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5-[3-(oxolan-3-yl)-1-(pyridin-3-yl)-1H-1,2,4-triazol-5-yl]pyridine-2-carbonitrile
1-(4-{[2-(diethylamino)-2-(furan-2-yl)ethyl]amino}-2-methyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl)ethan-1-one
N-(3-methylcinnolin-5-yl)-2-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carboxamide
N-(2,3-dihydro-1H-inden-2-yl)-3-(8-methoxy-2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)propanamide
5-methyl-1-(2-methylphenyl)-4-[(6-methylquinolin-5-yl)methyl]piperazin-2-one
8-fluoro-N-methyl-N-[1-(pyridin-3-yl)propyl]quinoline-2-carboxamide
5,6-dimethyl-3-[4-(thiomorpholin-4-yl)piperidine-1-carbonyl]-1,2-dihydropyridin-2-one
3-{[(3S,4R)-3-hydroxy-4-(hydroxymethyl)piperidin-1-yl]methyl}-5,6,7-trimethoxy-1,2-dihydroquinolin-2-one
ethyl 2-[2-({4-cyclopentyl-3-oxo-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-11-yl}amino)ethyl]-1,3-thiazole-4-carboxylate
N-[2-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-6-methoxy-3-methyl-1-benzofuran-2-carboxamide
N-cyclopentyl-2-(3-methoxy-2-oxo-1,2-dihydropyridin-1-yl)-N-[(5-methylthiophen-2-yl)methyl]acetamide
5-{[4-(4-hydroxybut-1-yn-1-yl)phenyl]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylic acid
methyl 6-cyclopentyl-2-{[(4-fluorophenyl)methyl]sulfamoyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
2-[1-benzyl-5-(1-cyclopentyl-5-oxopyrrolidin-3-yl)-1H-1,2,4-triazol-3-yl]acetamide
(oxolan-2-ylmethyl)(pyridin-2-ylmethyl){[4-(2H-1,2,3,4-tetrazol-5-yl)phenyl]methyl}amine
5-({1-[3-(2-oxopiperidin-1-yl)propanoyl]pyrrolidin-3-yl}methyl)-1,2-dihydropyridin-2-one
(3S,4R)-4-(2,3-dimethoxyphenyl)-1-[(3-methyl-1H-1,2,4-triazol-5-yl)methyl]pyrrolidine-3-carboxylic acid
2-{2-methylimidazo[1,2-a]pyridin-3-yl}-N-{2-[3-(trifluoromethyl)phenyl]ethyl}acetamide
5-[(2R,3R,6R)-3-(3,5-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]-3,4-dihydropyrimidin-4-one
4-({6-[4-(1H-pyrazol-5-yl)phenyl]pyridin-3-yl}methyl)morpholine
1-(1-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}cyclopentyl)pyrrolidine
3-{[(1-ethylcyclopropyl)amino]methyl}-1-[(2-fluoro-5-methoxyphenyl)methyl]-3-hydroxypiperidin-2-one
N-cyclopentyl-2-({[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}amino)propanamide
2-[4-cyclohexyl-3-(2-hydroxyethyl)piperazin-1-yl]-1,3-thiazole-4-carboxamide
N-(4-fluorophenyl)-1-(quinolin-5-ylmethyl)piperidin-3-amine
{[2-(4-methoxyphenyl)-7-methylquinolin-3-yl]methyl}(methyl)(1,2-oxazol-5-ylmethyl)amine
(2R,3S,6R)-3-(2,3-difluorophenyl)-5-(pyrrolidine-1-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-[(2,3-dimethoxyphenyl)methyl]-[1,2,3,4]tetrazolo[1,5-a]pyridine-7-carboxamide
2-(methoxymethyl)-5-{[4-(2-methoxyphenyl)-3,3-dimethylpiperazin-1-yl]methyl}pyrimidine
5-methyl-1-(pyridin-2-yl)-N-[(1r,4r)-4-(4H-1,2,4-triazol-4-yl)cyclohexyl]-1H-pyrazole-4-carboxamide
N-(3-chlorophenyl)-2-[2-(2-oxopyrrolidin-1-yl)ethyl]piperidine-1-carboxamide
2-(furan-2-yl)-5-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}pyrimidine
(1R,9S)-11-[2-(trimethyl-1H-pyrazol-1-yl)acetyl]-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-6-one
N-[(2,6-difluoro-3-methoxyphenyl)methyl]-3-ethyl-4-methyl-1H-pyrazole-5-carboxamide
(4S)-1-{[6-(dimethylamino)pyridin-3-yl]methyl}-3,3,4-trimethylpiperidin-4-ol
1-{4-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-3-(1H-1,2,3,4-tetrazol-1-yl)propan-1-one
5-{3-oxo-2-[2-(pyridin-2-yl)ethyl]-2,9-diazaspiro[5.5]undecane-9-carbonyl}pyridine-2-carbonitrile
3-(3-methylphenyl)-N-{2-[(pyridin-3-yl)amino]ethyl}-1H-pyrazole-4-carboxamide
{5-[6-(cyclopentylamino)-1H-pyrrolo[2,3-b]pyridin-4-yl]-1H-1,3-benzodiazol-2-yl}methanol
4-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)pyrrolidin-1-yl]-4-oxobutane-1-sulfonamide
4-fluoro-N-(2-{imidazo[2,1-b][1,3]thiazol-6-ylformamido}ethyl)benzamide
N-[(3S,4R)-1-(cyclobutylmethyl)-4-(5-methylfuran-2-yl)pyrrolidin-3-yl]acetamide
1-[3-(4-chlorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-4-(1H-pyrazol-4-yl)butan-1-one
2-{3-[3-(4-fluorophenyl)oxolan-3-yl]-1,2,4-oxadiazol-5-yl}-1,4-dihydroquinolin-4-one
1-(4-methanesulfonylpiperazin-1-yl)-3-(4,5,6,7-tetrahydro-1H-indazol-3-yl)propan-1-one
(4aS,7aR)-1-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]-4-propanoyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-methyl-2-(methylamino)-N-(oxolan-2-ylmethyl)-N-(pyridin-2-ylmethyl)-1,3-thiazole-5-carboxamide
(4aR,8aS)-1-[2-(3,4-dimethoxyphenyl)ethyl]-6-[(2E)-3-(thiophen-2-yl)prop-2-enoyl]-decahydro-1,6-naphthyridin-2-one
1-(2-methoxyacetyl)-N-{2-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}piperidine-4-carboxamide
3-{1-[1-(2-fluorobenzoyl)piperidin-4-yl]-1H-pyrazol-5-yl}-1-(2-methoxyphenyl)urea