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N-ethyl-2-(4-{[(2S,5R)-5-(pyrrolidin-1-ylmethyl)oxolan-2-yl]methyl}phenyl)acetamide
1-[(2-ethylpyrimidin-4-yl)methyl]-4-(4-fluorophenyl)-1,4-diazepane
N-(4-{3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-4-oxobutyl)acetamide
N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-2-(morpholin-4-yl)-6-{8-thiatricyclo[7.4.0.02,7]trideca-1(9),2(7),3,5,10,12-hexaen-6-yl}pyridine-3-carboxamide
N-(1H-1,2,3-benzotriazol-4-yl)azepane-1-carboxamide
1-[(3-cyclohexyl-1,2-oxazol-5-yl)methyl]pyrrolidin-2-one
N-{[1-(1H-1,3-benzodiazol-2-ylmethyl)pyrrolidin-3-yl]methyl}-3-methylpyridine-2-carboxamide
8-[4-(1H-pyrazol-1-yl)phenyl]-2-(pyrrolidin-1-yl)-4H,5H,6H,7H,8H-[1,3]thiazolo[4,5-c]azepin-6-one
1-(2-fluorophenyl)-4-[1-(3-propyl-1H-pyrazole-4-carbonyl)piperidin-3-yl]piperazine
methyl 3-{[(4-methyl-1H-imidazol-2-yl)formamido]methyl}-5-[(2E)-3-phenylprop-2-enamido]benzoate
1-[(2,3-dichlorophenyl)methyl]-4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperidine
3-[5-(2,8-dimethylquinoline-3-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]propanoic acid
2-(4-methyl-1,2,5-oxadiazol-3-yl)-1-{3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
5-methyl-3-({2-methyl-2,8-diazaspiro[4.5]decan-8-yl}methyl)-1H-indole-2-carboxylic acid
1-(4-benzylpiperazin-1-yl)-3-[1-(2-phenylethyl)piperidin-3-yl]propan-1-one
3-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]-3H,4H-pyrido[3,4-d]pyrimidin-4-one
3-[3,5-dimethyl-1-(propan-2-yl)-1H-pyrazol-4-yl]-1-{2-[(4-ethyl-5-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}urea
N-methyl-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-3-(3-oxo-3,4-dihydro-2H-1,4-benzoxazin-4-yl)propanamide
3-(2-{1-[2-(1H-1,2,3,4-tetrazol-5-yl)benzoyl]piperidin-2-yl}ethyl)phenol
N-{[1-(1-benzofuran-2-ylmethyl)pyrrolidin-3-yl]methyl}-2-methyl-2-(methylamino)propanamide
N-[(3R,5S)-5-(diethylcarbamoyl)-1-(oxan-4-yl)pyrrolidin-3-yl]-1-methyl-1H-pyrazole-5-carboxamide
N,N-dimethyl-2-[(1S,5R)-6-[3-(5-methyl-1H-1,2,4-triazol-3-yl)propanoyl]-3,6-diazabicyclo[3.2.2]nonan-3-yl]acetamide
3-[(3R,4S)-4-(4-methylpiperazin-1-yl)-1-[(2E)-3-phenylprop-2-en-1-yl]piperidin-3-yl]propanoic acid
(1S,4S)-5-(cyclopropanesulfonyl)-2-(2-methoxy-5-phenylphenyl)-2,5-diazabicyclo[2.2.1]heptan-3-one
N-[(3,5-dimethyl-2-phenyl-1H-indol-7-yl)methyl]-4-(1H-1,2,4-triazol-1-yl)butanamide
3-phenyl-N-{2-[2-(pyrazin-2-yl)-1,3-thiazol-4-yl]ethyl}-1H-pyrazole-4-carboxamide
N-(propan-2-yl)-2-[4-(propan-2-yloxy)phenyl]pyrimidin-4-amine
3-cyclopropyl-1-[(3S,4S)-3-hydroxy-4-(naphthalen-2-yl)piperidin-1-yl]propan-1-one
N-[3-(1,3-benzothiazol-2-yl)propyl]-5-oxo-1-(pyridin-4-ylmethyl)pyrrolidine-3-carboxamide
8-({7-methylimidazo[1,2-a]pyridin-2-yl}methyl)-3-phenyl-1,8-diazaspiro[4.5]decan-2-one
5-fluoro-3-methyl-2-{[3-(1H-pyrazol-5-yl)piperidin-1-yl]methyl}-1H-indole
3-[(1S,9aR)-octahydro-1H-quinolizin-1-yl]-N-[2-(5-amino-1,3,4-thiadiazol-2-yl)ethyl]propanamide
3-cyclopropyl-N-[(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)methyl]-1H-pyrazole-5-carboxamide
7-cyclohexyl-2-[4-(hydroxymethyl)-1,3-thiazol-2-yl]-2,7-diazaspiro[4.5]decan-6-one
2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]-N-(prop-2-en-1-yl)-N-(pyridin-3-ylmethyl)acetamide
1-[(3,4-dimethoxypyridin-2-yl)methyl]-4-phenyl-3-(piperidin-3-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
7-(2-hydroxyethyl)-2-(4,5,6,7-tetrahydro-1-benzothiophene-2-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
2-(methoxymethyl)-6-methyl-N-{[1-(morpholin-4-yl)cyclopentyl]methyl}-1-(naphthalen-1-ylmethyl)-4-oxo-1,4-dihydropyridine-3-carboxamide
2-{5-[(2-methyl-1H-1,3-benzodiazol-5-yl)methyl]-3-(1-phenylcyclopropyl)-1H-1,2,4-triazol-1-yl}ethan-1-ol
N-[(3S,4R)-4-(5-methylfuran-2-yl)-1-{[4-(1H-pyrazol-1-yl)phenyl]methyl}pyrrolidin-3-yl]acetamide
N-butyl-N-[(4-fluorophenyl)methyl]-2-{2-oxo-1-oxa-3,8-diazaspiro[4.5]decan-3-yl}acetamide
3-(2-ethoxyethyl)-1-(4-methylpent-3-en-1-yl)-2-oxo-1H,2H,3H-imidazo[4,5-b]pyridine-6-carboxylic acid
4-[6-(2-aminoethyl)-2-methylpyrimidin-4-yl]-3-butyl-1-methylpiperazin-2-one
3-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-[(2,4-difluorophenyl)methyl]benzamide
3-[5-({2-[5-methyl-2-(thiophen-2-yl)-1,3-oxazol-4-yl]-1H-imidazol-1-yl}methyl)-1,2-oxazol-3-yl]pyridine
N-[2-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]-6-[(1,3-dihydroxy-2-methylpropan-2-yl)amino]pyridine-3-carboxamide
2-(1-benzofuran-2-yl)-N-methylbenzamide
8-(2-aminopyrimidin-4-yl)-2-(3-methylbutyl)-2,8-diazaspiro[5.5]undecan-3-one
4-(1H-imidazol-1-ylmethyl)-1-{[5-(oxan-2-yl)furan-2-yl]methyl}piperidin-4-ol
N-(1,1-dioxo-1λ6-thiolan-3-yl)-N-ethyl-2,3-dihydro-1-benzofuran-7-carboxamide