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2-methoxy-N-(1-{1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]piperidin-4-yl}-1H-pyrazol-5-yl)benzamide
(1R,5S,6R,7S)-3-methyl-4-oxo-N-[(1r,4r)-4-(4H-1,2,4-triazol-4-yl)cyclohexyl]-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
1-{3-[(2R,6R)-6-methyl-2-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridine-1-carbonyl]phenyl}imidazolidin-2-one
2-[(1S,5R)-3-(4,6-dimethoxypyrimidin-2-yl)-7-oxo-3,6-diazabicyclo[3.2.2]nonan-6-yl]-N,N-dimethylacetamide
6-fluoro-3-(2-methoxyethyl)-3,4-dihydroquinazolin-4-one
N-(2-hydroxyethyl)-1-{1-[(4-methoxynaphthalen-1-yl)methyl]piperidin-3-yl}-N-methyl-1H-1,2,3-triazole-4-carboxamide
2-{4-[(dimethylamino)methyl]phenyl}pyridin-4-amine
1-cyclopentyl-4-{[4-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-1,4-diazepane
[(6-fluoroquinolin-2-yl)methyl]({1-[2-(4-methoxyphenyl)ethyl]piperidin-4-yl}methyl)methylamine
N-({5-cyclobutanecarbonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)cyclopentanecarboxamide
1-{4-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]piperidin-1-yl}-2-phenoxypropan-1-one
4-(2-{[4-(trifluoromethyl)pyrimidin-2-yl]oxy}hex-5-en-1-yl)morpholine
(1R,7S)-3-(3,4-dimethylphenyl)-N-methyl-4-oxo-N-(pyrimidin-4-ylmethyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
1-{7-methyl-6-oxo-2,7-diazaspiro[4.5]decan-2-yl}-2-(pyridin-3-yl)ethane-1,2-dione
4-[4-(trifluoromethyl)pyridin-2-yl]benzamide
(4aS,8aR)-1-(2-aminoethyl)-6-{[5-(1H-pyrazol-3-yl)thiophen-2-yl]methyl}-decahydro-1,6-naphthyridin-2-one
2-{4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}pyridine
2-[1-(furan-3-ylmethyl)-3-oxopiperazin-2-yl]-N-[2-(1H-indol-1-yl)ethyl]acetamide
2-methoxy-4-{3-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine-3-carbonitrile
N-(4,6-dimethyl-2-oxo-1,2-dihydropyridin-1-yl)-2-(4-fluorophenoxy)acetamide
9-(2,6-dimethylquinoline-4-carbonyl)-5-methoxy-1-oxa-9-azaspiro[5.5]undecane
N-[2-(2-methyl-1H-indol-1-yl)ethyl]-1H-1,2,3-triazole-5-carboxamide
1-[2-(4-methoxyphenyl)ethyl]-N-[3-(methylsulfanyl)propyl]-6-oxopiperidine-3-carboxamide
8-(3,3-dimethylbutanoyl)-2-[2-(1H-imidazol-4-yl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
4-[3-(1-benzyl-1H-imidazol-2-yl)piperidin-1-yl]-6-methylpyrimidin-2-amine
3-methanesulfonamido-N-{1-[4-methyl-2-(pyridin-4-yl)pyrimidin-5-yl]ethyl}propanamide
5-(2-{[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]amino}ethyl)-1-{[2-fluoro-4-(trifluoromethyl)phenyl]methyl}pyrrolidin-2-one
3-[1-(1-benzofuran-2-ylmethyl)piperidin-3-yl]-N-[(2,4-dimethoxyphenyl)methyl]propanamide
2-[1-(furan-2-ylmethyl)-4-[4-(propan-2-yl)pyrimidin-2-yl]piperazin-2-yl]ethan-1-ol
N-[2-methyl-2-(1,2,3,4-tetrahydroisoquinolin-2-yl)propyl]-2,7-dioxo-1,3-diazepane-4-carboxamide
2-(5-amino-1,3,4-thiadiazol-2-yl)-N-[1-(2,4-dimethylphenyl)propyl]acetamide
3-(azepane-1-carbonyl)-1-methyl-5-(thiomorpholin-4-yl)-4,5,6,7-tetrahydro-1H-indazole
N-(1,3-thiazol-2-ylmethyl)-3,4-dihydro-2H-1-benzopyran-3-carboxamide
N-[(3-methylthiophen-2-yl)methyl]-4-(1,2,3,6-tetrahydropyridine-1-carbonyl)aniline
1-[(4-methyl-5-{1-[3-(methylsulfanyl)propyl]piperidin-3-yl}-4H-1,2,4-triazol-3-yl)methyl]piperidin-4-ol
1-methyl-N-{[2-(pyridin-2-yl)pyrimidin-5-yl]methyl}-N-(pyridin-3-ylmethyl)piperidin-4-amine
7-(cyclopropylmethyl)-2-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}-2,7-diazaspiro[4.5]decan-6-one
1-methyl-3-{[3-(pyridin-3-yl)azetidin-1-yl]methyl}-1,2-dihydroquinolin-2-one
4-(hydroxymethyl)-1-(2-methyl-1H-1,3-benzodiazole-4-carbonyl)piperidin-4-ol
6-[1-(furan-2-ylmethyl)piperidin-3-yl]-2-(pyrazin-2-yl)-3,4-dihydropyrimidin-4-one
3-(2-{[4-(pyridin-2-yl)pyrimidin-2-yl]amino}ethyl)-1,3-oxazinan-2-one
1-{4-[4-ethyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-3-(1H-1,2,4-triazol-1-yl)propan-1-one
8-methoxy-N-[(3-methylquinoxalin-2-yl)methyl]-3,4-dihydro-2H-1-benzopyran-3-amine
3-[1-(5-fluoro-2-methylbenzenesulfonyl)piperidin-4-yl]-N-(3-methoxyphenyl)propanamide
2-methyl-8-(5-propyl-1,3,4-oxadiazol-2-yl)-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
N-(3-methyl-1-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}butyl)-6-oxo-1,6-dihydropyridine-3-carboxamide
N-cyclopropyl-5-(quinoxalin-2-yl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
N-phenyl-5-(2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazol-1-yl)pyridin-2-amine
8-(cyclopentylcarbamoyl)-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
2-{3-oxo-1-[(4-phenylphenyl)methyl]piperazin-2-yl}-N-[2-(propan-2-yloxy)ethyl]acetamide