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N-{[7-(pyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2,3,4,9-tetrahydro-1H-carbazole-1-carboxamide
4-{3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine
3-{[5-oxo-1-(3-phenylpropyl)pyrrolidin-3-yl]carbamoyl}pyridin-1-ium-1-olate
9-(2,5-dimethylfuran-3-carbonyl)-2-[2-(pyridin-3-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
(3S,4S)-1-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-4-(propan-2-yl)pyrrolidine-3-carboxylic acid
N-{[3-(ethoxymethyl)-4-methoxyphenyl]methyl}pyrazin-2-amine
N-[(2-methylphenyl)methyl]-2-(phenoxymethyl)-1,3-oxazole-4-carboxamide
N-ethyl-4-[(furan-2-ylmethyl)amino]-5-methyl-N-(pyridin-4-ylmethyl)thieno[2,3-d]pyrimidine-6-carboxamide
3-(2-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-2-oxoethyl)-6-methyl-2,3-dihydro-1H-indol-2-one
1-[3-(furan-2-yl)propanoyl]-4-(4-methylphenoxy)piperidine-4-carboxylic acid
({2-[4-(2-methoxyphenyl)piperazin-1-yl]pyridin-3-yl}methyl)[(1-methyl-1H-pyrazol-4-yl)methyl]amine
9-(5-hydroxypyrazine-2-carbonyl)-2-[(1r,4r)-4-hydroxycyclohexyl]-2,9-diazaspiro[5.5]undecan-3-one
7-methyl-3-[2-(phenylsulfanyl)acetyl]-3,7,11-triazaspiro[5.6]dodecan-12-one
5-methoxy-9-[4-(trifluoromethyl)pyrimidin-2-yl]-1-oxa-9-azaspiro[5.5]undecane
1-{1-[(2-fluorophenyl)methyl]-1H-pyrazol-4-yl}-3-[(3-methyloxetan-3-yl)methyl]urea
2-cycloheptyl-1-(4-{[4-(1-hydroxyethyl)-1H-1,2,3-triazol-1-yl]methyl}piperidin-1-yl)ethan-1-one
5-{5-[(2-methoxy-4-methylphenyl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}-1,2-dimethyl-1H-imidazole
1-[2-(3-methyl-1,2-oxazol-5-yl)pyrrolidin-1-yl]-3-(3-phenyl-1,2,4-oxadiazol-5-yl)propan-1-one
(1S,5R)-6-(2-methoxyethyl)-3-[(8-methoxyquinolin-2-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
2-[({[4-(3-chlorophenyl)-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}(methyl)amino)methyl]-6-ethoxyphenol
4-(1-benzyl-1H-pyrazol-4-yl)-1-[2-(piperidin-1-yl)ethyl]-1,2,3,6-tetrahydropyridine
6-[3-(2-phenylethyl)-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-[(4-fluorophenyl)methyl]-4-{[6-methyl-2-(propan-2-yl)pyrimidin-4-yl]amino}pyrrolidin-2-one
5-ethyl-N-{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-N-methylthiophene-3-carboxamide
3-[(1R,5R)-6-(cyclobutylmethyl)-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]-4,5,6,7-tetrahydro-1,2-benzoxazole
4-({3-[2-(2-fluorophenyl)ethyl]piperidin-1-yl}methyl)-2-methoxyphenol
N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-N,1-dimethyl-3-propyl-1H-pyrazole-5-carboxamide
3,5-difluoro-2-[4-(4-fluorophenoxy)piperidine-1-carbonyl]pyridine
1-[4-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]-2-[5-(4-fluorophenyl)-2H-1,2,3,4-tetrazol-2-yl]ethan-1-one
N-(1,1-dioxo-1λ6-thiolan-3-yl)-N-ethyl-2-{imidazo[2,1-b][1,3]thiazol-6-yl}acetamide
methyl (2S,4S)-1-(cyclohexylmethyl)-4-(pyridine-2-amido)pyrrolidine-2-carboxylate
2-{5-[2-(1H-imidazol-2-yl)phenyl]-1,2,4-oxadiazol-3-yl}pyrimidine
4-{2,2-dimethyl-3-[4-(pyridin-3-yl)piperazin-1-yl]propyl}morpholine
5-cyclopropyl-N-[3-(1H-imidazol-1-yl)propyl]-N-(pyridin-3-ylmethyl)-1,3-oxazole-4-carboxamide
3-[(3R,4S)-3-(2-methoxy-2-methylpropanamido)-4-propylpyrrolidin-1-yl]propanoic acid
6-{2-[3-(2-methylphenyl)pyrrolidin-1-yl]ethyl}-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
(3R)-1-(5-{[methyl(2-phenylethyl)amino]methyl}-1,2-oxazole-3-carbonyl)pyrrolidin-3-ol
1-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-2-[2-(1-methyl-1H-imidazol-2-yl)ethyl]piperidine
N-[3-methyl-1-(pentan-3-yl)-1H-pyrazol-5-yl]-2-(2-oxo-1,3-oxazolidin-3-yl)acetamide
5-{[4-(5-chloropyrimidin-2-yl)piperazin-1-yl]methyl}-2-hydroxybenzoic acid
4-(4-hydroxyphenyl)-N-[2-(3-hydroxypiperidin-1-yl)ethyl]benzamide
5-[1-(2H-1,3-benzodioxol-5-ylmethyl)-1H-1,2,3-triazol-4-yl]pyrimidine
5-(4-chloro-2-methoxyphenoxymethyl)-N-[(4-methyl-1H-imidazol-2-yl)methyl]-1,2-oxazole-3-carboxamide
1-{2-[(3R,4R)-4-ethyl-3,4-dihydroxypiperidin-1-yl]-2-oxoethyl}-4,6-dimethyl-1,2-dihydropyrimidin-2-one
(cyclopentylmethyl)({[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl})methylamine
1-(cyclopropylmethyl)-5-[1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]-N-(pyridin-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
(1R,3S)-7-[6-(3-fluorophenyl)pyridine-3-carbonyl]-3-methoxy-7-azaspiro[3.5]nonan-1-ol
N-[(3R,4R)-3-hydroxy-1-{2-[4-(hydroxymethyl)phenyl]acetyl}piperidin-4-yl]pyrazine-2-carboxamide
N,N-dimethyl-6-[3-(5-oxo-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-3-yl)piperidin-1-yl]pyridine-3-carboxamide
1-hydroxy-N-[4-methyl-1-(pentan-3-yl)-1H-pyrazol-5-yl]naphthalene-2-carboxamide