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N-[6,6-dimethyl-1-(4-methylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-(pyridin-4-ylsulfanyl)acetamide
4-(4-{3-[5-(2-chlorophenyl)pyrimidin-4-yl]piperidine-1-carbonyl}phenyl)morpholine
1-(2-methylphenyl)-4-(pyrimidin-4-yl)-1,4-diazepane
N3-benzyl-1-cyclopropyl-4-oxo-N5-[2,2,2-trifluoro-1-(pyridin-2-yl)ethyl]-1,4-dihydropyridine-3,5-dicarboxamide
3-(morpholin-4-yl)-1-{3-phenyl-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl}butan-1-one
4-[1-(4-chlorophenyl)-3-methyl-1H-1,2,4-triazol-5-yl]benzene-1-sulfonamide
5-(2-chloro-4,6-dimethoxyphenyl)-1-ethyl-1H,4H-pyrazolo[3,4-d]imidazole
N-{4-[4-(2-ethoxyethyl)piperazine-1-carbonyl]phenyl}-2-methylfuran-3-carboxamide
4-(4-chlorophenoxy)-1-(3-cyanopyridin-2-yl)piperidine-4-carboxylic acid
5-{[3-(2-fluorophenoxymethyl)piperidin-1-yl]methyl}-2-methoxyphenol
1-methyl-3-(2-phenylethyl)-8-{[2-(trifluoromethyl)phenyl]methyl}-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-[(1-{[5-(hydroxymethyl)furan-2-yl]methyl}piperidin-4-yl)oxy]-N-(pyridin-4-ylmethyl)benzamide
(2S,4S)-N-ethyl-4-({[2-(prop-2-en-1-yloxy)phenyl]methyl}amino)-1-(propan-2-yl)pyrrolidine-2-carboxamide
3-(1,1-dioxo-1λ6-thiolan-3-yl)-3-(2-hydroxyethyl)-1-[3-(2-oxo-1,3-oxazolidin-3-yl)phenyl]urea
ethyl 1-[(2-hydroxyphenyl)methyl]-4-(2-phenoxyethyl)piperidine-4-carboxylate
2-[6-(4H-1,2,4-triazol-4-yl)pyridine-2-carbonyl]-1,2,3,4-tetrahydroisoquinoline
2-ethyl-4-phenyl-9-(pyrrolidine-1-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
4-[4-(4-{[cyclohexyl(methyl)amino]methyl}-1H-1,2,3-triazol-1-yl)piperidine-1-carbonyl]pyrrolidin-2-one
2-(2,4-dioxoimidazolidin-1-yl)-N-({1-[2-(2-fluorophenyl)ethyl]piperidin-3-yl}methyl)-N-methylacetamide
2-methyl-1-{[3-(3-methylphenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}-1,4-diazepan-5-one
4-(5-cyclopropyl-3-methyl-1H-pyrazole-4-carbonyl)-1-(4-methoxyphenyl)-2,2-dimethylpiperazine
N-[3-(cyclopentyloxy)propyl]-2,6-dimethylimidazo[1,2-a]pyridine-3-carboxamide
N-[1-(morpholine-4-carbonyl)piperidin-4-yl]imidazo[2,1-b][1,3]thiazole-6-carboxamide
1-(2,3-dichlorobenzoyl)-4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine
(2S)-4-methanesulfonyl-2-{[5-(4-methylphenyl)-1H-pyrazol-3-yl]formamido}butanoic acid
methyl 3-{[1-(3-fluoro-4-hydroxyphenyl)ethyl]carbamoyl}benzoate
ethyl 1-[1-(2-phenylethyl)-1H-1,2,3-triazole-4-carbonyl]piperidine-3-carboxylate
2-(dimethyl-1,2-oxazol-4-yl)-N-({4-[(3-phenylpropyl)amino]quinazolin-2-yl}methyl)acetamide
2-(4-{[3-(aminomethyl)piperidin-1-yl]methyl}phenyl)-6-(pyridin-3-yl)-3,4-dihydropyrimidin-4-one
6-[(2R,3S,6R)-3-(3-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]pyridine-2-carbonitrile
6-ethoxy-3-{[3-(2-methylpiperidin-1-yl)azetidin-1-yl]methyl}-1,2-dihydroquinolin-2-one
N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-N,2,4-trimethyl-1,3-thiazole-5-carboxamide
N-[3-(1H-indazol-1-yl)propyl]-3-(1H-pyrazol-1-yl)benzamide
N-(1-benzothiophen-5-ylmethyl)-1-[2-(4-chlorophenyl)ethyl]-6-oxopiperidine-3-carboxamide
9-[(3E)-pent-3-enoyl]-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
1-(azepan-1-yl)-3-{5-[2-(1H-indol-3-yl)ethyl]-1,3,4-oxadiazol-2-yl}propan-1-one
N-[4-({[2-(dimethylamino)ethyl](thiophen-3-ylmethyl)amino}methyl)phenyl]acetamide
N-[(3S,4R)-1-{[2-(furan-2-yl)phenyl]methyl}-4-propylpyrrolidin-3-yl]acetamide
4-[2-(4-chlorophenoxy)ethyl]-1,2-dihydropyridin-2-one
2-fluoro-N-[2-(pyridin-3-yl)ethyl]-5-sulfamoylbenzamide
4-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-3,4-dihydro-2H-1,4-benzothiazin-3-one
[1-(2-{[2-(2-aminoethyl)quinazolin-4-yl]amino}ethyl)piperidin-2-yl]methanol
2-{[6-(2-chlorophenyl)-8-oxo-7-(prop-2-en-1-yl)-7H,8H-imidazo[1,2-a]pyrazin-2-yl]formamido}-N-methylpropanamide
2-amino-6-(2-hydroxypropan-2-yl)-4-(1-phenyl-1H-pyrazol-5-yl)pyridine-3-carbonitrile
4-[(4-chlorophenyl)methyl]-1-(6-ethylpyrimidin-4-yl)piperidine-4-carboxylic acid
[5-(1-{[2-(2-methoxyphenyl)-1,3-thiazol-5-yl]methyl}-1H-imidazol-2-yl)furan-2-yl]methanol
3-(4-acetyl-3,5-dimethyl-1H-pyrazol-1-yl)-N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]propanamide
(2S,4R)-4-amino-1-[4-(methoxymethyl)-5-methyl-1,2-oxazole-3-carbonyl]-N-methylpyrrolidine-2-carboxamide
N-({6-ethyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-3-(1,2-oxazinan-2-yl)propanamide
2-{[1-(4-tert-butylphenyl)-1H-1,2,4-triazol-5-yl]methoxy}acetamide