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1-cyclobutanecarbonyl-4-[2-(4-fluorophenyl)pyrrolidine-1-carbonyl]piperidine
[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl][3-(pyrrolidin-1-yl)propyl]amine
(3S,4R)-4-(hydroxymethyl)-1-[4-(1-phenyl-1H-imidazol-4-yl)benzoyl]piperidin-3-ol
2-{4-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyrazine
1-ethyl-N-{imidazo[1,2-a]pyridin-3-ylmethyl}-N,3-dimethyl-1H-pyrazole-4-carboxamide
4-(2-{[5-(methoxymethyl)pyrazolo[1,5-a]pyrimidin-7-yl]amino}ethyl)benzene-1-sulfonamide
N-{[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl}-1-(pyrimidin-2-yl)piperidin-3-amine
(3aS,6aS)-2-cyclopentanecarbonyl-5-[(2-methyl-1,3-thiazol-4-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-(benzylsulfamoyl)-N-ethyl-2,2-dimethyloxan-4-amine
6-methyl-2-({4-[6-(4-methyl-1H-pyrazol-1-yl)pyrimidin-4-yl]piperazin-1-yl}methyl)pyridin-3-ol
2-amino-7-[2-(methylamino)pyridine-3-carbonyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
2-[3-(2,6-dimethylphenoxy)azetidine-1-carbonyl]-1-methyl-1H-pyrrole
N-(2-phenoxyethyl)-2-(pyridin-3-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
4-[(1-ethyl-5-methyl-1H-pyrazol-4-yl)sulfonyl]-2-(trifluoromethyl)morpholine
2-[2-(7-chloro-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-2-oxoethyl]-1,2-dihydrophthalazin-1-one
1-({1-[(3-cyanophenyl)methyl]piperidin-3-yl}methyl)-3-ethylurea
(dicyclopropylmethyl)({[3-(diphenylmethyl)-1,2,4-oxadiazol-5-yl]methyl})methylamine
(2S)-2-[(1-cyclohexylpiperidin-4-yl)formamido]-2-phenylacetamide
(4aS,8aR)-6-(naphthalene-1-carbonyl)-1-propyl-decahydro-1,6-naphthyridin-2-one
1-{[2-(2,5-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidine
5-{[4-(4-methoxybenzoyl)piperazin-1-yl]methyl}-2,1,3-benzoxadiazole
(3aS,6aR)-5-(1,3-benzoxazol-2-yl)-3-[3-(morpholin-4-yl)propyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
2-{2-oxo-1H,2H,5H,6H,7H-cyclopenta[b]pyridine-3-carbonyl}-7-propyl-2,7-diazaspiro[4.5]decan-6-one
(2S,4S)-4-{[(3,4-difluorophenyl)methyl]amino}-N-ethyl-1-(propan-2-yl)pyrrolidine-2-carboxamide
N-(1,4-dioxan-2-ylmethyl)-2,3-dimethyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine
5-[(1S,5R)-3-benzyl-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
methyl (2S)-2-{[5-(tert-butylcarbamoyl)-1-cyclohexyl-4-oxo-1,4-dihydropyridin-3-yl]formamido}-2-phenylacetate
(3-{2-[1-(3-chloro-5-fluorobenzoyl)piperidin-4-yl]-1H-imidazol-1-yl}propyl)dimethylamine
(3R,5S)-N-(2-methylpropyl)-5-{[(6-methylpyridin-3-yl)oxy]methyl}-1-(pyridin-4-ylmethyl)piperidine-3-carboxamide
2-(5-{[methyl(propan-2-yl)amino]methyl}-1H-1,2,3,4-tetrazol-1-yl)-1-{4-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}ethan-1-one
4-[2-fluoro-3-(trifluoromethyl)phenyl]-6-(methoxymethyl)pyrimidine
N-(3-ethylphenyl)-4-[2-(4-methyl-1,2,5-oxadiazol-3-yl)pyrrolidin-1-yl]-4-oxobutanamide
3-[(4-methylpiperazin-1-yl)sulfonyl]-5-(1H-pyrazol-1-yl)benzoic acid
3-(1,3-benzothiazol-5-yl)-1-[2-(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)ethyl]urea
6-[4-(4-cyclopentyl-1H-1,2,3-triazol-1-yl)piperidin-1-yl]-9H-purin-2-amine
N-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-1-(oxan-4-yl)piperidine-3-carboxamide
1-(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-carbonyl)-4-(thiophen-3-ylmethyl)piperazine
[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl](methyl)({1-[2-(2-methylphenyl)ethyl]piperidin-3-yl}methyl)amine
1-(4-benzyl-3-ethyl-5-oxo-1,4-diazepan-1-yl)butane-1,2-dione
N-[(4,6-dimethylpyridin-2-yl)methyl]-N-methyl-4-(1H-pyrazol-4-yl)butanamide
2-(ethylsulfanyl)-5-{[3-(pyridine-2-carbonyl)piperidin-1-yl]methyl}pyrimidine
1-(3-methoxypropyl)-3-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidine
1-benzyl-5-{[(4-cyclohexyl-4H-1,2,4-triazol-3-yl)methyl]amino}azepan-2-one
4-({5-methyl-2-[3-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)-1-phenylpiperazin-2-one
6-methyl-N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}-2-oxo-1,2-dihydropyridine-4-carboxamide
2-(adamantan-1-yl)-4-hydroxy-N-[(2S)-pyrrolidin-2-ylmethyl]pyrimidine-5-carboxamide
3-(oxolan-2-ylmethyl)-5-(pyridin-2-yl)-5-{1-[2-(thiophen-3-yl)acetyl]piperidin-4-yl}imidazolidine-2,4-dione
(3R,4R)-3-[ethyl({[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl})amino]-4-hydroxy-1λ6-thiolane-1,1-dione
(4aS,8aR)-6-(1,3-thiazole-4-carbonyl)-1-[2-(thiophen-2-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
5-(2-chloro-4-fluorophenoxymethyl)-N-[2-(dimethyl-1,3-thiazol-2-yl)ethyl]-1,2-oxazole-3-carboxamide