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1-{1'-[5-(hydroxymethyl)furan-2-carbonyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}propan-1-one
2-({[5-(1-cyclopentylpiperidin-4-yl)-4-methyl-4H-1,2,4-triazol-3-yl]methyl}(methyl)amino)ethan-1-ol
4-{3-[4-(2-propoxyethyl)piperazine-1-carbonyl]phenyl}phenol
2-methyl-3-{3-[3-(trifluoromethyl)benzoyl]piperidine-1-carbonyl}pyridine
5-[1-(2-fluorobenzoyl)piperidin-4-yl]-5-(pyridin-2-yl)-3-[2-(thiophen-2-yl)ethyl]imidazolidine-2,4-dione
1-(cyclohexylmethyl)-4-{[3-(3-methoxyphenyl)-1,2-oxazol-5-yl]methyl}piperidin-4-ol
6-{[3-(morpholin-4-yl)propyl]amino}-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3(8),6,12,14-pentaen-4-one
1-(2-oxo-2-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}ethyl)-1,2-dihydroquinolin-2-one
1-cyclopentyl-4-{[4-(1-ethyl-1H-1,3-benzodiazol-2-yl)-1H-1,2,3-triazol-1-yl]methyl}pyrrolidin-2-one
(1R,2R)-2-[5-(1H-imidazol-1-ylmethyl)-3-[(2-methoxyphenyl)methyl]-1H-1,2,4-triazol-1-yl]cyclohexan-1-ol
N,2-dimethyl-6-(piperidin-3-yl)-N-{[3-(1H-1,2,3,4-tetrazol-5-yl)phenyl]methyl}pyrimidin-4-amine
N-[2-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)ethyl]-2-(4-ethyl-5-oxo-3-phenyl-4,5-dihydro-1H-1,2,4-triazol-1-yl)acetamide
N-phenyl-5-(pyridin-3-yl)furan-2-carboxamide
N-[2-(dimethylamino)ethyl]-N-methyl-1-(2-methyl-4-phenylpyrimidine-5-carbonyl)piperidin-3-amine
(2R,6R)-4-cyclopentanecarbonyl-10-methoxy-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
[(3R,4S)-4-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-1-[(5-ethylpyridin-2-yl)methyl]pyrrolidin-3-yl]methanol
{[1-(2,4-difluorophenyl)-3-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}[3-(morpholin-4-yl)propyl]amine
(1S,9S)-11-({4-[(2H-1,3-benzodioxol-5-yl)amino]-8-methylquinazolin-2-yl}methyl)-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-6-one
N-{[2-(dimethylamino)-5,8-dimethoxyquinolin-3-yl]methyl}-N-(furan-2-ylmethyl)-2-methylpropanamide
5-{1-[2-(oxan-2-yl)ethyl]-1H-imidazol-2-yl}-2-(thiophen-2-yl)pyrimidine
2-ethyl-N-[(4-methylphenyl)methyl]-3-oxo-2,9-diazaspiro[5.5]undecane-9-carboxamide
5-[(benzyloxy)methyl]-3-cyclopropyl-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazole
N,N-dimethyl-2-[1-methyl-5-(piperidin-1-yl)-1H-1,2,4-triazol-3-yl]aniline
2-(3-ethoxy-5-fluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
(2R,3R,6R)-3-(3-methoxyphenyl)-5-(pyridine-4-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
4-chloro-N,1,5-trimethyl-N-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}-1H-pyrazole-3-carboxamide
1-[(8-methoxy-2H-chromen-3-yl)methyl]-4-(5-methylpyridin-2-yl)piperidin-4-ol
2-(1H-1,3-benzodiazol-1-yl)-N-{pyrazolo[1,5-a]pyridin-3-ylmethyl}propanamide
N-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
5-[(3R,4R)-3-({[2-(dimethylamino)ethyl](methyl)amino}methyl)-4-(hydroxymethyl)pyrrolidine-1-carbonyl]-1-methyl-1,2-dihydropyridin-2-one
1-{4-[2-(4-fluorophenyl)morpholine-4-carbonyl]-3,5-dimethyl-1H-pyrrol-2-yl}ethan-1-one
(3S,4S)-4-[methyl(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)amino]-1-(pyridin-2-ylmethyl)pyrrolidin-3-ol
(1R,3S)-7-(5-cyclopropyl-3-methyl-1H-pyrazole-4-carbonyl)-3-methoxy-3-methyl-7-azaspiro[3.5]nonan-1-ol
6-[(6-methylpyridin-2-yl)methyl]-N-[(4-phenyloxan-4-yl)methyl]-6-azaspiro[2.5]octane-1-carboxamide
N-cyclohexyl-1,3-dimethyl-2,6-dioxo-N-(pyridin-2-ylmethyl)-1,2,3,6-tetrahydropyrimidine-4-carboxamide
ethyl 4-(4-{4-[(2,2-dimethyloxan-4-yl)amino]piperidin-1-yl}benzoyl)piperazine-1-carboxylate
N-cyclohexyl-N-[2-(ethylsulfanyl)ethyl]-6-methyl-4-oxo-1,4-dihydroquinoline-3-carboxamide
N-[(3,5-dimethyl-2-phenyl-1H-indol-7-yl)methyl]-6-oxo-1,4,5,6-tetrahydropyridazine-3-carboxamide
4-{1-phenyl-4-[1-(propan-2-yl)-1H,4H-pyrazolo[3,4-d]imidazol-5-yl]-1H-pyrazol-3-yl}pyridine
2,3-dimethoxy-N-{[4-({[3-(trifluoromethyl)phenyl]methyl}amino)quinazolin-2-yl]methyl}benzamide
2-benzyl-8-[(5-cyclopropyl-1-methyl-1H-pyrazol-4-yl)methyl]-2,8-diazaspiro[4.5]decan-3-one
3-(3,5-dimethyl-1H-pyrazol-1-yl)-N-{2-[4-(2-fluorophenyl)-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]ethyl}propanamide
2,4-dimethyl-N-{2-[(pyridin-3-yl)amino]ethyl}pyrimidine-5-carboxamide
1-cyclohexyl-3-(cyclopropylmethyl)-N-methyl-N-(1,2-oxazol-5-ylmethyl)-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
2-(5-amino-3-methyl-1H-pyrazol-1-yl)-N-({5-cyclohexyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)acetamide
(2S,4R)-1-benzyl-4-{[(4-chlorophenyl)methyl]amino}-N-(2-methoxyethyl)pyrrolidine-2-carboxamide
methyl 2-[8-(1-methoxypropan-2-yl)-2,4-dioxo-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decan-3-yl]acetate
4-[(2-{4-[(dimethylamino)methyl]phenyl}piperidin-1-yl)methyl]-1,5-dimethyl-1H-pyrrole-2-carbonitrile
1-{1-[(4-chlorophenyl)methyl]piperidin-4-yl}-N-(3-hydroxypropyl)-1H-1,2,3-triazole-4-carboxamide
1-{4-[(4-hydroxy-6,8-dimethylquinolin-2-yl)methyl]piperazin-1-yl}ethan-1-one