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[(4-{6-tert-butyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-1,4-oxazepan-6-yl)methyl]dimethylamine
2-[(3,4-dimethoxyphenyl)methyl]-N-methyl-N-[1-(pyridin-2-yl)ethyl]-1,3-benzoxazole-6-carboxamide
(2,1,3-benzoxadiazol-5-ylmethyl)({1-[2-(4-methoxyphenyl)ethyl]piperidin-4-yl}methyl)methylamine
3-(4-tert-butylbenzoyl)-1-(1H-pyrazol-3-ylmethyl)piperidine
4-chloro-1,5-dimethyl-N-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)-1H-pyrazole-3-carboxamide
1-[(4-chlorophenyl)methyl]-N-{[1-(2-phenylethyl)piperidin-4-yl]methyl}-1H-1,2,3-triazole-4-carboxamide
N-[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl]-N-ethylmorpholine-2-carboxamide
1-(oxan-4-yl)-N-{2-[(pyridin-3-yl)amino]ethyl}piperidine-3-carboxamide
7-(cyclopropylmethyl)-N-(4-ethoxyphenyl)-6-oxo-2,7-diazaspiro[4.5]decane-2-carboxamide
2-{2-[(3-{[2-(3,4-dimethoxyphenyl)ethyl](methyl)amino}piperidin-1-yl)methyl]phenoxy}ethan-1-ol
ethyl 4-[7-(cyclohexylmethyl)-2,7-diazaspiro[4.5]decan-2-yl]piperidine-1-carboxylate
2-amino-4-[1-(2-hydroxyethyl)-3-methyl-1H-pyrazol-4-yl]-6-(2-methylphenyl)pyridine-3-carbonitrile
2-[(1S,6R)-3,9-diazabicyclo[4.2.1]nonane-9-carbonyl]-4H-chromen-4-one
1-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-5-(2-{[2-(4-fluorophenoxy)ethyl]amino}ethyl)pyrrolidin-2-one
methyl 2-[7-(5-chloropyridin-2-yl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]propanoate
4-[4-(2-methylphenyl)-3-oxopiperazine-1-carbonyl]benzene-1-sulfonamide
1-{4-[3-(4-benzylpiperidin-1-yl)-3-oxopropyl]piperidin-1-yl}-2-hydroxypropan-1-one
2-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-6-methylpyridine
2-methyl-8-{7-methyl-2,7-diazaspiro[4.4]nonane-2-carbonyl}-1,4-dihydroquinolin-4-one
5-(4-methoxy-2,3,6-trimethylphenyl)-1-methyl-1H,4H-pyrazolo[3,4-d]imidazole
1-{[4-(methylsulfanyl)phenyl]methyl}-4-(pyrrolidine-1-sulfonyl)-1,4-diazepane
2-{4-[(1S,4S)-2,5-diazabicyclo[2.2.1]heptan-2-yl]-6-methylpyrimidin-2-yl}phenol
N-methyl-N-{2-[(4-methylphenyl)sulfanyl]ethyl}-2-(propan-2-yl)pyrimidine-4-carboxamide
(4aS,8aR)-6-(1-methyl-1H-imidazole-5-carbonyl)-1-(2-phenylethyl)-decahydro-1,6-naphthyridin-2-one
N-{1-[(4-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}methanesulfonamide
2-{[4-(dimethylamino)-5-methylpyrimidin-2-yl]amino}-N-(5-fluoro-2-methylphenyl)propanamide
N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}-N-[3-(dimethylamino)propyl]propanamide
N-(2,3-dihydroxypropyl)-2-[methyl(2-phenylethyl)amino]-2,3-dihydro-1H-indene-2-carboxamide
3-(2H-1,3-benzodioxol-5-yl)-3-phenyl-N-{5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridin-3-ylmethyl}propanamide
7-[2-(3-fluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]-1,3-diazepane-2,4-dione
5-chloro-2-fluoro-N-methyl-N-[(1-phenylpyrrolidin-3-yl)methyl]benzamide
(3S,4S)-1-{6-[(dimethylamino)methyl]pyrazin-2-yl}-4-(naphthalen-2-yl)piperidin-3-ol
ethyl 4-(5-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-1,2-oxazole-3-carbonyl)piperazine-1-carboxylate
2-(methoxymethyl)-1-{5-[2-(methylsulfanyl)phenoxymethyl]-1,2-oxazole-3-carbonyl}piperidine
3-{2-[1-({5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl}methyl)piperidin-2-yl]ethyl}phenol
2-({5-[3-(2,3-dimethoxyphenyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}amino)-3-methylbutan-1-ol
N-[2-(cyclohex-1-en-1-yl)ethyl]-N-(cyclopropylmethyl)-9-oxo-1-azatricyclo[6.3.1.04,12]dodeca-4(12),5,7,10-tetraene-10-carboxamide
ethyl 2-{[(3aS,6aR)-3-[2-(4-methoxyphenyl)ethyl]-2-oxo-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazole-5-carbonyl]amino}acetate
3-butanamido-N-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]benzamide
1-[(1S,5R)-3-acetyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-3-(3-methoxyphenyl)propan-1-one
N-[2-(benzyloxy)ethyl]-1,3-dimethyl-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
8-(9H-purin-6-yl)-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
2-[(3-ethyl-1H-1,2,4-triazol-5-yl)sulfanyl]-N-[2-(furan-2-yl)-2-(pyrrolidin-1-yl)ethyl]acetamide
N-[(4-methoxyphenyl)methyl]-1-methyl-3-(piperidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
3-[(3R,4S)-3-{2-[4-(hydroxymethyl)phenyl]acetamido}-4-(propan-2-yl)pyrrolidin-1-yl]propanoic acid
{[5-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}(3-phenylprop-2-yn-1-yl)propylamine
5-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}-2-cyclopropyl-4-methylpyrimidine
2-butyl-N-(1H-indol-5-yl)-4-methyl-3-oxopiperazine-1-carboxamide
1-{4-[3-(furan-2-yl)benzoyl]-6-hydroxy-1,4-diazepan-1-yl}ethan-1-one
N-ethyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)-1H-pyrrole-3-carboxamide