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2-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]acetamide
1-[(1R,5R)-6-(cyclopropylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-2-(thiophen-2-yl)ethan-1-one
2-(2H-1,3-benzodioxol-5-yl)-N,1-bis(propan-2-yl)-1H-1,3-benzodiazole-5-sulfonamide
4-(2-hydroxybenzoyl)-3-methyl-1-[(4-methylphenyl)methyl]piperazin-2-one
N-{[4-(2,3-dihydro-1H-inden-2-yloxy)phenyl]methyl}-2-(4-fluorophenyl)-N-[(3S)-2-oxoazepan-3-yl]acetamide
1-[2-(5-chloro-2-methoxypyridin-4-yl)pyrimidin-4-yl]piperidin-4-ol
(1R,7S)-6-(2,3-dihydro-1H-isoindole-2-carbonyl)-3-[2-(4-methylphenyl)ethyl]-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-4-one
N-[(2-{4-[3-(4-methoxyphenyl)propanamido]phenyl}-5-methyl-1,3-oxazol-4-yl)methyl]-3,5-dimethyl-1H-pyrrole-2-carboxamide
3-[(5-methyl-1-phenyl-1H-pyrazol-4-yl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-(2-cyclohexaneamido-5-methylphenyl)pyridazine-4-carboxamide
(2R)-2-phenyl-2-[4-(2-phenylethyl)-1H-1,2,3-triazol-1-yl]ethan-1-ol
2-(3-chloro-4-hydroxyphenyl)-1-[4-(4-methyl-1H-pyrazol-3-yl)piperidin-1-yl]ethan-1-one
2-(5-amino-3-methyl-1H-pyrazol-1-yl)-N-[1-(pyridin-4-yl)propyl]acetamide
3-(3,5-dimethyl-1H-pyrazol-1-yl)-N-[2-(4-fluorophenyl)ethyl]-N-{[2-(3-hydroxypiperidin-1-yl)-5,8-dimethoxyquinolin-3-yl]methyl}propanamide
6-(5-fluoroquinolin-8-yl)pyridine-2-carboxamide
3-[2-(piperidin-2-yl)ethyl]-5-[1-(propan-2-yl)-1H-imidazol-2-yl]phenol
2-(furan-2-yl)-5-(1-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}-1H-imidazol-2-yl)pyrimidine
(1R,5R)-6-[(5-propylfuran-2-yl)methyl]-3-(pyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
1-(cyclohexylmethyl)-N-[(4-methyl-1H-1,3-benzodiazol-2-yl)methyl]-6-oxopiperidine-3-carboxamide
N-methyl-N-[(2-methyl-1,3-thiazol-4-yl)methyl]-2-(pyridin-4-yl)acetamide
2-(5-{[2-(pyridin-2-yl)pyrrolidin-1-yl]methyl}furan-2-yl)benzonitrile
N-{2-[1-(2-ethoxy-5-methylbenzenesulfonyl)piperidin-2-yl]ethyl}acetamide
N-methyl-N-(1,2-oxazol-3-ylmethyl)-5-oxo-1-(pyridin-3-ylmethyl)pyrrolidine-3-carboxamide
5-acetyl-N-(1-phenylbutyl)thiophene-3-carboxamide
3-{2-[(4-methylphenyl)methyl]-5-oxopyrrolidin-2-yl}-N-[2-(pyridin-3-yloxy)propyl]propanamide
5-fluoro-3-methyl-2-{[4-(pyridin-2-ylmethoxy)piperidin-1-yl]methyl}-1H-indole
(1R,2R,4R)-N-(2-hydroxyethyl)-N-(thiophen-2-ylmethyl)bicyclo[2.2.1]hept-5-ene-2-carboxamide
N-[(3R,4S)-4-propyl-1-(pyrimidin-2-ylmethyl)pyrrolidin-3-yl]oxane-4-carboxamide
8-{[2-(2-hydroxyethoxy)phenyl]methyl}-3-(pentan-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
8-[(2,3-difluorophenyl)methyl]-1-oxa-8-azaspiro[4.6]undecan-9-one
(3S,4S)-1-[2-amino-6-(2-methylpropyl)pyrimidine-4-carbonyl]-4-(4-fluorophenyl)piperidin-3-ol
1-{[2-(3-methoxypyridin-2-yl)phenyl]methyl}piperidin-4-one
N-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]-3-(trifluoromethyl)-1H-pyrazole-5-carboxamide
3-{5-[3-(trimethyl-1H-pyrazol-4-yl)propanoyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanoic acid
(1R,5R)-6-(2-methoxyethyl)-3-(4-methyl-1,2,3-thiadiazole-5-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-4-methylpiperazine-1-carboxamide
3-(4-methyl-1H-pyrazol-1-yl)-5-[(propan-2-yl)sulfamoyl]benzoic acid
4-[1-(2H-1,3-benzodioxol-5-yl)propan-2-yl]-1-{[1,2,4]triazolo[4,3-a]pyridin-3-ylmethyl}-1H-1,2,3-triazole
N-{2-[4-phenyl-5-(2-phenyl-1,3-oxazol-4-yl)-1H-imidazol-1-yl]ethyl}acetamide
N-[3-(2-methyl-1H-imidazol-1-yl)propyl]-5-propyl-1,3,4-oxadiazol-2-amine
6-fluoro-N-{[1-methyl-2-(methylsulfanyl)-1H-imidazol-5-yl]methyl}-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
N-(1-{[2-(furan-2-yl)pyrimidin-5-yl]methyl}piperidin-4-yl)methanesulfonamide
2-(2-{1H-pyrazolo[3,4-b]pyridin-1-yl}phenyl)acetic acid
2-[methyl(1-methylpiperidin-4-yl)amino]-N-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)acetamide
5-(4-chloro-1H-pyrazol-3-yl)-3-cyclopropyl-1-(2-phenylethyl)-1H-1,2,4-triazole
6-ethyl-3-({[1-(4-fluorophenyl)propan-2-yl]amino}methyl)-2-methoxy-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
1-{7-methylpyrazolo[1,5-a]pyrimidine-6-carbonyl}-3-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine
6-methoxy-N-[2-(pyridin-3-yloxy)propyl]pyrimidin-4-amine
1-[(1-methyl-3-phenyl-1H-pyrazol-4-yl)methyl]-8-(pyrimidin-2-yl)-1,8-diazaspiro[4.5]decane
1-(1-{5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidin-4-yl)-N-cyclopropylpiperidine-3-carboxamide