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1-(2-ethyl-4-methyl-1,3-oxazole-5-carbonyl)-4-[(2-methylphenyl)sulfanyl]piperidine
2-fluoro-6-{1H-pyrazolo[3,4-b]pyridin-1-yl}benzamide
(2S,4R)-N-(2-methyl-1,3-benzothiazol-5-yl)-4-(pyridin-2-ylsulfanyl)-1-{[4-(trifluoromethoxy)phenyl]methyl}pyrrolidine-2-carboxamide
2-{[(2-chlorophenyl)methyl]sulfanyl}-N-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]acetamide
3-methoxy-N-methyl-N-{[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}propanamide
[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl][(5-methyl-1,2,4-oxadiazol-3-yl)methyl](propan-2-yl)amine
1-(1H-1,3-benzodiazol-2-ylmethyl)-4-(1H-pyrrole-3-carbonyl)-1,4-diazepan-6-ol
3-[2-fluoro-5-(4H-1,2,4-triazol-4-yl)phenyl]-1-[2-(morpholin-4-yl)ethyl]urea
3-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)-N-{3-[(pyridin-3-yl)amino]propyl}propanamide
N-{2-[3-(thiomorpholin-4-ylmethyl)phenoxy]propyl}pyridine-3-carboxamide
N-[(5-chloro-1H-1,3-benzodiazol-2-yl)methyl]-2-methoxy-N-methyl-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
1-(3-methoxyphenyl)-4-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}piperazin-2-one
2-(2-methoxyethyl)-9-(2-phenylpropanoyl)-2,9-diazaspiro[5.5]undecan-3-one
2-cyclopropanecarbonyl-8-[(2,5-difluorophenyl)methyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
1-{[2-(4-fluoro-3-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(pyrrolidine-1-carbonyl)piperidine
1-(1H-imidazol-2-ylmethyl)-8-[8-(trifluoromethyl)quinolin-4-yl]-1,8-diazaspiro[4.5]decane
2-[3-(3-hydroxy-1,2-oxazol-5-yl)propanamido]-N-[(3-methylphenyl)methyl]benzamide
N-ethyl-N-[(3R,4R)-4-hydroxy-1,1-dioxo-1λ6-thiolan-3-yl]-3-methylfuran-2-carboxamide
2-({3-[4-(cyclopropylmethyl)-3-(2-hydroxyethyl)piperazine-1-carbonyl]phenyl}amino)acetic acid
7-(2-methylphenyl)-4-(pyridin-3-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-[(2S)-2-{4-[(4-chlorophenyl)methyl]-4-(hydroxymethyl)piperidine-1-carbonyl}pyrrolidin-1-yl]ethan-1-one
1-{1-[(2,4-difluorophenyl)methyl]piperidin-3-yl}-4-(4-fluorophenyl)piperazine
1-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-5-methyl-5-phenylpiperidin-2-one
N-(2-methyl-4,5,6,7-tetrahydro-1,3-benzothiazol-4-yl)-3-(2-oxo-2,3-dihydro-1H-1,3-benzodiazol-1-yl)propanamide
N-[4-methoxy-2-(2-methylpropanamido)phenyl]-1H-indole-3-carboxamide
1-[7-(hydroxymethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(naphthalen-2-yloxy)propan-1-one
4-(4-cyclohexylpiperazine-1-carbonyl)-1-(pyridin-4-ylmethyl)pyrrolidin-2-one
(3aR,7aS)-5-methyl-2-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]-2,3,3a,4,7,7a-hexahydro-1H-isoindole
N-[(3S,4R)-1-[2-(methylsulfanyl)pyrimidin-4-yl]-4-(propan-2-yl)pyrrolidin-3-yl]acetamide
1-{[2-(7-methoxy-2H-1,3-benzodioxol-5-yl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazine
N-(1-{4-[3-(pyrazin-2-yl)-1H-pyrazol-1-yl]phenyl}ethyl)acetamide
5-{4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepane-1-carbonyl}-N-methylpyrimidin-2-amine
(3R,4S)-4-(5-methylfuran-2-yl)-1-(thiophene-2-sulfonyl)pyrrolidin-3-amine
1-(piperidin-1-yl)-2-{4-[4-(1H-pyrazol-3-yl)benzoyl]piperazin-1-yl}ethan-1-one
(4aS,8aR)-1-(4-hydroxybutyl)-6-(6-oxo-1,4,5,6-tetrahydropyridazine-3-carbonyl)-decahydro-1,6-naphthyridin-2-one
5-(propan-2-yl)-N-{[5-(thiophen-2-ylmethyl)-1,2,4-oxadiazol-3-yl]methyl}pyrazolo[1,5-a]pyrimidin-7-amine
1,5-dimethyl-4-{[4-(pyrrolidine-1-carbonyl)piperidin-1-yl]methyl}-1H-pyrrole-2-carbonitrile
8-[2-(dimethylamino)-6-methylpyrimidin-4-yl]-2-(3-hydroxypropyl)-2,8-diazaspiro[5.5]undecan-3-one
N-[3-(1H-1,2,3-benzotriazol-1-yl)propyl]-5-(pyridin-4-yl)pyrazolo[1,5-a]pyrimidin-7-amine
1-(4-{[2-(1H-pyrazol-1-yl)ethyl]amino}-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl)ethan-1-one
1-[2-(3-fluorophenyl)ethyl]-N-[3-(4-methoxyphenyl)propyl]-6-oxopiperidine-3-carboxamide
1-({3-methoxy-2-[2-(morpholin-4-yl)ethoxy]phenyl}methyl)piperidine-3-carboxamide
dimethyl({[(3S,4R)-4-(propan-2-yl)-1-(quinoxalin-2-yl)pyrrolidin-3-yl]sulfamoyl})amine
4-{[2-(3-methoxypyridin-2-yl)phenyl]methyl}morpholine
3-({5-methyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}carbonyl)-1,2,5,6,7,8-hexahydroquinolin-2-one
(4aS,8aR)-6-(3-methyl-1H-pyrazole-5-carbonyl)-1-[2-(thiophen-2-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
5-{[4-(5-{[(3-chlorophenyl)methyl]sulfanyl}-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl)piperidin-1-yl]methyl}quinoline
4-[5-(ethoxymethyl)-3-phenyl-1H-1,2,4-triazol-1-yl]-3-methylpyridine
8-benzyl-3-(2-methoxyethyl)-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[(3R,4R)-3-hydroxy-1-[(3-methylquinoxalin-2-yl)methyl]piperidin-4-yl]pyridine-4-carboxamide