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2-(dimethylamino)-8-(2-ethylphenyl)-4H,5H,6H,7H,8H-[1,3]thiazolo[4,5-c]azepin-6-one
5-(oxolane-2-carbonyl)-3-(4-phenylphenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
4-(1-butyl-3-cyclopentyl-1H-1,2,4-triazol-5-yl)-1-methylpiperidin-4-ol
2-chloro-N-[1-(3-phenylpropyl)piperidin-3-yl]pyridine-4-carboxamide
3-{[1-(4-methyl-1,2,5-oxadiazole-3-carbonyl)piperidin-4-yl]methyl}-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
1-[2-({[2-(1H-1,2,4-triazol-1-yl)phenyl]methyl}amino)pyrimidin-4-yl]piperidin-3-ol
2-(5-acetylthiophen-3-yl)-N-[(3,4-difluorophenyl)methyl]acetamide
[3-(3-methylbut-2-en-1-yl)-1-(pyridine-2-carbonyl)piperidin-3-yl]methanol
6-methyl-5-(2-{2-methyl-4-[(3-methylphenyl)methyl]-3-oxopiperazin-1-yl}-2-oxoethyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-phenyl-4-[1-(3-phenylpropyl)piperidin-3-yl]piperazine
(3aR,6aS)-5-(1-ethyl-3-methyl-1H-pyrazole-5-carbonyl)-1-oxo-2-propyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2,4-dimethyl-N-(4-{4-[4-(pyrimidin-2-yl)-1,4-diazepan-1-yl]piperidin-1-yl}phenyl)benzamide
N-[(4-cyclohexyl-4H-1,2,4-triazol-3-yl)methyl]-3-(5-methylfuran-2-yl)-1H-pyrazole-5-carboxamide
(1S,5R)-6-benzyl-3-[(4-methoxy-3,5-dimethylpyridin-2-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
(4aS,8aR)-1-[3-(methylsulfanyl)propyl]-6-(5-oxo-2,5-dihydro-1H-pyrazole-3-carbonyl)-decahydro-1,6-naphthyridin-2-one
1-(3-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}phenyl)-1H-pyrazole
3-{4-phenyl-1-[4-(pyrrolidin-1-yl)butyl]-1H-imidazol-5-yl}pyridine
3-(2-oxopyrrolidin-1-yl)-N-(pyridin-3-ylmethyl)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)propanamide
{4-[(2-chlorophenyl)methyl]-1-(thiophene-3-sulfonyl)piperidin-4-yl}methanol
1-{1'-[(2-butyl-1H-imidazol-4-yl)methyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}ethan-1-one
4-{4-[(4-cyclobutanecarbonyl-1,4-diazepan-1-yl)methyl]phenyl}-2-methylbutan-2-ol
N-(2H-1,3-benzodioxol-5-ylmethyl)-2-methoxy-N-methyl-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
7-(2-ethoxybenzoyl)-2-[(2-methyl-1H-imidazol-4-yl)methyl]-2,7-diazaspiro[4.5]decane
6-(5-aminopyridin-3-yl)-5-chloropyridine-3-carboxylic acid
N-[(3-methoxyphenyl)methyl]-3-[1-(1H-pyrrole-3-carbonyl)piperidin-3-yl]propanamide
(2S,4R)-N-(propan-2-yl)-1-(1,3-thiazol-2-ylmethyl)-4-[2-(1H-1,2,4-triazol-1-yl)acetamido]pyrrolidine-2-carboxamide
N-[(7-chloro-4-{[(4-fluorophenyl)methyl]amino}quinazolin-2-yl)methyl]-1,3,5-trimethyl-1H-pyrazole-4-sulfonamide
N-[2-(1H-imidazol-4-yl)ethyl]-2-[4-(propan-2-yl)morpholin-2-yl]acetamide
5-phenyl-2-(pyridin-4-yl)-4-[1-(thiophene-2-carbonyl)piperidin-3-yl]pyrimidine
3-[4-(1,3-benzothiazol-2-yl)piperazine-1-carbonyl]-4,5,6,7-tetrahydro-1,2-benzoxazole
1-(2-{[(1,4-dithiepan-6-yl)amino]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl)ethan-1-one
methyl 1-[(3R,5S)-1-(2-ethylbutyl)-5-{[(4-methoxyphenyl)methyl]carbamoyl}pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
2-[4-(ethanesulfonyl)piperazin-1-yl]-2-(4-methoxy-3,5-dimethylphenyl)acetic acid
4-{[(2R,3S,6R)-3-(3-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]methyl}phenol
N-(pyridin-2-ylmethyl)-4-(quinolin-5-yloxy)piperidine-4-carboxamide
N-[2-(1H-indol-3-yl)ethyl]-3-(1H-pyrazol-1-yl)benzamide
1-[(1-cyclopropyl-1H-imidazol-2-yl)methyl]-4-phenylpyrrolidin-2-one
3-(4-chlorobenzoyl)-1-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}piperidine
N-[2-(pyridin-3-yloxy)propyl]-2-[5-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
2-methyl-4-[5-({[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]sulfanyl}methyl)-3-phenyl-1H-1,2,4-triazol-1-yl]pyridine
(1R,5R)-6-[(2-butyl-5-chloro-1H-imidazol-4-yl)methyl]-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
1-{4-[2-(isoquinolin-1-yloxy)hex-5-en-1-yl]piperazin-1-yl}ethan-1-one
4-[(3S,4R)-4-hydroxyoxolan-3-yl]-N-[3-(methylsulfanyl)phenyl]-1,4-diazepane-1-carboxamide
3-(2-methylpropyl)-6-(1-phenylethyl)-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazole
2-{8-methylimidazo[1,2-a]pyridin-3-yl}-N-(propan-2-yl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]acetamide
N-(5-methyl-1,3,4-thiadiazol-2-yl)-2-(2-methylpentanoyl)-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
1-(1-{4-[(3S)-3-ethylmorpholine-4-carbonyl]phenyl}-2,5-dimethyl-1H-pyrrol-3-yl)ethan-1-one
N-[2-({[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}amino)ethyl]pyridine-4-carboxamide
N-[2-(pyridin-2-ylsulfanyl)ethyl]-2,3-dihydro-1,4-benzodioxine-6-carboxamide
1-(2,3-dihydro-1H-inden-2-yl)-4-[2-(pyrrolidin-3-yl)benzoyl]-1,4-diazepane