methyl]-3-hydroxy-2-oxopiperidin-3-yl}methyl)-3,3-dimethylpiperazin-2-one
3-hydroxy-1-[(3-methylphenyl)methyl]-3-({[(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)methyl]amino}methyl)piperidin-2-one
methyl({4-methyl-5-[(2-phenoxyethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)(quinolin-5-ylmethyl)amine
4,6-dimethyl-1-{2-[3-(2-methylphenyl)piperidin-1-yl]-2-oxoethyl}-1,2-dihydropyrimidin-2-one