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1-(4-{5-cyclopropyl-1-[4-(2-methoxyphenyl)pyrimidin-2-yl]-1H-pyrazole-4-carbonyl}piperazin-1-yl)ethan-1-one
(2S,4S)-1-[(3-cyclohexyl-1,2-oxazol-5-yl)methyl]-N-ethyl-4-(2-hydroxyacetamido)pyrrolidine-2-carboxamide
N-{[7-(3,6-dimethylpyrazin-2-yl)-4-fluoro-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(2-methyl-1H-indol-3-yl)acetamide
5-[(3-methylthiophen-2-yl)methyl]-2-(3,4,5-trimethoxyphenyl)-2,3,4,5-tetrahydro-1,5-benzothiazepine
N,1-dimethyl-3-(2-methylpropyl)-N-[1-(pyridin-3-yl)ethyl]-1H-pyrazole-5-carboxamide
1-[(4-methoxypyridin-2-yl)methyl]-4-phenyl-3-(piperidin-3-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
3-(1-butyl-1H-imidazol-2-yl)-1-{pyrazolo[1,5-a]pyrimidine-2-carbonyl}piperidine
N-{[1-(1,3-dihydroxypropan-2-yl)pyrrolidin-3-yl]methyl}-4,5,6,7-tetrahydro-2-benzothiophene-1-carboxamide
N-[1-(1-methyl-1H-pyrazol-4-yl)propyl]-4-(propylsulfamoyl)benzamide
3-{1-[3-(trifluoromethyl)-1H-pyrazole-5-carbonyl]piperidin-3-yl}propanamide
(3aS,6aR)-5-[6-(dimethylamino)pyrimidin-4-yl]-3-[3-(4-methoxyphenyl)propyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
4-[2-(1-{[2-(pyridin-2-yl)pyrimidin-5-yl]methyl}piperidin-2-yl)ethyl]morpholine
N-{3-[(furan-2-ylmethyl)sulfanyl]propyl}-3,6-dimethyl-[1,2]oxazolo[5,4-d]pyrimidin-4-amine
1-[(3-cyclopropyl-1H-pyrazol-5-yl)methyl]-4-(2-methyl-1H-pyrrole-3-carbonyl)-1,4-diazepan-6-ol
(3R,9aR)-3-[(1S)-1-hydroxyethyl]-8-(4-phenylbenzoyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
5-[4-(1-hydroxy-3-phenylpropyl)piperidine-1-carbonyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-[(2-fluorophenyl)methyl]-3-{1-[1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]piperidin-3-yl}propanamide
2-[3-(pyridin-3-yl)azetidin-1-yl]-1-(pyrrolidin-1-yl)propan-1-one
N-{pyrazolo[1,5-a]pyridin-3-ylmethyl}-1-(pyridin-2-yl)piperidine-3-carboxamide
5-(3,4-dimethylphenyl)-4-(4-methylphenyl)-N-(1H-1,2,3,4-tetrazol-5-ylmethyl)pyrimidin-2-amine
({1-[2-(4-methoxyphenyl)ethyl]piperidin-3-yl}methyl)(methyl)[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]amine
5-(propan-2-yl)-N-{[1,2,4]triazolo[4,3-a]pyridin-3-ylmethyl}pyrazolo[1,5-a]pyrimidin-7-amine
3-(1-methanesulfonylpiperidin-4-yl)-1-[2-methyl-3-(pyrrolidin-1-yl)phenyl]urea
3-cyclopropyl-1-(2,3-dihydro-1H-inden-2-yl)-5-[1-(methylsulfanyl)ethyl]-1H-1,2,4-triazole
(3R,5S)-N-[(4,6-dimethylpyridin-3-yl)methyl]-5-(pyrrolidine-1-carbonyl)piperidine-3-carboxamide
4-{4-[(2-ethoxyphenyl)methyl]piperazin-1-yl}-2-[(2-fluorophenyl)methyl]-2,3-dihydro-1H-isoindole-1,3-dione
(1R,5R)-6-[(3,5-dichloropyridin-4-yl)methyl]-3-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonane
6-(3,5-dimethyl-1H-pyrazol-4-yl)-N,N-dimethylpyridine-2-carboxamide
1-methyl-N-(1,2-oxazol-3-ylmethyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-[1-(4-hydroxyphenyl)ethyl]-2-(2,2,6,6-tetramethylpiperidin-4-yl)acetamide
5-{1-[(3-chlorophenyl)methyl]-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}-1-methyl-1H-imidazole
9-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-2-[2-(1H-imidazol-4-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
N-(2-methylprop-2-en-1-yl)-1-[1-(propan-2-yl)piperidin-4-yl]piperidine-3-carboxamide
5-[(3aR,6aS)-octahydropyrrolo[3,4-c]pyrrole-2-carbonyl]-2-(adamantan-1-yl)pyrimidin-4-ol
1-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-3-{[4-(pyrrolidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]methyl}piperidine
1-methyl-4-{4-[1-(morpholin-4-yl)ethyl]phenyl}phthalazine
N-({2-[benzyl(methyl)amino]pyridin-3-yl}methyl)-2-(morpholin-2-yl)acetamide
1-[3-(1H-imidazol-2-yl)benzoyl]-4-(2-methoxyphenyl)-2-methylpiperazine
3-ethyl-3-[(5-methylfuran-2-yl)methyl]-1-(5,7,8-trimethyl-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-6-yl)urea
2-(4-fluorophenyl)-N-(2-{7-[2-(2,6,6-trimethylcyclohex-1-en-1-yl)ethyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)acetamide
[(5-cyclopropyl-1-methyl-1H-pyrazol-4-yl)methyl][(1,5-dimethyl-1H-pyrazol-4-yl)methyl]methylamine
N-{[1-(methoxymethyl)cyclopentyl]methyl}-2-methyl-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-amine
1-{imidazo[1,2-a]pyrimidine-2-carbonyl}-4-(1H-pyrazol-1-yl)piperidine-4-carboxylic acid
2-methoxy-N-(5-oxo-1-{[2-(trifluoromethyl)phenyl]methyl}pyrrolidin-3-yl)acetamide
4-[4-(cyclopropylamino)piperidin-1-yl]-N-(1-phenylethyl)benzamide
3-(azepane-1-carbonyl)-N-methyl-1-(prop-2-en-1-yl)-N-(thiophen-3-ylmethyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
8-{[4-(pyrrolidine-1-carbonyl)-1,3-oxazol-2-yl]methoxy}quinoline
1'-[6-oxo-2-(propan-2-yl)-1,6-dihydropyrimidine-5-carbonyl]-1,2-dihydrospiro[indole-3,3'-piperidine]-2-one
2-(3-chlorophenyl)-5-methyl-4-[(4-methyl-1H-imidazol-1-yl)methyl]-1,3-oxazole
2-methyl-4-[3-(2-phenylethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine-7-carbonyl]-1,3-thiazole