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N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-1-[2-(methylsulfanyl)pyrimidin-4-yl]piperidin-4-amine
5-[3-(oxolan-2-yl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]-1-phenyl-1H-1,2,3,4-tetrazole
3-(2H-1,3-benzodioxol-5-yl)-1-[4-(furan-2-ylmethyl)-3-(2-hydroxyethyl)piperazin-1-yl]propan-1-one
2-benzyl-8-(6-methyl-2-propylpyrimidin-4-yl)-2,8-diazaspiro[4.5]decan-3-one
2-(2,3-dihydro-1-benzofuran-7-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
1-{4-[(4-chlorophenyl)methyl]-4-(hydroxymethyl)piperidin-1-yl}-3-(4-methoxyphenyl)propan-1-one
4-[4-fluoro-2-(trifluoromethyl)phenyl]-6-(4-methylpiperazin-1-yl)pyrimidin-2-amine
N-[2-(1H-imidazol-1-yl)ethyl]-2-[2-(1-methyl-1H-imidazol-4-yl)ethyl]-1-oxo-2,3-dihydro-1H-isoindole-4-carboxamide
N-[2-(azepan-1-yl)ethyl]-1-(2-ethoxyethyl)-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
5-(3,4-dimethoxyphenyl)-3-methyl-1-phenyl-1H,4H-pyrazolo[3,4-d]imidazole
(3aR,6aS)-5-{[4-methoxy-2-methyl-5-(propan-2-yl)phenyl]methyl}-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-(3,4-dihydro-2H-1-benzopyran-6-ylmethyl)-4-(oxolan-3-yl)-1H-1,2,3-triazole
1-{[1-(2-chlorophenyl)-1H-pyrazol-4-yl]methyl}-3-(piperidin-1-ylmethyl)pyrrolidin-3-ol
N-{[2-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}-1,9-dioxaspiro[5.5]undecan-4-amine
2-[2-fluoro-4-(pyrrolidin-1-ylmethyl)phenoxy]-6-(pyrrolidine-1-carbonyl)pyrazine
6-{3-[3-(4-ethylpiperazin-1-yl)propyl]-2-oxo-1-oxa-3,8-diazaspiro[4.5]decan-8-yl}pyridine-2-carbonitrile
N-{[2-(2-methoxyphenoxy)pyridin-3-yl]methyl}cyclopentanamine
(2R,3R,6R)-N,N-dimethyl-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carboxamide
2-{[1-(2-methylpropyl)-5-oxopyrrolidin-3-yl]formamido}-N-(1,3-thiazol-2-yl)acetamide
N-(3-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}propyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxamide
5-[1-(2,1,3-benzothiadiazol-5-ylmethyl)piperidin-4-yl]-3-[2-(4-methoxyphenyl)ethyl]-5-methylimidazolidine-2,4-dione
N-(2-methylphenyl)-1-{2-[(thiophen-2-ylmethyl)amino]ethyl}-1H-1,2,3-triazole-4-carboxamide
N-(1H-indol-6-ylmethyl)-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-amine
1-benzoyl-N-[1-(1-methyl-1H-pyrazol-5-yl)propyl]piperidin-4-amine
(2S)-2-hydroxy-4-({6-methylimidazo[1,2-a]pyridin-2-yl}formamido)butanoic acid
8-[2-(ethylamino)pyrimidine-5-carbonyl]-2-(2-methoxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
{4-[(E)-2-phenylethenyl]pyridin-2-yl}methanol
1-[4-({[(3-chlorophenyl)methyl]amino}methyl)phenoxy]-3-(4-methylpiperazin-1-yl)propan-2-ol
N-[2-(1H-indol-3-yl)ethyl]-4-(4-methylphenoxy)piperidine-4-carboxamide
5-methyl-N-[1-(morpholine-4-carbonyl)azepan-3-yl]pyrazine-2-carboxamide
3-benzyl-1-methyl-8-{[2-(trifluoromethyl)phenyl]methyl}-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-(1,4-oxazepan-6-ylmethyl)-7H-pyrrolo[2,3-d]pyrimidin-4-amine
N,N-dimethyl-5-{4-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}pyridin-2-amine
5-{5H,6H,7H,8H-imidazo[1,5-a]pyrazine-7-carbonyl}-N-(propan-2-yl)pyrimidin-2-amine
2-methoxy-6-({methyl[(5-methyl-1H-1,3-benzodiazol-2-yl)methyl]amino}methyl)phenol
2-[1-cyclopentyl-4-(2,2-diphenylethyl)piperazin-2-yl]ethan-1-ol
5-fluoro-6-methyl-2-[2-({methyl[(3-methylpyridin-2-yl)methyl]amino}methyl)phenyl]-3,4-dihydropyrimidin-4-one
3-{3,9-diazaspiro[5.5]undecane-3-carbonyl}-2-methyl-N-(pyridin-3-ylmethyl)aniline
N-[4-(5-methylfuran-3-amido)phenyl]-1H-pyrrole-2-carboxamide
1-[(2,3-difluoro-6-methoxyphenyl)methyl]piperidine-4-carbonitrile
8-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}-3-(pentan-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-(4-{[(butan-2-yl)(pyridin-3-ylmethyl)amino]methyl}phenyl)acetamide
2-ethyl-6-methyl-1-[2-(piperidin-1-yl)ethyl]-3-{1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl}-1,4-dihydropyridin-4-one
5-{6-chloro-2-methylimidazo[1,2-a]pyridin-3-yl}-3-(oxolan-3-yl)-1,2,4-oxadiazole
6-(4-methoxy-3,5-dimethylphenyl)-N-{[1-(2-methylpropyl)pyrrolidin-3-yl]methyl}pyridine-3-carboxamide
methyl[1-(3-methyl-1,2,4-oxadiazol-5-yl)ethyl][(6-methylquinolin-5-yl)methyl]amine
ethyl 2-({3-[(3,4-dimethylphenyl)amino]piperidine-1-carbonyl}amino)acetate
1-(2,3-dihydro-1,4-benzodioxin-6-yl)-2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazole
(3S,4S)-3-hydroxy-N-(4-methanesulfonylphenyl)-4-(morpholin-4-yl)pyrrolidine-1-carboxamide
N-[(5-chlorothiophen-2-yl)methyl]-5-[3-(trifluoromethyl)phenoxymethyl]-1,2-oxazole-3-carboxamide