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(1S,5R)-3-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}-3,9-diazabicyclo[3.3.2]decan-10-one
(1S,6R)-9-[(4,5-dichlorothiophen-2-yl)sulfonyl]-3,9-diazabicyclo[4.2.1]nonane
2-(4-{[(furan-3-ylmethyl)(methyl)amino]methyl}phenyl)-6-(pyridin-4-yl)-3,4-dihydropyrimidin-4-one
N-({5-methanesulfonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-(propylsulfanyl)acetamide
1-(4-methylpiperazin-1-yl)-3-(1-{[4-(1H-pyrazol-1-yl)phenyl]methyl}piperidin-3-yl)propan-1-one
5-(4-fluorophenoxymethyl)-3-(2,3,4-trimethoxyphenyl)-1,2,4-oxadiazole
4-[4-(pyridin-3-ylmethoxy)piperidine-1-carbonyl]-1-oxaspiro[4.4]nonan-2-one
N-cyclopentyl-N-{[4-methoxy-3-(propan-2-yloxy)phenyl]methyl}pyridine-3-carboxamide
2-benzyl-N-(2-methylphenyl)-3-oxo-2,9-diazaspiro[5.5]undecane-9-carboxamide
N-[1-(1-ethyl-1H-1,2,4-triazol-5-yl)ethyl]-5-(2-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-amine
N-[(1R,2R)-2-(benzyloxy)cyclopentyl]-1-phenyl-1H-1,2,3-triazole-4-carboxamide
1-[6-(hydroxymethyl)-1,4-oxazepan-4-yl]-4-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}butan-1-one
N-(1-benzyl-1H-pyrazol-3-yl)-2-[3,5-dimethyl-4-(5-methylfuran-2-yl)-1H-pyrazol-1-yl]acetamide
4-(4-chlorophenyl)-N-[(3S,4S)-4-hydroxy-1,1-dioxo-1λ6-thiolan-3-yl]-N-methylbutanamide
(1R,9aR)-1-(3-methylphenoxymethyl)-octahydro-1H-quinolizine
N-(2-fluoro-4-methylphenyl)-3-(3-methoxyphenoxymethyl)piperidine-1-carboxamide
N-{2-[5-(hydroxymethyl)-1,2,4-oxadiazol-3-yl]ethyl}-1H-indazole-3-carboxamide
N-(1-phenylethyl)-2-(1H-pyrrole-2-carbonyl)-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
6-{3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine-2-carbonitrile
4-[2-oxo-4-(3,3,4,4-tetrafluorobutyl)piperazin-1-yl]benzonitrile
3-(4,5-dimethyl-1H-pyrazol-3-yl)-1-[3-(1H-pyrazol-5-yl)piperidin-1-yl]propan-1-one
1-({5-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl]furan-2-yl}methyl)pyrrolidine
(2E)-N-{[5-(3,6-dimethylpyrazin-2-yl)-7-fluoro-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-(thiophen-2-yl)prop-2-enamide
N-[(3R,4R)-3-hydroxy-1-[2-(pyridin-4-yl)acetyl]piperidin-4-yl]pyridine-4-carboxamide
2-hydroxy-N-{[1-(3,3,3-trifluoropropyl)piperidin-3-yl]methyl}acetamide
4-hydroxy-N-methyl-N-[(4-methyl-1,3-thiazol-2-yl)methyl]-2-[(phenylsulfanyl)methyl]pyrimidine-5-carboxamide
1-(3,4-difluorobenzoyl)-2-(3-methoxyphenyl)piperidine
(3S,4S)-4-(piperidin-1-yl)-1-(3,4,7-trimethyl-1H-indole-2-carbonyl)pyrrolidin-3-ol
4-(2-ethylpyrrolidine-1-carbonyl)-2,5,7-trimethylquinoline
5-[3-(2-methylphenoxy)azetidine-1-carbonyl]-4-phenylpyrimidin-2-amine
2-methoxy-N-[1-(2-methylpropanoyl)piperidin-4-yl]quinoline-4-carboxamide
4-[5-(2-ethoxypyridin-3-yl)furan-2-carbonyl]morpholine
2-{[(4S)-4-hydroxy-4-(methoxymethyl)-3,3-dimethylpiperidin-1-yl]methyl}benzoic acid
N-[2-(4-amino-6-hydroxypyrimidin-2-yl)ethyl]-1-(2-phenylethyl)-1H-1,2,3-triazole-4-carboxamide
(3R,4R)-1-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-3-methyl-4-(oxan-4-yl)piperidin-4-ol
3-(2-chlorophenyl)-1-(4-methoxypiperidin-1-yl)-3-phenylpropan-1-one
2-chloro-4-{[(propan-2-yl)[(trimethyl-1H-pyrazol-4-yl)methyl]carbamoyl]amino}benzamide
6-[(2-{imidazo[1,2-a]pyridin-3-yl}ethyl)amino]pyridine-3-carboxamide
4-{[(2,3-dihydro-1H-inden-2-yl)(methyl)amino]methyl}-5-(hydroxymethyl)-2-methylpyridin-3-ol
1-{2-[3-(thiophen-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl}ethan-1-one
1-{[1-methyl-3-(4-phenoxyphenyl)-1H-pyrazol-4-yl]methyl}-4-(pyridin-3-ylmethyl)piperazine
2-{1'-[(4-hydroxy-3-methylphenyl)methyl]-2-oxo-1,2-dihydrospiro[indole-3,3'-pyrrolidine]-1-yl}acetamide
2-methoxy-4-({1-[methyl(1-methylpiperidin-4-yl)amino]hex-5-en-2-yl}oxy)pyridine-3-carbonitrile
7-(4-amino-6-fluoroquinoline-3-carbonyl)-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide
8-[(2E)-but-2-en-1-yl]-2-[2-(pyridin-2-yl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N-methyl-N-[1-(1,2-oxazol-3-yl)ethyl]benzamide
({5-[1-(1-benzofuran-5-ylmethyl)piperidin-3-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)dimethylamine
3-[(2-ethylbutyl)amino]-N-[2-(1H-imidazol-1-yl)ethyl]-5-(pyrrolidine-1-sulfonyl)benzamide
3-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-N-phenylpiperidine-1-carboxamide
4-methyl-6-{4-[(2-propylpyrimidin-5-yl)methyl]piperazin-1-yl}pyrimidin-2-amine