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N-(1H-imidazol-4-ylmethyl)-1-{[4-(2-methylpropyl)phenyl]methyl}piperidin-3-amine
2-methyl-N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]-1,3-thiazole-4-carboxamide
N3-tert-butyl-1-cyclohexyl-4-oxo-N5-[2-(pyridin-3-yl)ethyl]-1,4-dihydropyridine-3,5-dicarboxamide
3-[4-({6-[(dimethylamino)methyl]-1,4-oxazepan-4-yl}methyl)-1H-pyrazol-1-yl]propanoic acid
(3R,4R)-4-hydroxy-4-(2-methoxyethyl)-N,3-dimethyl-N-(propan-2-yl)piperidine-1-sulfonamide
N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}-2-(pyridin-3-yl)pyrimidine-5-carboxamide
4-(2H-1,3-benzodioxol-5-ylmethyl)-N-(5-ethyl-1-methyl-1H-1,2,4-triazol-3-yl)-3-oxopiperazine-1-carboxamide
2-[3-({4-[2-(methylsulfanyl)ethyl]piperazin-1-yl}methyl)phenoxy]acetamide
N-[2-(3-fluorophenyl)-2-hydroxyethyl]-2-[1-(propan-2-yl)piperidin-4-yl]acetamide
1-methyl-2-oxo-N-{[2-(pyrrolidin-1-yl)-1,3-thiazol-4-yl]methyl}-1,2,5,6,7,8-hexahydroquinoline-3-carboxamide
1-methyl-5-{2-[2-(pyrrolidin-1-yl)ethyl]piperidine-1-carbonyl}-1,2-dihydropyridin-2-one
5-(2-methoxyphenoxymethyl)-N-(2-methylbutyl)-1H-pyrazole-3-carboxamide
1-(3-methoxybenzoyl)-4-(2-phenylethyl)piperidine-4-carboxylic acid
N-[1-(dimethylamino)butan-2-yl]-6-(3-fluorophenyl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
3-(1H-pyrazol-5-yl)-1-[4-(1H-1,2,3,4-tetrazol-1-ylmethyl)benzoyl]piperidine
1-ethyl-N-methyl-5-{[(4-methylphenyl)methyl]amino}-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
7-(2-cyclohexylethyl)-2-(5-methyl-1,2-oxazole-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
1-(furan-2-carbonyl)-4-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)-1,4-diazepane
4-[1-(cyclopropylmethyl)-1H,4H-pyrazolo[3,4-d]imidazol-5-yl]-1-(2-methylphenyl)-1H-pyrazole
4-fluorophenyl (7R,9aR)-7-[(benzylsulfanyl)methyl]-6,9-dioxo-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxylate
N-(4-{[benzyl(prop-2-yn-1-yl)carbamoyl]methoxy}phenyl)propanamide
1-{4-[(3-chlorophenyl)methyl]piperazin-1-yl}-2-(1-methylpiperidin-2-yl)ethan-1-one
5-(2H-1,3-benzodioxol-5-ylmethyl)-1-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-5-methylpiperidin-2-one
N-methyl-N-[2-(pyridin-2-yl)ethyl]-3-{1-[2-(thiophen-2-yl)acetyl]piperidin-3-yl}propanamide
N,3,5-trimethyl-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-4-oxo-3H,4H-thieno[2,3-d]pyrimidine-6-carboxamide
3-(1-{2-[(4S)-2-oxo-4-(propan-2-yl)-1,3-oxazolidin-3-yl]acetyl}piperidin-4-yl)benzonitrile
2-ethyl-7-(2-methoxybenzamido)-N,1-dimethyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-1H-1,3-benzodiazole-5-carboxamide
2-(methylsulfanyl)-3-{4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyridine
3-(furan-2-yl)-N-[4-methyl-1-(pentan-3-yl)-1H-pyrazol-5-yl]-3-phenylpropanamide
{[2-(4-fluoro-3-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)(quinolin-5-ylmethyl)amine
N-[1-(1,5-dimethyl-1H-pyrazol-4-yl)ethyl]thieno[2,3-d]pyrimidin-4-amine
1-{3-[3-(morpholin-4-yl)-3-oxopropyl]piperidin-1-yl}-3-phenylprop-2-yn-1-one
benzyl (7S,9aR)-7-[(1R)-1-hydroxyethyl]-6,9-dioxo-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxylate
3-[(3-phenylpiperazin-1-yl)methyl]-1,2-dihydroquinolin-2-one
1-[2-(3-methylthiophen-2-yl)ethyl]-4-(oxolan-3-yl)-1H-1,2,3-triazole
3-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)ethyl]-1-[3-(methylsulfamoyl)phenyl]urea
4-(5-ethyl-2-methylpyrimidin-4-yl)piperazine-1-carboxamide
4-{3-[4-(4-methoxypyrimidin-2-yl)piperazine-1-carbonyl]phenyl}-2-methylbutan-2-ol
3-{[1-(1,2-oxazole-5-carbonyl)pyrrolidin-3-yl]methyl}benzamide
2-{4-[3-(2-chlorophenyl)pyrrolidin-1-yl]azepan-1-yl}-7-methanesulfonyl-4-methylquinazoline
1-(3-{[(4-hydroxy-6-methylquinolin-2-yl)methyl]amino}propyl)pyrrolidin-2-one
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-2-(morpholin-4-yl)pyridine-3-carboxamide
(4aR,8aR)-7-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-4a-hydroxy-N,N-dimethyl-decahydro-2,7-naphthyridine-2-sulfonamide
(4aR,7aS)-N-[2-methyl-3-(pyrrolidin-1-yl)phenyl]-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
N-methyl-N-[(2-phenyl-1,3-oxazol-4-yl)methyl]-1-(2-phenylethyl)piperidin-3-amine
N-[(5-methylpyrazin-2-yl)methyl]-4-propylpyrimidine-5-carboxamide
2-ethyl-9-[4-(4-methoxyphenyl)butanoyl]-2,9-diazaspiro[5.5]undecan-3-one
5-chloro-2-[(4-methyl-1H-imidazol-2-yl)methyl]-1,2,3,4-tetrahydroisoquinoline
4-[(4-methyl-1H-pyrazol-1-yl)methyl]-1-[1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]piperidine
1-{5-hydroxy-1-oxa-9-azaspiro[5.5]undecan-9-yl}-2-[2-(trifluoromethyl)phenyl]ethan-1-one