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2,2-difluoro-N-[2-(4-{[2-(propan-2-yl)-1,3-oxazol-4-yl]methyl}morpholin-2-yl)ethyl]acetamide
5-(5-chloro-1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-1-[2-(morpholin-4-yl)ethyl]piperidin-2-one
(3-{[(1-{imidazo[2,1-b][1,3,4]thiadiazol-6-yl}ethyl)amino]methyl}-2,4,6-trimethylphenyl)methanol
(1R,5R)-6-[(5-methylfuran-2-yl)methyl]-3-(pyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
methyl (2S,4R)-1-[(6-chloro-2-fluoro-3-methoxyphenyl)methyl]-4-(dimethylamino)pyrrolidine-2-carboxylate
2-{[4-(4-phenyl-1H-imidazol-5-yl)-1H-pyrrolo[2,3-b]pyridin-6-yl]amino}acetic acid
N,N-diethyl-1-[(1s,4s)-4-(pent-4-enamido)cyclohexyl]-1H-1,2,3-triazole-4-carboxamide
2-{1-[(2-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-(furan-3-ylmethyl)acetamide
4-(1H-imidazol-1-yl)-1-[(3-methyl-1-benzofuran-2-yl)methyl]piperidine-4-carboxylic acid
1-[1-(2-methoxyphenyl)-1H-pyrazole-4-carbonyl]-4-(4-methyl-4H-1,2,4-triazol-3-yl)piperidine
2-(3-methoxypiperidin-1-yl)-5-[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]pyridine
N-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}-3-[4-(3-methylphenyl)piperazin-1-yl]propanamide
2-amino-4-(3-ethoxy-4-hydroxyphenyl)-5-methyl-6-(1-methyl-1H-pyrazol-4-yl)pyridine-3-carbonitrile
1-[(3-fluorophenyl)methyl]-4-(4-methylpiperidine-4-carbonyl)-1,4-diazepan-6-ol
1-{1-[6-(3-chlorophenyl)pyridine-3-carbonyl]piperidin-3-yl}-3-methylbutan-1-one
2-{[1-(2-hydroxyacetyl)piperidin-4-yl]oxy}-4-methoxy-N-(2-methoxyethyl)benzamide
N-[(3R,4S)-1-(4-phenylbutanoyl)-4-propylpyrrolidin-3-yl]methanesulfonamide
N-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-methyl-2-(methylsulfanyl)pyrimidine-5-carboxamide
3-{[2-(1-ethyl-1H-1,2,4-triazol-5-yl)-1H-imidazol-1-yl]methyl}pyridine
1-[4-({4-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}methyl)thiophen-2-yl]ethan-1-one
N-ethyl-5-{[4-(pyrrolidine-1-sulfonyl)-1,4-diazepan-1-yl]methyl}pyrimidin-2-amine
2-(dimethylamino)-2-(2-methylphenyl)-N-propyl-N-(thiophen-3-ylmethyl)acetamide
2-[1-(2-ethylpyrimidine-5-carbonyl)piperidin-4-yl]-1,2,3,4-tetrahydroisoquinoline
2-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-N-{[2-(1H-1,2,4-triazol-1-yl)phenyl]methyl}-1,3-oxazole-4-carboxamide
N-(2-{4-[(3-chloropyridin-4-yl)methyl]morpholin-2-yl}ethyl)-3-methylbut-2-enamide
N-(1-benzylpiperidin-3-yl)-2-[5-(pyrrolidin-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
2-[5-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-N-[2,2,2-trifluoro-1-(pyridin-2-yl)ethyl]acetamide
[(3,5-dimethoxyphenyl)methyl]({1-[2-(4-fluorophenyl)ethyl]piperidin-3-yl}methyl)methylamine
N-(2-chloro-4-methylphenyl)-3-(diethylamino)pyrrolidine-1-carboxamide
(1S,5R)-6-(3-methylbut-2-en-1-yl)-3-({4-oxo-4H-pyrido[1,2-a]pyrimidin-2-yl}methyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
3,5-difluoro-2-{4-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyridine
N-(furan-2-ylmethyl)-5-methyl-4-(methylamino)thieno[2,3-d]pyrimidine-6-carboxamide
4-(1H-imidazol-1-yl)-1-(1H-indole-5-carbonyl)piperidine-4-carboxylic acid
1'-[2-(2-phenyl-1H-imidazol-1-yl)acetyl]-3,4-dihydrospiro[1-benzopyran-2,3'-pyrrolidine]-4-one
N-{5-propylpyrazolo[1,5-a]pyrimidin-7-yl}-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}-3-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]piperidine
3-[(4-ethyl-1,4-diazepan-1-yl)methyl]-1-[(2-fluoro-5-methoxyphenyl)methyl]-3-hydroxypiperidin-2-one
3-[(cyclobutylamino)methyl]-1-(2,2-dimethylpropyl)-3-hydroxypiperidin-2-one
(pyridin-4-ylmethyl)({3-[4-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl}methyl)amine
{4-methyl-5-[1-(quinolin-4-ylmethyl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methanol
8-[3-(3-hydroxy-1,2-oxazol-5-yl)propanoyl]-2-(3-methylbutyl)-2,8-diazaspiro[5.5]undecan-3-one
1-[(3R,4R)-4-{4-[2-(furan-2-yl)phenyl]-1H-1,2,3-triazol-1-yl}oxolan-3-yl]piperidine
{[2-(4-fluoro-3-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(isoquinolin-5-ylmethyl)methylamine
N-(3-methyl-1-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}butyl)-4-oxo-4H-chromene-2-carboxamide
N-methyl-6-(4-methylphenyl)-N-[1-(pyridin-3-yl)propyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
N-[(3R,4S)-4-cyclopropyl-1-(2-fluoro-4-methylbenzenesulfonyl)pyrrolidin-3-yl]acetamide
1-{2-[methyl(pyridin-4-ylmethyl)amino]acetyl}-3-(3-methylbut-2-en-1-yl)piperidine-3-carboxylic acid
2-({[(3R,4R)-1-(1-benzoxepine-4-carbonyl)-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
N-[(4-cyclohexyl-4H-1,2,4-triazol-3-yl)methyl]-6-methylimidazo[1,2-a]pyridine-2-carboxamide
1-(3-oxo-3-{4-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}propyl)pyrrolidin-2-one