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1-(3,5-dimethylphenyl)-4-[(2S)-2-hydroxy-3-phenylpropanoyl]piperazin-2-one
[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl](methyl)(3,3,3-trifluoro-2-methylpropyl)amine
(1S,2S)-2-[4-(5-propyl-1,2-oxazole-3-carbonyl)piperazin-1-yl]cyclohexan-1-ol
ethyl 4-(1-{[5-(hydroxymethyl)furan-2-yl]methyl}piperidin-3-yl)piperazine-1-carboxylate
3-methyl-4-{1-methyl-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}piperazin-2-one
(3S,4S)-4-({6-cyclopentyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)-1-(propan-2-yl)pyrrolidin-3-ol
7-{[(4aS,8aR)-4a-(hydroxymethyl)-decahydro-1,6-naphthyridin-6-yl]methyl}-2-methyl-5H-[1,3]thiazolo[3,2-a]pyrimidin-5-one
2-{5-[2-amino-4-(trifluoromethyl)pyrimidin-5-yl]-1-benzyl-1H-1,2,4-triazol-3-yl}acetamide
8-chloro-N-{1-[2-(methylsulfanyl)ethyl]piperidin-4-yl}quinoline-2-carboxamide
N-{[3-(pyrrolidin-1-yl)phenyl]methyl}-2-(1,2,3,4-tetrahydroisoquinolin-2-yl)propanamide
2-{4-[4-methyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}phenol
4-[4-(methoxymethyl)-5-methyl-1,2-oxazole-3-carbonyl]-3-methyl-1-[(4-methylphenyl)methyl]piperazin-2-one
2-[4-(1H-imidazol-2-yl)piperidin-1-yl]-4-(trifluoromethyl)pyridine
1-{2-methyl-3-[(pyridin-2-ylmethyl)amino]benzoyl}azetidin-3-ol
1-[3-(3-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-2-(piperidin-1-yl)ethan-1-one
4-[(2-chlorophenyl)methyl]-1-(1H-indol-3-ylmethyl)-1,4-diazepan-5-one
3-{[(1,2-dimethyl-1H-imidazol-5-yl)methyl](prop-2-en-1-yl)amino}-3-methyl-1λ6-thiolane-1,1-dione
2-methyl-5-({5-propanoyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}carbonyl)-1,4-dihydropyridin-4-one
N-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-N-methyl-1-(oxolan-2-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
N-{[4-(4-methylphenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}pyridazine-3-carboxamide
5-(dimethylamino)-2-[2-(2-ethyl-1H-imidazol-1-yl)ethyl]-2,3-dihydropyridazin-3-one
{[2-(morpholin-4-yl)pyridin-3-yl]methyl}(pyridin-2-ylmethyl)amine
diphenyl[1-(1H-pyrrole-3-carbonyl)piperidin-4-yl]methanol
2-(1-{[5-(1,5-dimethyl-1H-pyrrol-2-yl)-1,3,4-oxadiazol-2-yl]methyl}pyrrolidin-2-yl)-1,3-benzothiazole
2-(5-amino-1,3,4-thiadiazol-2-yl)-1-{2-methyl-4-[(prop-2-en-1-yl)amino]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl}ethan-1-one
N,N,4-trimethyl-3-{[methyl(2-methylpropyl)carbamoyl]methyl}-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
2-[4-(1-cyclohexanecarbonylpyrrolidine-2-carbonyl)piperazin-1-yl]-N-(propan-2-yl)acetamide
(1S,4S)-5-(5-chloro-3-methyl-1H-indole-2-carbonyl)-2-(2-fluorophenyl)-2,5-diazabicyclo[2.2.1]heptan-3-one
4-(3-hydroxy-3-methylbutyl)-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}benzamide
N-[3-(methylsulfanyl)butyl]-N-(pyridin-3-ylmethyl)cyclopropanamine
6-{2-cyclopropyl-3-oxo-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}pyridine-3-carbonitrile
3-{[(3aR,6aR)-2-methyl-octahydropyrrolo[3,4-c]pyrrol-3a-yl]formamido}-N-(2-ethylphenyl)propanamide
1-[2-benzyl-5-oxo-4-(2-phenylphenyl)piperazin-1-yl]propane-1,2-dione
6-[2-(3,4-dimethylphenoxy)ethyl]pyrazolo[1,5-a]pyrimidine-3-carbonitrile
N,N-dimethyl-2-[4-(3-methylthiophen-2-yl)-1H-1,2,3-triazol-1-yl]-2-phenylacetamide
3-[4-(thiophen-2-ylmethyl)piperazin-1-yl]-1,2-dihydropyrazin-2-one
4-(4-acetyl-4-phenylpiperidine-1-carbonyl)-1-oxaspiro[4.4]nonan-2-one
2-(3-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)pyrazine
(4aS,7aR)-1-(5-fluoropentyl)-4-(pyrimidin-2-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2,6,8-trimethyl-4-[3-(pyridin-3-yloxy)azetidine-1-carbonyl]quinoline
(3aR,6aR)-2-methanesulfonyl-5-(5-propyl-1,3,4-thiadiazol-2-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
4-{[1-(2-methoxyacetyl)piperidin-4-yl]oxy}-N-methyl-N-[(1-methylpiperidin-3-yl)methyl]benzamide
6-{pyrazolo[1,5-a]pyridin-7-yl}pyridine-2-carboxamide
3-oxo-N-[1-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-yl]-3,4-dihydro-2H-1,4-benzoxazine-7-carboxamide
3-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-1-{4-[(1-methylpiperidin-4-yl)oxy]phenyl}urea
2-[(4-methoxyphenyl)methyl]-N-(oxan-4-yl)-1,3-benzoxazole-6-carboxamide
1-[(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]butan-1-one
methyl 1-{[6-(azocane-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}piperidine-4-carboxylate
4-[(4-methylphenyl)methyl]-11-(pyrrolidin-1-yl)-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
2-(piperidine-1-carbonyl)-7-(prop-2-en-1-yl)-6-(thiophen-2-yl)-7H,8H-imidazo[1,2-a]pyrazin-8-one