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1-[3-(3-ethylphenoxy)azetidin-1-yl]-3-(pyridin-4-yl)propan-1-one
methyl (2S)-1-[5-cyclohexaneamido-1-(2-methoxyethyl)-1H-1,3-benzodiazole-7-carbonyl]pyrrolidine-2-carboxylate
3-[3-(dimethylamino)propyl]-5-[(3-fluorophenyl)methyl]-5-{1-[2-(methylsulfanyl)acetyl]piperidin-4-yl}imidazolidine-2,4-dione
[(4-chloro-1-methyl-1H-indazol-3-yl)methyl](methyl)[2-(1-methyl-1H-pyrazol-4-yl)ethyl]amine
2-{[3-(3-{furo[3,2-c]pyridin-4-yl}phenyl)-1H-pyrazol-1-yl]methyl}-1,3-thiazole
3-[1-(1-benzoxepine-4-carbonyl)azetidin-3-yl]pyridine
1-(1-ethyl-2,5-dimethyl-1H-pyrrole-3-carbonyl)-2-[2-(1H-pyrazol-1-yl)ethyl]piperidine
2-cyclopropyl-3-[4-(2,4-dimethylphenyl)piperazine-1-carbonyl]-6-methyl-1-(thiophen-2-ylmethyl)-1,4-dihydropyridin-4-one
3-methoxy-1-[3-(4-phenylpiperazin-1-yl)piperidin-1-yl]propan-1-one
5-(1H-imidazol-2-yl)-4-phenyl-1-[(5-phenyl-1H-pyrazol-3-yl)methyl]-1H-imidazole
(4aS,8aR)-6-(2-amino-5,6,7,8-tetrahydroquinazoline-4-carbonyl)-1-(3-methylbutyl)-decahydro-1,6-naphthyridin-2-one
N-{2-[2-(2,3-dimethoxyphenyl)-1H-imidazol-1-yl]ethyl}-3-methylpyridin-2-amine
(3aR,6aR)-2-(cyclopentylcarbamoyl)-5-(pyridin-3-ylmethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
9-hydroxy-4-oxo-N-[2-(3-phenylpyrrolidin-1-yl)ethyl]-4H-pyrido[1,2-a]pyrimidine-3-carboxamide
2-[3-(2-hydroxyethyl)-4-[(3-methoxyphenyl)methyl]piperazin-1-yl]ethan-1-ol
(3S,4R)-1-(5-fluoropyrimidin-2-yl)-4-(4-methoxyphenyl)-N,N-dimethylpyrrolidin-3-amine
1-[(3-fluorophenyl)methyl]-4-(6-oxo-1,6-dihydropyridine-3-carbonyl)piperazin-2-one
1-(but-2-ynoyl)-N-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]piperidine-4-carboxamide
1-cyclopentyl-4-[5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]-1,4-diazepane
6-[1-(dimethyl-1,3-thiazole-4-carbonyl)piperidin-4-yl]pyrimidin-4-ol
9-(2-methoxyethyl)-1-methyl-4-(morpholine-4-carbonyl)-1,4,9-triazaspiro[5.6]dodecan-10-one
4-{[(5-methyl-2-{3-[2-(4-methylphenoxy)acetamido]phenyl}-1,3-oxazol-4-yl)methyl]carbamoyl}pyridin-1-ium-1-olate
(1R,5S,8S)-8-methoxy-3-(5-propyl-1,3,4-oxadiazol-2-yl)-3-azabicyclo[3.2.1]octane
7-(cyclobutylmethyl)-2-[(3-phenyl-1,2-oxazol-5-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one
3-[4-(dimethylamino)-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]pyridin-2-ol
1-[4-(hydroxymethyl)-4-[(3-methoxyphenyl)methyl]piperidin-1-yl]-3-phenylprop-2-yn-1-one
3-methyl-2-[(1-methyl-1H-imidazol-2-yl)methyl]-1-phenyl-1,2-diazinane
1-(9H-fluoren-2-ylmethyl)-4-(2-methoxyethyl)-1,4-diazepan-5-one
1-(3-chloro-2-methylphenyl)-3-methyl-3-[3-(1-methyl-1H-pyrazol-4-yl)propyl]urea
(3S,4R)-4-(2,3-dimethoxyphenyl)-1-(1H-pyrrole-2-carbonyl)pyrrolidine-3-carboxylic acid
1-{[2-(2,4-dimethoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-3-propyl-1H-1,2,4-triazole
1-[4-(2-methoxyphenyl)-2-methylpiperazin-1-yl]-3-(1H-1,2,3,4-tetrazol-1-yl)propan-1-one
2-({[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl](methyl)amino}methyl)-6-methoxyphenol
N-[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]-N,1,3,6-tetramethyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-(2-fluoro-4-methylphenyl)-3-methyl-3-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]urea
3-phenoxy-1-[2-(thiomorpholine-4-carbonyl)morpholin-4-yl]propan-1-one
N-(2-methoxyethyl)-4-methyl-3-[(methylcarbamoyl)methyl]-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
1-cyclopropanecarbonyl-3-[(2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazol-1-yl)methyl]piperidine
3,5-dimethyl-1-(1-{[5-(oxan-2-yl)furan-2-yl]methyl}azetidin-3-yl)-1H-pyrazole
1-[2-amino-4-(2,5-dihydro-1H-pyrrol-1-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl]-3-(1H-imidazol-1-yl)propan-1-one
2-{1-[3-(1H-pyrazol-1-yl)benzoyl]azetidin-3-yl}pyridine
4-({4-[1-(2-methylphenyl)-1H-pyrazol-4-yl]-1,2,3,6-tetrahydropyridin-1-yl}methyl)benzoic acid
3-(1-{[2-(ethanesulfonyl)-1-(2-phenylethyl)-1H-imidazol-5-yl]methyl}piperidin-3-yl)propan-1-ol
3-(quinolin-4-ylmethyl)-3H,4H-pyrido[2,3-d]pyrimidin-4-one
2-methoxy-N-{2-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]phenyl}acetamide
4-{[2-(2-methoxyethyl)-3-oxo-2,9-diazaspiro[5.5]undecan-9-yl]methyl}-N-methylbenzamide
N-({5-cyclobutanecarbonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-1-ethyl-1H-pyrazole-4-carboxamide
N-(1-methyl-1H-pyrazol-5-yl)-2-[4-(4-phenoxyphenyl)-1H-pyrazol-1-yl]acetamide
4-{4-[1-(pyrrolidin-1-yl)ethyl]phenyl}pyridin-2-amine
1-{3-methyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}-4-(oxolan-2-ylmethyl)piperazine