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(3-{5-[(trimethyl-1H-pyrazol-1-yl)methyl]-1,2,4-oxadiazol-3-yl}phenyl)methanol
2-(3-chlorophenyl)-4-{4-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]piperazin-1-yl}-2,3-dihydro-1H-isoindole-1,3-dione
3-(3-hydroxy-3-methylbut-1-yn-1-yl)-N-methyl-N-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}benzamide
5-{5-butyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-ylmethyl}-N-(propan-2-yl)pyrimidin-2-amine
1-[cyclohexyl(methyl)amino]-3-{4-[(dimethylamino)methyl]-2-methoxyphenoxy}propan-2-ol
5-[4-methoxy-3-(methoxymethyl)phenyl]-3-(2-phenylethyl)-1H-1,2,4-triazole
2-(2-{[3-(4-hydroxyphenyl)-1H-pyrazol-5-yl]formamido}ethyl)-4-methyl-1,3-thiazole-5-carboxylic acid
3-[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl]-5-methoxy-3,4-dihydroquinazolin-4-one
1-methyl-N-{[3-(2-methylpropyl)-1,2-oxazol-5-yl]methyl}-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
3-(5-fluoro-1H-1,3-benzodiazol-2-yl)-N-[(3R)-piperidin-3-yl]propanamide
N-(3,4-dihydro-2H-1-benzopyran-6-ylmethyl)-2-(4-methyl-1-oxo-1,2-dihydrophthalazin-2-yl)acetamide
1-(2-{[(3-ethoxypropyl)amino]methyl}phenoxy)-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-ol
N-methyl-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-5-[3-(3-phenylpropyl)-1,2,4-oxadiazol-5-yl]pyridin-2-amine
N-[1-(3-fluorophenyl)-4-(propan-2-yloxy)-1H-indazol-3-yl]-3-methyl-1,2-oxazole-5-carboxamide
(1R,5R)-3-(1-ethyl-1H-indole-5-carbonyl)-6-propyl-3,6-diazabicyclo[3.2.2]nonane
2-[2-(2-methoxyphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-N-[(5-phenyl-1H-pyrazol-3-yl)methyl]acetamide
2-(2,4-dimethyl-6-oxo-1,6-dihydropyrimidin-5-yl)-N-{1-[5-methyl-1-(2-methylphenyl)-1H-pyrazol-4-yl]ethyl}acetamide
2-cyclopentanecarbonyl-7-[(2,3-dimethoxyphenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
4-[2-(methoxymethyl)naphthalen-1-yl]-N,N-dimethylbenzamide
(3S,4S)-4-methyl-1-(3-phenoxybenzoyl)piperidine-3,4-diol
9-(1H-indol-4-yl)-1-methyl-1H,2H,3H,6H,7H,8H,9H-[1,4]oxazino[3,2-g]quinoline-2,7-dione
4-[2-(2-hydroxyphenyl)-6-methylpyrimidin-4-yl]piperazin-2-one
[(3-ethyl-1,2-oxazol-5-yl)methyl]({[2-(2-fluoro-4-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl})methylamine
2,6-dimethoxy-N-(1-methyl-2-oxopyrrolidin-3-yl)pyridine-3-carboxamide
8-[(2S,3R)-2-amino-3-hydroxybutanoyl]-2-[(2E)-3-phenylprop-2-en-1-yl]-2,8-diazaspiro[4.5]decan-3-one
2-[(5-{[2-(2,5-dimethylphenoxy)propanamido]methyl}-1,3,4-oxadiazol-2-yl)sulfanyl]acetic acid
N-ethyl-5-[4-(2-methanesulfonylethyl)piperazine-1-carbonyl]pyrimidin-2-amine
methyl 4-(4-{[(cyclopropylmethyl)(oxolan-2-ylmethyl)amino]methyl}-5-methyl-1,3-oxazol-2-yl)benzoate
(4aS,7aR)-1-(3-methyl-4-oxo-3,4-dihydroquinazoline-7-carbonyl)-4-propyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
8-[2-(5-amino-3-methyl-1H-pyrazol-1-yl)acetyl]-3-hexyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-[(3S,5S)-1-(3-ethoxypropanoyl)-5-(ethylcarbamoyl)pyrrolidin-3-yl]pyridine-3-carboxamide
N-(2,1,3-benzothiadiazol-5-ylmethyl)-N-methyl-1-(pyridin-2-yl)piperidine-3-carboxamide
N-(4-fluorophenyl)-1-[2-(1H-1,2,3,4-tetrazol-5-yl)benzoyl]piperidin-3-amine
N-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-1-(3-methoxypropanoyl)piperidine-2-carboxamide
(4aS,7aR)-N-tert-butyl-4-[(dimethylcarbamoyl)methyl]-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
6-[(2E)-3-(2-fluorophenyl)prop-2-enoyl]-N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-6-azaspiro[2.5]octane-1-carboxamide
3-[(3,4-dimethoxyphenyl)methyl]-5-{[1-(propan-2-yl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}-1,2,4-oxadiazole
ethyl 3-[(3-chlorophenyl)methyl]-1-methanesulfonylpiperidine-3-carboxylate
methyl[(1-methyl-1H-indol-5-yl)methyl][2-(1H-pyrazol-1-yl)ethyl]amine
1-{5-[(2H-1,3-benzodioxol-5-yloxy)methyl]-1H-pyrazole-3-carbonyl}azonane
1-cyclobutanecarbonyl-4-[4-cyclopropyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
1-(3-fluorophenyl)-3-{1-[1-(2-methoxyacetyl)piperidin-4-yl]-1H-pyrazol-5-yl}urea
3-{[1-(3-methyl-1H-pyrazole-5-carbonyl)piperidin-4-yl]methyl}benzoic acid
2-[(3-methoxyphenyl)methyl]-8-(2-methylfuran-3-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
2-[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]-7-(2-methoxyphenyl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
2-(3-butyl-5-oxo-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-1-yl)-N-[(dimethyl-1,2-oxazol-4-yl)methyl]acetamide
2-(3-cyclopentyl-5-{2-[(propan-2-yl)amino]pyrimidin-5-yl}-1H-1,2,4-triazol-1-yl)ethan-1-ol
(3S,4R)-1-[2-(ethylamino)pyrimidine-5-carbonyl]-4-(3-methylthiophen-2-yl)piperidin-3-ol
1-{[3-(2-fluoro-4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-1,4-diazepan-5-one
3-hydroxy-5-{6-[(pyridin-3-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}benzoic acid