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1-methyl-N-(2-phenylethyl)-N-{[1-(propan-2-yl)-1H-imidazol-5-yl]methyl}piperidin-4-amine
1-methyl-4-{5-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}piperazine
1-(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-carbonyl)-4-(pyridin-4-ylmethyl)-1,4-diazepane
2-{4-[5-(2-methoxy-2-phenylacetamido)-1H-pyrazol-1-yl]piperidin-1-yl}-N,N-dimethylacetamide
2-acetyl-8-[2-(3,4-dimethylphenyl)acetyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
N-{1-[(4-chlorophenyl)methyl]piperidin-3-yl}cyclopropanecarboxamide
2-fluoro-N-[(5-phenyl-1,2-oxazol-3-yl)methyl]-5-sulfamoylbenzamide
3-ethyl-1-(6-methyl-4-oxo-1,4-dihydropyridine-3-carbonyl)piperidine-3-carboxylic acid
2-[3-(dimethylamino)propyl]-9-[6-methyl-2-(methylamino)pyrimidin-4-yl]-2,9-diazaspiro[5.5]undecan-3-one
N-methyl-3-[(3-oxo-3,4-dihydro-2H-1,4-benzothiazin-4-yl)methyl]-1,2,4-oxadiazole-5-carboxamide
2-{4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-1-yl}-N-(propan-2-yl)acetamide
N-[2-(4-methylpiperazin-1-yl)propyl]-4-(propan-2-yl)pyrimidin-2-amine
N-{[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]methyl}-2,2,6,6-tetramethylpiperidin-4-amine
1-[4-(3,4-dichlorophenyl)piperazin-1-yl]-2-(pyridin-3-yl)ethan-1-one
(1-{[3-(4-fluorophenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}piperidin-3-yl)methanol
1-(cyclohexylmethyl)-5-[3-(morpholin-4-ylmethyl)-1,2,4-oxadiazol-5-yl]piperidin-2-one
1-(3-chloropyridin-2-yl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
1-[(1-methyl-1H-pyrazol-4-yl)methyl]-3-{5-[2-(morpholin-4-yl)ethyl]-1,3,4-thiadiazol-2-yl}urea
(3R,5S)-1-[(3,4-dimethoxyphenyl)methyl]-N-[2-(dimethylamino)ethyl]-5-(3-fluorophenoxymethyl)piperidine-3-carboxamide
N-{[5-(2H-1,3-benzodioxol-5-yl)-1,2,4-oxadiazol-3-yl]methyl}-3-(4-methyl-1,3-thiazol-5-yl)propanamide
N-({5-cyclohexyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-2-(ethylamino)pyrimidine-5-carboxamide
6-{1-[3-(trifluoromethyl)-1H-pyrazole-5-carbonyl]piperidin-4-yl}pyrimidin-4-ol
3-(2-methoxyphenyl)-1-(3-methoxypropyl)-3-[2-oxo-2-(3-oxo-4-phenylpiperazin-1-yl)ethyl]pyrrolidine-2,5-dione
N-cyclopropyl-1-[2-(4-methoxyphenyl)ethyl]-5-(pyridine-4-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
7-[(2,3-difluorophenyl)methyl]-2-methanesulfonyl-2,7-diazaspiro[4.5]decane
2-{2-[(4-hydroxy-4-methylazepan-1-yl)methyl]-4-(pyrazin-2-yl)phenoxy}acetic acid
4-{2-[4-(1H-imidazol-2-yl)-1H-1,2,3-triazol-1-yl]ethyl}benzene-1-sulfonamide
N-{[5-(benzylsulfanyl)-4-(4-methoxyphenyl)-4H-1,2,4-triazol-3-yl]methyl}-3,5-dimethoxybenzamide
2-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-7-[(2-fluorophenyl)methyl]-2,7-diazaspiro[4.5]decane
4-(5-{[4-(cyclohexylmethyl)-3-(2-hydroxyethyl)piperazin-1-yl]methyl}thiophen-2-yl)-2-methylbut-3-yn-2-ol
2-amino-N-[3-(2-methoxybenzamido)phenyl]-4-methylpyrimidine-5-carboxamide
4-(2,3-dihydro-1H-inden-5-yloxy)-1-(pyrazin-2-yl)piperidine-4-carboxylic acid
N-[2-(1H-1,3-benzodiazol-2-yl)ethyl]-2-(pyridin-3-yl)pyrimidine-5-carboxamide
N-benzyl-5-(cyclopentylamino)-N,1-dimethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
6-{3-[1-(4-fluorobutyl)-1H-pyrazol-3-yl]phenyl}-N,N-dimethylpyrimidin-4-amine
1-[(2-fluorophenyl)methyl]-4-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidine
2-(2-{[2-(1-methyl-1H-1,3-benzodiazol-2-yl)pyrrolidin-1-yl]methyl}phenoxy)ethan-1-ol
3-{[(3S)-3-hydroxypyrrolidin-1-yl]methyl}-1H,2H,6H,7H,8H-cyclopenta[g]quinolin-2-one
N-{[4-hydroxy-1-(1H-imidazol-4-ylmethyl)azepan-4-yl]methyl}-2-phenoxyacetamide
1-(4-chloro-1,3-dimethyl-1H-pyrazole-5-carbonyl)-4-(2-methoxyphenoxy)piperidine
5-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-3-(2-methylphenyl)-1,2,4-oxadiazole
4-methyl-N-[2-(piperidin-1-yl)-2-(pyridin-3-yl)ethyl]-2-(propan-2-yl)-1,3-thiazole-5-carboxamide
2-(4-chlorophenyl)-5-(4H-1,2,4-triazol-4-yl)-1,3-benzoxazole
1-[3-(hydroxymethyl)quinolin-2-yl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
1-(oxan-4-yl)-N-[4-(1,3-thiazol-4-yl)phenyl]piperidine-3-carboxamide
N-(3-chloro-4-methoxyphenyl)-3-[1-(furan-3-ylmethyl)piperidin-3-yl]propanamide
(3aS,6aS)-2-[(2,4-dimethoxyphenyl)methyl]-5-(dimethylcarbamoyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-(1-benzothiophen-2-ylmethyl)-1-ethyl-N-methyl-3-(morpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
3-[2-(2,6-difluorophenyl)ethyl]-1-(3-methyl-1,2-oxazole-5-carbonyl)piperidine
(2R,6S)-4-(1-{5-cyclopropyl-1-[4-(5-methylfuran-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carbonyl}piperidin-4-yl)-2,6-dimethylmorpholine