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1-cyclopropyl-N-[2-(4,6-dimethylpyrimidin-2-yl)ethyl]-5-oxopyrrolidine-3-carboxamide
N-[(5-methylpyrazin-2-yl)methyl]-2-(piperidin-1-yl)-2,3-dihydro-1H-indene-2-carboxamide
4-[2-(dimethylamino)-2-(3-fluorophenyl)acetyl]-N,N-dimethylpiperazine-1-carboxamide
N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}-3-(5-methylfuran-2-yl)benzamide
N-[1-ethyl-2-(pyridin-3-yl)-7-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-1H-1,3-benzodiazol-5-yl]-2-methoxyacetamide
4-phenyl-5-[3-(pyridin-3-yl)azetidine-1-carbonyl]pyrimidin-2-amine
6-methyl-2-{2-[(4-phenyl-1,4-diazepan-1-yl)methyl]phenyl}-3,4-dihydropyrimidin-4-one
1,4,6-trimethyl-3-{3-[methyl(2-phenylethyl)amino]piperidine-1-carbonyl}-1,2-dihydropyridin-2-one
N-[2-(1H-imidazol-4-yl)ethyl]-1-phenyl-1H-1,2,3-triazole-4-carboxamide
(3R,5S)-N-[(5-methyl-1H-1,2,4-triazol-3-yl)methyl]-5-(morpholine-4-carbonyl)piperidine-3-carboxamide
1-(4-{4-[1-(2-fluorophenyl)-1H-pyrazol-4-yl]pyrimidin-2-yl}-1,4-diazepan-1-yl)ethan-1-one
4-cyclobutyl-N,6-dimethyl-N-(pyrazin-2-ylmethyl)pyrimidin-2-amine
2-acetyl-8-[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
5-{[3-(3-chlorophenyl)pyrrolidin-1-yl]methyl}-2-(pyrrolidin-1-yl)-1,3-thiazole
N-({5-cyclohexyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-1,3-benzoxazol-2-amine
1-[(3R,5R)-3-[(dimethylamino)methyl]-5-(hydroxymethyl)piperidin-1-yl]-2-(4-phenylpiperidin-1-yl)ethan-1-one
2-methoxy-N-({2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}methyl)quinoline-4-carboxamide
[(2-methoxyphenyl)methyl](methyl)({4-methyl-5-[(2-phenoxyethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)amine
2-(furan-2-yl)-5-[(3-propoxypiperidin-1-yl)methyl]pyrimidine
{[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]methyl}[(1-methyl-1H-imidazol-2-yl)methyl](propan-2-yl)amine
1-cyclohexyl-4-(1-{8-methoxy-5H,6H-benzo[h]quinazolin-2-yl}-5-methyl-1H-pyrazole-4-carbonyl)piperazine
N-[(2-fluorophenyl)methyl]-3-[1-(oxane-4-carbonyl)piperidin-3-yl]propanamide
5-{1-[2-(1-methyl-1H-pyrrol-3-yl)acetyl]pyrrolidin-2-yl}-N-propylthiophene-2-carboxamide
N-[(1-ethyl-1H-imidazol-2-yl)methyl]-5-[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]pyridin-2-amine
(2S,4S)-4-amino-1-(2,6-dichlorobenzenesulfonyl)-N-(propan-2-yl)pyrrolidine-2-carboxamide
4-(2-ethoxyphenyl)-3-[(trimethyl-1H-pyrazol-1-yl)methyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
4-{[3-(4-butylpiperazine-1-carbonyl)-1,2-oxazol-5-yl]methyl}morpholine
2-{1-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]piperidin-4-yl}-1-methyl-1H-1,3-benzodiazole
(2S,4R)-4-cyclobutaneamido-N-ethyl-1-[(1-methyl-1H-imidazol-2-yl)methyl]pyrrolidine-2-carboxamide
3-[3-(4-phenylphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-1,2-oxazole
(1S,5R)-3-[(dimethyl-1,2-oxazol-4-yl)methyl]-6-(thiophene-2-sulfonyl)-3,6-diazabicyclo[3.2.2]nonane
3-[(2-methyl-1H-imidazol-1-yl)methyl]-1-(3-phenylpropyl)piperidine
N-(2-methanesulfonylethyl)-1,6-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-({1-[2-(4-methyl-1,2,5-oxadiazol-3-yl)acetyl]piperidin-3-yl}methyl)-1H-indole-2-carboxamide
N-cyclopropyl-1-[(1s,4s)-4-(4-chlorobenzamido)cyclohexyl]-1H-1,2,3-triazole-4-carboxamide
1-[5-(furan-3-ylmethyl)-1-[(3-methoxyphenyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]piperidin-3-ol
2,6-dimethyl-N-[2-(4-methyl-1H-1,2,3-triazol-1-yl)ethyl]pyrimidine-4-carboxamide
(2S,4S)-N-ethyl-1-(3-ethyl-1H-pyrazole-5-carbonyl)-4-(furan-2-amido)pyrrolidine-2-carboxamide
2-phenyl-1-(1-{2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-yl}piperidin-4-yl)ethan-1-ol
N-methyl-N-{[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}-2-(thiophen-3-yl)acetamide
4-fluoro-3-methoxy-N-methyl-N-[2-(4-methylpiperidin-1-yl)ethyl]benzamide
3-{2-[1-(3-methylbutyl)-3-(morpholine-4-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-2-oxoethyl}-2,3-dihydro-1,3-benzoxazol-2-one
N-[2-(4-{1-[(4-fluorophenyl)methyl]-3-methyl-1H-1,2,4-triazol-5-yl}phenoxy)ethyl]acetamide
N-methyl-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-2-[(4S)-2-oxo-4-phenyl-1,3-oxazolidin-3-yl]acetamide
3,3,3-trifluoro-N-[(3R,4S)-1-[(1-methyl-1H-imidazol-5-yl)methyl]-4-(propan-2-yl)pyrrolidin-3-yl]propanamide
(3S,4S)-1-(4-chloro-1-ethyl-1H-pyrazole-5-carbonyl)-4-propylpyrrolidine-3-carboxylic acid
[(3R,4R)-4-(morpholin-4-ylmethyl)-1-{thieno[2,3-d]pyrimidin-4-yl}pyrrolidin-3-yl]methanol
1-[(3-fluorophenyl)methyl]-4-[4-(thiophen-2-yl)butanoyl]piperazin-2-one
3-(2-methoxyethyl)-1-(6-phenylpyridazin-3-yl)piperidine-3-carboxylic acid
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-1-[2-(3-fluorophenyl)ethyl]-6-oxopiperidine-3-carboxamide