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1-[(2R,6R)-6-methyl-2-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridin-1-yl]-3-(1H-1,2,4-triazol-1-yl)propan-1-one
N-[2-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]-2-(pyridin-4-ylsulfanyl)acetamide
4-cyclopropyl-6-{4-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrimidine
(1R,6S)-9-methyl-3-{[5-(1,3-oxazol-5-yl)thiophen-2-yl]sulfonyl}-3,9-diazabicyclo[4.2.1]nonane
1-methyl-4-{[5-(2-propyl-1,3-thiazol-4-yl)-1,2,4-oxadiazol-3-yl]methyl}piperidine
(2S)-2-amino-1-[4-(4-fluorophenoxy)piperidin-1-yl]-3-(1H-imidazol-4-yl)propan-1-one
2-{[1-(2-fluorophenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}-1H-imidazole
2-[(3,3-diethylpyrrolidin-1-yl)methyl]pyridine-3-carboxylic acid
1-{3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}-3-(5-methyl-1H-1,2,4-triazol-3-yl)propan-1-one
(3aS,6aS)-2-(2-chloro-4-fluoro-5-methylbenzenesulfonyl)-5-methyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-{3-oxo-1-[(2E)-3-phenylprop-2-en-1-yl]piperazin-2-yl}-N-[3-(1H-pyrazol-1-yl)propyl]acetamide
1-[2-(2,2-diphenylethyl)morpholin-4-yl]-2-(1H-pyrazol-1-yl)ethan-1-one
N-(3-{[(2-hydroxyethyl)[(1-methyl-1H-imidazol-2-yl)methyl]carbamoyl]amino}-4-methylphenyl)propanamide
1-(4-{3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}thiophen-2-yl)ethan-1-one
3,5-dimethyl-2-[4-(thiomorpholin-4-yl)piperidine-1-carbonyl]-1H-indole
1-methyl-4-[6-methyl-2-(piperidin-1-yl)pyrimidin-4-yl]-1,4,9-triazaspiro[5.6]dodecan-10-one
(1S,5R)-3-[(5-acetylthiophen-3-yl)methyl]-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-butyl-3-(3,4-difluorophenyl)-5-[2-(4-methyl-4H-1,2,4-triazol-3-yl)ethyl]-1H-1,2,4-triazole
1-ethyl-3-(2-methylpropyl)-N-{1-oxaspiro[4.4]nonan-3-yl}-1H-pyrazole-5-carboxamide
2-{5H,6H-imidazo[2,1-b][1,3]thiazol-3-yl}-1-[3-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]ethan-1-one
N-[2-(N-methylmethanesulfonamido)ethyl]-2-(thiophen-2-yl)-1,3-thiazole-4-carboxamide
8-[(4-carboxy-1,3-oxazol-2-yl)methyl]-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
2-methoxy-5-{[4-(4-phenyl-1H-pyrazol-5-yl)piperidin-1-yl]methyl}pyrimidine
N-(adamantan-2-ylmethyl)-6-{[methyl(thiophen-3-ylmethyl)amino]methyl}-2-oxo-1,2-dihydropyridine-3-carboxamide
3-amino-1-{4-[4-cyclopropyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}propan-1-one
2-(butylsulfanyl)-6-[4-(1H-1,2,4-triazole-3-carbonyl)piperazin-1-yl]pyrimidin-4-amine
2-[2-(3,4-dimethoxyphenyl)ethyl]-4-[4-(3,5-dimethylbenzoyl)piperazin-1-yl]-2,3-dihydro-1H-isoindole-1,3-dione
3-(1-methyl-1H-pyrrol-2-yl)-N-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-ylmethyl}-1H-pyrazole-5-carboxamide
8-[(1-methyl-1H-imidazol-2-yl)methyl]-2-propyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
5-cyclopentyl-1-(2-phenylethyl)-N-(pyridin-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N,N-bis(1,3-oxazol-4-ylmethyl)-2,3-dihydro-1H-indene-1-carboxamide
N-(3-hydroxypropyl)-1-[1-(1H-indol-2-ylmethyl)piperidin-4-yl]-1H-1,2,3-triazole-4-carboxamide
4-{7-methylimidazo[1,2-a]pyridine-2-carbonyl}thiomorpholine
5-(4,5,6,7-tetrahydro-1-benzothiophene-3-carbonyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
N-[2-(diethylamino)ethyl]-1-{9-methoxy-5H,6H-benzo[h]quinazolin-2-yl}-N,5-dimethyl-1H-pyrazole-4-carboxamide
(4aR,7aS)-1-(2-hydroxyethyl)-4-(5-phenylpentanoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]-1-(2-methoxyphenyl)-N-methyl-1H-pyrazole-4-carboxamide
2-(4-{[(1,4-dioxan-2-ylmethyl)(methyl)amino]methyl}phenyl)-6-(trifluoromethyl)-3,4-dihydropyrimidin-4-one
N'-(3-chloro-4-methylphenyl)-N-[4-(1H-pyrazol-1-yl)butan-2-yl]propanediamide
8-(1-methoxypropan-2-yl)-1-(3-methylbutyl)-3-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-(2-ethylphenoxy)-1-{pyrazolo[1,5-a]pyridine-3-carbonyl}azetidine
5-[2-(2-aminoethyl)morpholin-4-yl]-2-[2-(propan-2-ylsulfanyl)ethyl]-2,3-dihydropyridazin-3-one
6-(1-methyl-1H-imidazol-2-yl)-N-(1-phenylethyl)pyridazin-3-amine
N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]oxan-4-amine
3-[2-({1-[3-(2-oxoimidazolidin-1-yl)phenyl]piperidin-4-yl}amino)ethyl]-1,3-oxazolidin-2-one
({1-[2-(3-fluorophenyl)ethyl]piperidin-4-yl}methyl)(methyl)(pyridin-4-ylmethyl)amine
4-[(2H-1,3-benzodioxol-5-ylmethyl)amino]-N-benzyl-N-(2-hydroxyethyl)-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
2-(5-methyl-1,2-oxazol-3-yl)-N-(4-methyl-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-6-yl)piperidine-1-carboxamide
3-(2-methyl-1H-indol-1-yl)-N-[4-(oxolan-2-yl)butyl]propanamide
2-[5-(acetamidomethyl)-1,2,3,6-tetrahydropyridin-1-yl]-N-[1-(4-methylphenyl)ethyl]acetamide