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1-(4-{4-[6-(propan-2-yl)pyridin-2-yl]piperazin-1-yl}piperidin-1-yl)ethan-1-one
2-{[5-(4-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-yl]amino}propan-1-ol
N-[3-(1H-1,2,3-benzotriazol-1-yl)propyl]-3-(2,5-dioxoimidazolidin-4-yl)propanamide
4-methyl-2-[(3-methyl-1H-1,2,4-triazol-5-yl)methyl]-1,2-dihydrophthalazin-1-one
9-(6-fluoro-4-hydroxyquinoline-3-carbonyl)-1-oxa-9-azaspiro[5.5]undecan-5-ol
5-{[benzyl(methyl)amino]methyl}-N-(2-oxo-1,2,3,4-tetrahydroquinolin-4-yl)-1,2-oxazole-3-carboxamide
2-ethyl-N-[4-methyl-3-(4-methylbenzamido)phenyl]pyrimidine-5-carboxamide
3-(dimethylsulfamoyl)-N-[(1R)-1-(4-methoxyphenyl)ethyl]-5-{[(2-methylphenyl)methyl]amino}benzamide
2-amino-4-[4-ethoxy-3-(hydroxymethyl)phenyl]-5,6,7,8-tetrahydroquinoline-3-carbonitrile
{[2-(4-fluoro-3-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl){[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
methyl 4-{4-[2-methyl-2-(morpholin-4-ylmethyl)propyl]piperazin-1-yl}benzoate
N-[3-(2,6-dimethylphenoxy)propyl]-N-methyl-4-(1H-1,2,3,4-tetrazol-1-yl)benzamide
N-methyl-2-oxo-N-{[2-(pyrrolidin-1-ylmethyl)phenyl]methyl}-2,3-dihydro-1H-imidazole-4-carboxamide
N,4-dimethyl-2-(methylamino)-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}-1,3-thiazole-5-carboxamide
1-(6-ethyl-2-methylpyrimidin-4-yl)-N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}piperidin-4-amine
5-[4-(1H-pyrazol-5-yl)phenyl]pyridin-2-ol
8-(2-ethylpyridine-4-carbonyl)-3-hexyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-tert-butyl-5-(2-chlorophenoxymethyl)-3-methyl-1H-1,2,4-triazole
(1R,7S)-6-(4-methylpiperazine-1-carbonyl)-3-(pyridin-3-ylmethyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-4-one
1,3-dimethyl-N-({6-methylimidazo[1,2-a]pyridin-2-yl}methyl)-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
N-(2H-1,3-benzodioxol-5-yl)-1-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}piperidin-3-amine
2-(4-{[3-(phenylamino)piperidin-1-yl]methyl}phenoxy)ethan-1-ol
1-[3-(1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-3-(4-methyl-1H-pyrazol-1-yl)propan-1-one
N,3-dimethyl-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]-3H-imidazo[4,5-b]pyridine-6-carboxamide
N-(2-methoxy-5-methylphenyl)-2-methyl-3-oxo-2,9-diazaspiro[5.5]undecane-9-carboxamide
2-(2H-1,2,3-benzotriazol-2-yl)-1-[4-(3-methyl-1H-1,2,4-triazol-5-yl)piperidin-1-yl]ethan-1-one
2-{1-[3-(trifluoromethyl)-1H-pyrazole-5-carbonyl]piperidin-4-yl}-1,2,3,4-tetrahydroisoquinoline
ethyl 1-[(4-acetamidophenyl)methyl]-4-(3-phenylpropyl)piperidine-4-carboxylate
10-[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidine-1-carbonyl]-1-azatricyclo[6.3.1.04,12]dodeca-4(12),5,7,10-tetraen-9-one
[2-(diethylamino)-2-(furan-2-yl)ethyl][(2,3-difluorophenyl)methyl]amine
methyl 2-[(5-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-1,2-oxazol-3-yl)formamido]-4-(methylsulfanyl)butanoate
(1R,5R)-6-benzyl-3-(2-propyl-1,3-thiazole-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
2-[(thiolan-3-yl)amino]-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
2-(5-phenyl-1,2-oxazole-4-carbonyl)-7-propyl-2,7-diazaspiro[4.5]decan-6-one
(1S,6R)-9-(2-amino-4-ethyl-1,3-thiazole-5-carbonyl)-3,9-diazabicyclo[4.2.1]nonan-4-one
2-(2,5-dioxoimidazolidin-1-yl)-N-[2-(4-phenylpyrimidin-2-yl)ethyl]acetamide
3-{[1-(2,3-dihydro-1H-inden-5-yl)-1H-1,2,4-triazol-5-yl]methyl}-5,5-dimethylimidazolidine-2,4-dione
3-(3-methylphenyl)-N-(2-methylpropyl)-N-(pyridin-2-ylmethyl)-1H-pyrazole-4-carboxamide
(4aS,7aR)-4-benzoyl-N-ethyl-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
7-[4-(4-methoxyphenyl)-4-oxobutanoyl]-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide
6-(2-aminoethyl)-2-methyl-N-({2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}methyl)pyrimidin-4-amine
[5-({[(1-cyclopentylpiperidin-4-yl)methyl](oxolan-2-ylmethyl)amino}methyl)-2-(propan-2-yloxy)phenyl]methanol
1-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl]-4-[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl]piperidine
3-(3-chloro-1,2-oxazol-5-yl)-1-[(3R,4S)-4-hydroxy-3,4-dimethylpiperidin-1-yl]propan-1-one
(1-methyl-5-{1H-pyrrolo[2,3-b]pyridin-6-yl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl)methanol
1-(2-methanesulfonylethyl)-4-{2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-yl}piperazine
4-chloro-N-[(3R,5S)-5-(diethylcarbamoyl)-1-methylpyrrolidin-3-yl]-1H-indole-2-carboxamide
1-{4-[(2,2-dimethylpyrrolidin-1-yl)methyl]-2-methoxyphenoxy}-3-(morpholin-4-yl)propan-2-ol
N-ethyl-N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-2,6-dimethylquinoline-3-carboxamide
N-[2-(propan-2-yloxy)ethyl]-5-[(quinolin-6-yloxy)methyl]-1,2-oxazole-3-carboxamide