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methyl 4-(4-{[4-(3,6-dimethylpyrazin-2-yl)piperazin-1-yl]methyl}-5-methyl-1,3-oxazol-2-yl)benzoate
1-(2-methyl-6-oxo-1,6-dihydropyrimidine-5-carbonyl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
methyl 5-(1-methyl-3-propyl-1H-pyrazole-5-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylate
[3-(1H-imidazol-1-yl)propyl][(1-methyl-1H-imidazol-2-yl)methyl](pyridin-3-ylmethyl)amine
2-(dimethylamino)-1-{4-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]piperidin-1-yl}-2-(2-methylphenyl)ethan-1-one
3-({[(3-fluorophenyl)methyl]amino}methyl)-3-hydroxy-1-{[4-(propan-2-yl)phenyl]methyl}piperidin-2-one
4-{[4-(2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazol-1-yl)phenyl]methyl}morpholine
4-{5-hydroxy-1-oxa-9-azaspiro[5.5]undecane-9-carbonyl}-6-(2-methylpropyl)-1,2-dihydropyrimidin-2-one
ethyl({[3-(2-fluoro-4-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl})[(1-methyl-1H-pyrazol-4-yl)methyl]amine
N-(2-methoxyethyl)-N-(pyridin-3-ylmethyl)-2-(1,3-thiazol-4-yl)acetamide
1-[3-(3-fluorophenyl)propanoyl]-4-(2-methyl-1H-imidazol-1-yl)piperidine-4-carboxylic acid
3-[1-(6-aminopyridine-3-carbonyl)piperidin-3-yl]-N-methyl-N-[2-(pyridin-2-yl)ethyl]propanamide
4-[4-(3,6-dimethylpyrazin-2-yl)piperazine-1-carbonyl]-1,2-dihydroquinazolin-2-one
2-amino-3-ethyl-N-{[2-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}-3H-imidazo[4,5-b]pyridine-6-carboxamide
6-fluoro-N-methyl-2-oxo-N-{2-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}-1,2,3,4-tetrahydroquinoline-4-carboxamide
4-benzyl-3-ethyl-1-[3-(2-methylpropyl)-1,2-oxazole-5-carbonyl]-1,4-diazepan-5-one
N-methyl-N-[1-(1,2-oxazol-3-yl)ethyl]-3-(propan-2-yl)-1,2-oxazole-5-carboxamide
N-[(5-methylfuran-2-yl)methyl]-3-(1H-pyrazol-1-ylmethyl)benzamide
8-cycloheptanecarbonyl-2-(diethylamino)-1,3,8-triazaspiro[4.5]dec-1-en-4-one
5-[(2E)-but-2-en-1-yl]-N-methyl-N-[(1-methylpyrrolidin-2-yl)methyl]-1,3,4-oxadiazole-2-carboxamide
N-cyclopentyl-1-{1-[2-(2-methylphenyl)acetyl]piperidin-4-yl}-1H-1,2,3-triazole-4-carboxamide
N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}-2-(morpholin-4-yl)benzamide
2-(2-{[(3aS,6aS)-1-methyl-octahydropyrrolo[3,4-b]pyrrol-5-yl]methyl}-4-(pyridin-2-yl)phenoxy)acetic acid
N-(2,1,3-benzothiadiazol-5-ylmethyl)-N,1-dimethyl-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
1-[3-(3-ethyl-1,2,4-oxadiazol-5-yl)phenyl]-3-[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]urea
(1S,5R)-6-propyl-3-{1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carbonyl}-3,6-diazabicyclo[3.2.2]nonan-7-one
4-(1-{1-[(3-methylphenyl)methyl]-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-5-yl}ethyl)morpholine
2-amino-1-{4-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}ethan-1-one
2-[4-(oxan-4-yl)-1-(thiophen-2-ylmethyl)piperazin-2-yl]ethan-1-ol
[(1-cyclopentylpiperidin-3-yl)methyl][2-(piperidin-1-yl)ethyl](pyridin-4-ylmethyl)amine
2-(4-methoxyphenoxymethyl)-N-(prop-2-en-1-yl)-1,3-oxazole-4-carboxamide
N-[(1S,2R)-2-[(2,3-dihydro-1H-inden-2-yl)amino]cyclobutyl]-2-(morpholin-4-yl)pyrimidine-5-carboxamide
2-{[(3aS,6aS)-1-methyl-octahydropyrrolo[3,4-b]pyrrol-5-yl]methyl}-3,5-dimethoxybenzoic acid
5-{[benzyl(methyl)amino]methyl}-N-[(3-phenyl-1H-pyrazol-4-yl)methyl]-1,2-oxazole-3-carboxamide
2-[1-(2,2-dimethylpropyl)-3-oxopiperazin-2-yl]-N-ethyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]acetamide
1-{2-[7-(cyclobutylmethyl)-6-oxo-2,7-diazaspiro[4.5]decan-2-yl]-2-oxoethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-(3-hydroxypropyl)-1-({3-[(2-methylprop-2-en-1-yl)oxy]phenyl}methyl)piperidine-3-carboxamide
1-{[1-(2-fluorophenyl)-3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}piperidine-4-carbonitrile
1-(2H-1,3-benzodioxol-5-yl)-N-(1H-imidazol-2-ylmethyl)-N-methylpiperidin-4-amine
1-[(4S)-4-hydroxy-3,3,4-trimethylpiperidin-1-yl]-2-[2-(trifluoromethyl)phenyl]ethan-1-one
8-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
5-hydroxy-N-[4-methoxy-2-(2-methylpropanamido)phenyl]pyrazine-2-carboxamide
1-(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-carbonyl)-4-[2-(1H-pyrazol-1-yl)ethyl]piperidine
4-({4-methyl-5-[1-(6-methylpyridazin-3-yl)piperidin-3-yl]-4H-1,2,4-triazol-3-yl}methyl)morpholine
3-[3-(dimethyl-1H-1,2,4-triazol-1-yl)propyl]-1-[3-(piperidine-1-carbonyl)phenyl]urea
4-[(3-methylpyridin-4-yl)methyl]-2H,3H,4H-pyrido[3,2-b][1,4]oxazin-3-one
9-[2-(dimethylamino)-6-ethylpyrimidin-4-yl]-2-(2-methoxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
(3R,4R)-1-(2-fluorobenzenesulfonyl)-3-methyl-4-(oxan-4-yl)piperidin-4-ol
N-[2-(dimethylamino)ethyl]-N-(thiophen-3-ylmethyl)quinoline-2-carboxamide
4-{2-[(4-methylpiperazin-1-yl)methyl]phenoxy}benzamide