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N-(2-{[6-methyl-2-(pyridin-3-yl)pyrimidin-4-yl]amino}ethyl)acetamide
4-[4-(3-methylphenyl)-1H-pyrazol-5-yl]-1-(piperidine-4-carbonyl)piperidine
1-methyl-N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl](isoquinolin-5-ylmethyl)methylamine
N-(3-acetamidophenyl)-3-[(2S)-2-(hydroxymethyl)pyrrolidin-1-yl]propanamide
1-(2-methyl-1-benzofuran-5-carbonyl)-4-(pyridin-2-ylmethyl)-1,4-diazepane
[(3S,5R)-5-[(dimethylamino)methyl]-1-[6-(3-fluorophenyl)pyridine-3-carbonyl]piperidin-3-yl]methanol
8-[(5-butylthiophen-2-yl)methyl]-2-(2-hydroxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
N-[(2-chlorophenyl)methyl]-2-methoxy-2-methyl-N-(prop-2-en-1-yl)propanamide
3-(3,4-difluorophenyl)-N-[(4-hydroxyazepan-4-yl)methyl]propanamide
3-{[(1-{3-methyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}piperidin-4-yl)oxy]methyl}pyridine
3-{2-[(1R,5R)-3-(pyrazin-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethyl}-2,3-dihydro-1,3-benzoxazol-2-one
4-(1-{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl}azetidin-3-yl)morpholine
N-[4-(3-acetylphenyl)phenyl]-6-hydroxy-1,4-oxazepane-4-carboxamide
1-{[2-(ethylamino)pyrimidin-5-yl]methyl}-4-phenoxypiperidine-4-carboxylic acid
methyl[(4-methylphenyl)methyl]{[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
2-(2-{1-[(dimethyl-1,2-oxazol-4-yl)sulfonyl]piperidin-3-yl}-1H-imidazol-1-yl)acetamide
2-(4-chloro-3-fluorophenyl)-6-methylpyridine-3-carboxamide
1,3-dimethyl-5-[({1-methyl-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)methyl]-2,3-dihydro-1H-1,3-benzodiazol-2-one
1-{[4-(benzyloxy)phenyl]methyl}-4-(1H-imidazol-1-ylmethyl)piperidin-4-ol
2-(2-chlorophenoxy)-1-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-1-yl]ethan-1-one
8-methyl-N-(1-phenylcyclopropyl)-2-propyl-2,8-diazaspiro[4.5]decane-3-carboxamide
[(3R,4R)-1-(6-ethyl-4-methylquinolin-2-yl)-4-{[(2-methoxyethyl)(methyl)amino]methyl}pyrrolidin-3-yl]methanol
2-{5-[3-(2-fluorophenyl)-1H-pyrazole-5-carbonyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-1-yl}ethan-1-ol
4-methyl-N-{2-[3-(4-methylphenoxymethyl)piperidin-1-yl]-2-oxoethyl}-1,2,5-oxadiazole-3-carboxamide
2-(dimethylamino)-2-(3-fluorophenyl)-N-[2-(2-methoxyphenoxy)ethyl]acetamide
(4aS,8aR)-6-(1-methyl-1H-pyrazole-4-carbonyl)-1-[2-(thiophen-2-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
N-[3-(furan-2-yl)propyl]-2,7-dioxo-1,3-diazepane-4-carboxamide
4-[1-(2-methoxyphenyl)piperidin-4-yl]-1-methylpiperazine-2-carboxylic acid
{[3-(2-chlorophenyl)-1-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}[3-(morpholin-4-yl)propyl]amine
(2R)-2-[5-(2-ethylphenyl)-4-phenyl-1H-imidazol-1-yl]propanamide
1-[(2-fluorophenyl)methyl]-5-(3-{imidazo[1,2-a]pyridin-2-yl}-1,2,4-oxadiazol-5-yl)piperidin-2-one
1-{5H,6H-benzo[h]quinazolin-2-yl}-5-cyclopropyl-N-[1-(6-methylpyridin-2-yl)propan-2-yl]-1H-pyrazole-4-carboxamide
N-{[1-(hydroxymethyl)cyclopentyl]methyl}-3-(3-methoxyphenyl)-N-methyl-1H-pyrazole-5-carboxamide
3-(3-chloro-1,2-oxazol-5-yl)-1-[4-(3-fluorophenoxy)piperidin-1-yl]propan-1-one
3-[2-(6-methoxynaphthalen-2-yl)morpholin-4-yl]-1-(pyrrolidin-1-yl)propan-1-one
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-2-(1,2,3,4-tetrahydroisoquinolin-2-yl)acetamide
1-[4-(2,6-dimethylpyridin-4-yl)piperazin-1-yl]-2-(morpholin-2-yl)ethan-1-one
N-(4-methoxy-2-methylphenyl)-4-{2-[(3-methoxyphenyl)carbamoyl]ethyl}piperidine-1-carboxamide
{2-[3-(naphthalen-1-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-2-oxoethyl}urea
[(3R,4R)-4-{[4-(hydroxymethyl)piperidin-1-yl]methyl}-1-(2-methyl-5-propylpyrimidin-4-yl)pyrrolidin-3-yl]methanol
2-cyclopentyl-N-cyclopropyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-amine
N-[2-chloro-5-(pyrrolidine-1-carbonyl)phenyl]-1-oxa-7-azaspiro[3.5]nonane-7-carboxamide
2-(3-cyclopropyl-5-{2-[4-(methylsulfamoyl)phenyl]ethyl}-1H-1,2,4-triazol-1-yl)acetic acid
5,6-dimethyl-2-oxo-N-[(2-phenyl-1,3-oxazol-4-yl)methyl]-1,2-dihydropyridine-3-carboxamide
N-[1-(cyclohex-1-en-1-yl)ethyl]-5,7-dimethyl-[1,2,4]triazolo[4,3-a]pyrimidine-3-carboxamide
2-(methoxymethyl)-6-methyl-4-oxo-1-(3-phenylpropyl)-N-[2-(pyridin-2-yl)ethyl]-1,4-dihydropyridine-3-carboxamide
4-[3-(4,5-dimethyl-1H-pyrazol-3-yl)propanoyl]-1-(4-methylphenyl)piperazin-2-one
2-{1-[3-(propan-2-yl)-1,2-oxazole-5-carbonyl]pyrrolidin-2-yl}pyridine
2-ethyl-1-[(1-ethylpyrrolidin-2-yl)methyl]-6-methyl-3-{1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl}-1,4-dihydropyridin-4-one