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2,6-dimethyl-N-[1-(1H-1,2,4-triazol-5-yl)ethyl]quinoline-3-carboxamide
2-amino-6-hydroxy-4-(isoquinolin-5-yl)-5H-indeno[1,2-b]pyridine-3-carbonitrile
4-{[5-chloro-1-methyl-3-(5-methyl-1,2-oxazol-3-yl)-1H-pyrazol-4-yl]methyl}-2-(pyridin-3-yl)morpholine
N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}-1-phenylcyclopentane-1-carboxamide
N-methyl-N-(1H-pyrazol-5-ylmethyl)-2-(2,3,6-trimethylphenoxy)acetamide
5-[1-(dimethyl-1,3-thiazole-5-carbonyl)piperidin-4-yl]-5-(pyridin-3-yl)-3-(thiophen-3-ylmethyl)imidazolidine-2,4-dione
2-[(dimethyl-1,3-thiazol-4-yl)formamido]-N-(propan-2-yl)acetamide
1-cyclobutanecarbonyl-N-[1-(5-methyl-1H-1,3-benzodiazol-2-yl)ethyl]piperidine-4-carboxamide
5-{4-methyl-3-[2-(3-methylthiophen-2-yl)-1H-imidazol-1-yl]phenyl}-1H-1,2,3,4-tetrazole
6-{2-[3-(1H-imidazol-1-yl)propyl]-3-oxo-2,9-diazaspiro[5.5]undecan-9-yl}pyridine-3-carboxylic acid
1-(4-{[1-(3,5-difluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]amino}piperidin-1-yl)ethan-1-one
1-butyl-5-(2-chloro-6-fluoro-3-methylphenyl)-1H-1,2,4-triazole
4-(3-hydroxy-3-methylbutyl)-N-[1-(6-methylpyridin-3-yl)ethyl]benzamide
4-[(1-ethyl-1H-imidazol-2-yl)methyl]-2-{[3-(trifluoromethyl)phenyl]methyl}morpholine
2-(1-benzofuran-2-yl)-2-[(1H-imidazol-2-ylmethyl)(methyl)amino]acetic acid
[(1R)-1-(4-methoxyphenyl)ethyl]({[2-(3-methylphenyl)pyrimidin-5-yl]methyl})amine
3-[(6-methoxypyrimidin-4-yl)amino]-1λ6-thiolane-1,1-dione
9-[2-(dimethylamino)-6-methylpyrimidin-4-yl]-2-(2-hydroxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
4-[2,2-bis(prop-2-en-1-yl)piperidine-1-carbonyl]-6-(propan-2-yl)pyrimidin-2-amine
2-(4-chloro-1-methyl-1H-pyrrole-2-carbonyl)-7-cyclohexyl-2,7-diazaspiro[4.5]decan-6-one
5-phenyl-N-{[1-(1H-pyrazol-1-ylmethyl)cyclopropyl]methyl}pyrazolo[1,5-a]pyrimidin-7-amine
N-cyclohexyl-N-[2-(ethylsulfanyl)ethyl]-5-methyl-1,2-oxazole-3-carboxamide
1-[(3,5-dimethylphenyl)methyl]-4-(2-fluoro-6-methoxybenzoyl)piperazin-2-one
(3S,4R)-1-(2,1,3-benzothiadiazol-5-ylmethyl)-4-(pyridin-4-yl)pyrrolidine-3-carboxylic acid
3-[(3S,7S,8aS)-3-[(benzyloxy)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(3,4-dimethylphenyl)urea
N-methyl-N-{[1-(2-methylphenyl)-1H-1,2,3,4-tetrazol-5-yl](phenyl)methyl}-1H-pyrazole-3-carboxamide
4,6-dimethyl-N-[2-(morpholin-4-yl)-2-(pyridin-3-yl)ethyl]-2-oxo-1,2-dihydropyridine-3-carboxamide
N-({5-[2-methyl-2-(piperidin-1-yl)propyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)cyclobutanecarboxamide
N,N-diethyl-1-[1-(thiophen-2-ylmethyl)piperidin-3-yl]-1H-1,2,3-triazole-4-carboxamide
9-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-3-oxa-9-azaspiro[5.5]undecane
N-(cyclohexylmethyl)-4-oxo-1-(propan-2-yl)-5-(thiomorpholine-4-carbonyl)-1,4-dihydropyridine-3-carboxamide
5-methyl-N-{[7-(methylsulfanyl)-2-(morpholin-4-yl)quinolin-3-yl]methyl}-N-[3-(2-oxopyrrolidin-1-yl)propyl]thiophene-2-carboxamide
(2S,4S)-1-(2,3-dihydro-1H-inden-2-yl)-4-{[(2,5-dimethylphenyl)methyl]amino}-N-(2-methoxyethyl)pyrrolidine-2-carboxamide
(2-{[(3-chloro-5-fluoro-4-methoxyphenyl)methyl](thiophen-3-ylmethyl)amino}ethyl)dimethylamine
3-[2-(5-amino-1H-1,2,4-triazol-3-yl)ethyl]-1-(2-{[cyclohexyl(methyl)amino]methyl}phenyl)urea
3-{3-[2-(4-fluorophenyl)pyrrolidin-1-yl]propyl}-5-methyl-4H-1,2,4-triazole
3-[4-(4H-1,2,4-triazol-4-yl)piperidine-1-carbonyl]-3,4-dihydro-2H-1λ6,2-benzothiazine-1,1-dione
N-[3-(1H-imidazol-1-yl)propyl]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
(3aS,6aS)-5-[(4-methanesulfonylphenyl)methyl]-octahydropyrrolo[3,4-b]pyrrole
1-cyclohexanecarbonyl-4-(5-methyl-1,3,4-oxadiazol-2-yl)piperazine
1-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl]-N-[3-(1,3-thiazol-4-yl)phenyl]piperidine-4-carboxamide
7-(2-methoxyethyl)-2-(2-methyl-1H-pyrrole-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
3-[(3,4-dichlorophenyl)methyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-cyclopropyl-3-(1-{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl}piperidin-4-yl)propanamide
(2S,4S)-4-amino-1-[(1-ethyl-1H-indol-4-yl)methyl]pyrrolidine-2-carboxylic acid
5-{2-[(3R,4S)-3-amino-4-(3-methoxyphenyl)pyrrolidin-1-yl]-2-oxoethyl}-3-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
5-(hydroxymethyl)-4-{[(2S,6S)-6-(hydroxymethyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-trien-4-yl]methyl}-2-methylpyridin-3-ol
1-phenyl-4-{5-[1-(piperidin-1-yl)ethyl]furan-2-carbonyl}piperazin-2-one
2-amino-6-(2,2-dimethyloxan-4-yl)-4-(1-methyl-1H-pyrazol-4-yl)-5-propylpyridine-3-carbonitrile
5-{[(3S,4R)-3-(dimethylamino)-4-(4-methylphenyl)pyrrolidin-1-yl]methyl}-N,N-dimethylpyridin-2-amine