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(1,4-dioxan-2-ylmethyl)(methyl){[3-(4-phenylphenyl)-1H-pyrazol-4-yl]methyl}amine
N-(1,4-dioxan-2-ylmethyl)-5-(3-fluorophenoxymethyl)-1H-pyrazole-3-carboxamide
1-ethyl-N-{[2-(1H-imidazol-1-yl)phenyl]methyl}-2,5-dimethyl-1H-pyrrole-3-carboxamide
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-2-(hydroxymethyl)-1H-1,3-benzodiazole-5-carboxamide
1-methyl-6-{[4-(thiomorpholin-4-yl)piperidin-1-yl]methyl}-1H-indole
N-(2,3-dihydro-1-benzofuran-2-ylmethyl)-N,2-dimethyl-1H-imidazole-4-carboxamide
{1-ethyl-5-[3-(5-methylfuran-2-yl)-1H-pyrazole-5-carbonyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl}methanol
N-[(1-{[(1-methyl-1H-pyrazol-4-yl)carbamoyl]methyl}-1,2,5,6-tetrahydropyridin-3-yl)methyl]pyrrolidine-1-carboxamide
6-{[1-(2,3-dihydro-1H-inden-2-yl)-5-oxopyrrolidin-3-yl]amino}pyridine-3-carbonitrile
(2S,4R)-N-ethyl-1-methyl-4-{2-[(4-methylphenyl)methyl]benzamido}pyrrolidine-2-carboxamide
1-(4-chlorophenyl)-N-[(3-methyloxetan-3-yl)methyl]cyclopropane-1-carboxamide
2-[7-methoxy-2-oxo-6-(pyrrolidin-1-yl)-1,2,3,4-tetrahydroquinolin-4-yl]benzonitrile
2-methyl-6-{3-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-2,3-dihydropyridazin-3-one
2-(2-chlorophenyl)-N-(2-hydroxyethyl)-3-methyl-N-propyl-3H-imidazo[4,5-b]pyridine-6-carboxamide
2-[4-(6-methylpyridin-2-yl)piperazin-1-yl]-2-[4-(1H-pyrazol-1-yl)phenyl]acetic acid
3-({2-[1-(5-propyl-1,3,4-thiadiazol-2-yl)piperidin-4-yl]-1H-imidazol-1-yl}methyl)pyridine
N-{1-[(3R,4R)-3-hydroxy-3,4-dimethylpyrrolidin-1-yl]-2-methyl-1-oxopropan-2-yl}acetamide
N-[(6-chloropyridin-3-yl)methyl]-N-methyl-2-(pyridin-4-yl)pyrimidine-5-carboxamide
N,N-dimethyl-2-[5-(pyrrolidin-1-ylmethyl)pyridin-2-yl]aniline
3-(1H-1,3-benzodiazol-1-yl)-N-{[1-(pyrimidin-2-yl)piperidin-3-yl]methyl}propanamide
4-[5-({4-[(2-fluorophenyl)methyl]piperidin-1-yl}methyl)-1,3-thiazol-2-yl]morpholine
1-methyl-4-{5-[(methylsulfanyl)methyl]-3-(thiophen-2-ylmethyl)-1H-1,2,4-triazol-1-yl}piperidine
2-[1-(2,3-dihydro-1,4-benzodioxin-6-yl)-5-[(oxolan-2-ylmethoxy)methyl]-1H-1,2,4-triazol-3-yl]acetamide
3-{2-[(3-methylquinoxalin-2-yl)methyl]-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-1-yl}phenol
{2-fluoro-5-[2-methoxy-5-(pyrrolidin-1-ylmethyl)phenoxy]phenyl}methanol
N-({1-[2-(4-fluorophenyl)ethyl]piperidin-3-yl}methyl)-N-methyl-2-(2-oxo-1,3-oxazolidin-3-yl)acetamide
1-[4-hydroxy-2-(2-methyl-1,3-thiazol-4-yl)pyrimidine-5-carbonyl]piperidine-3-carbonitrile
9-{3-[4-(dimethylamino)phenyl]propanoyl}-2-methyl-2,9-diazaspiro[5.5]undecan-3-one
3,5,7-trimethyl-2-[3-(pyridin-2-yl)azetidine-1-carbonyl]-1H-indole
3-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}-1-[4-(morpholine-4-carbonyl)phenyl]urea
2-[3-(2-methyl-1,3-thiazol-4-yl)-5-(morpholin-3-ylmethyl)-1H-1,2,4-triazol-1-yl]acetic acid
3-{1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-ylmethyl}-1,2-dihydroquinolin-2-one
2-hydroxy-2-(4-methoxyphenyl)-N-(pyrimidin-4-ylmethyl)acetamide
2-[2-({3-cyclopentyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}methyl)-1H-pyrrol-1-yl]-4-methylpyridine
N-methyl-N-(3-methylbutyl)-3-[(thiophen-3-ylmethyl)sulfamoyl]benzamide
3-(4-{[2-(2-methylpropyl)morpholin-4-yl]methyl}-1H-pyrazol-1-yl)propanoic acid
1-[2-amino-6-(pyrrolidin-1-yl)pyrimidin-4-yl]-4-(1H-imidazol-1-yl)piperidine-4-carboxylic acid
(1S,5R)-6-(5,6-dimethylpyridine-3-carbonyl)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octane
(2S,4R)-4-hydroxy-N-{[4-(4-methylphenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}pyrrolidine-2-carboxamide
3-(5-methylfuran-2-yl)-N-[2-(pyrrolidine-1-sulfonyl)ethyl]benzamide
1-[(2,4-difluorophenyl)methyl]-4-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidine
N-methyl-2-(3-methyl-1,2-oxazol-5-yl)-N-{[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}acetamide
N-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}-3-[2-(furan-2-ylmethyl)-5-oxopyrrolidin-2-yl]-N-methylpropanamide
2-{1-[(2,4-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-(3-hydroxy-2,2-dimethylpropyl)acetamide
3-[(3R,4S)-4-(4-methylpiperazin-1-yl)-1-{7-methylthieno[3,2-d]pyrimidin-4-yl}piperidin-3-yl]propanoic acid
1-(2-chlorophenyl)-4-(2-propyl-1,3-thiazole-4-carbonyl)piperazine
3-{[(3R,4S)-3-(hydroxymethyl)-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-1-yl]methyl}-1-methyl-1,2-dihydroquinolin-2-one
N-[2-(1-methyl-1H-1,2,4-triazol-5-yl)ethyl]-3-(3-phenyl-1,2,4-oxadiazol-5-yl)propanamide
1-(1-ethyl-1H-pyrazole-5-carbonyl)-3-[4-(4-fluorophenyl)-1H-pyrazol-5-yl]piperidine
2-cyclopropyl-8-({9-hydroxy-4-oxo-4H-pyrido[1,2-a]pyrimidin-2-yl}methyl)-2,8-diazaspiro[5.5]undecan-3-one