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2-[(4aR,7aS)-6,6-dioxo-4-[(1-propyl-1H-imidazol-2-yl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]-N,N-dimethylacetamide
2-[1-(2,2-dimethylpropyl)-3-oxopiperazin-2-yl]-N-{[1-(morpholin-4-yl)cyclopentyl]methyl}acetamide
5-{[3-(2-chlorophenyl)pyrrolidin-1-yl]methyl}-2-methoxybenzoic acid
(3S,4S)-1-(2-{[(4-fluorophenyl)methyl]carbamoyl}ethyl)-4-(propan-2-yl)pyrrolidine-3-carboxylic acid
N-(2-tert-butyl-7,7-dimethyl-5,6,7,8-tetrahydroquinazolin-5-yl)-4-(2-oxopyrrolidin-1-yl)butanamide
2-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}-1,2,3,4-tetrahydroisoquinolin-4-ol
1-{4-[2-(2H-1,3-benzodioxol-5-yl)-5-fluoro-1H-1,3-benzodiazol-1-yl]piperidin-1-yl}-2-(1H-pyrazol-1-yl)ethan-1-one
N-[(3R,4R)-3-hydroxypiperidin-4-yl]-2-(1,1,2,2-tetrafluoroethoxy)benzamide
6-{[4-(3-hydroxy-3-methylbut-1-yn-1-yl)phenyl]methyl}-N-[2-(1-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-6-azaspiro[2.5]octane-1-carboxamide
2-(4-{[5-methyl-2-(5-methylfuran-2-yl)-1,3-oxazol-4-yl]methyl}piperazin-1-yl)quinazoline
4-methanesulfonyl-N-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}benzamide
2-[7-(5-chloropyridin-2-yl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-N,N-diethylacetamide
1-methyl-4-[2-(6-oxo-1,6-dihydropyrimidin-5-yl)acetyl]-1,4,9-triazaspiro[5.6]dodecan-10-one
N-[(1S,2R)-2-aminocyclobutyl]-2-(4-fluoro-3-methylbenzenesulfonamido)acetamide
5-[(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-3-hydroxypiperidine-1-carbonyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
4-{1-[(5-phenylthiophen-2-yl)methyl]azetidin-3-yl}morpholine
3-[(1R,5S)-3,8-diazabicyclo[3.2.1]octan-3-ylmethyl]-N-(1-ethyl-1H-1,2,3-triazol-4-yl)benzamide
2-{4-[3-(aminomethyl)pyrrolidin-1-yl]-6-oxo-1,6-dihydropyridazin-1-yl}-N-methyl-N-(propan-2-yl)acetamide
N-[(4-{2-[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]ethoxy}-3-methoxyphenyl)methyl]-N-[(3S)-2-oxoazepan-3-yl]pyridine-2-carboxamide
5-({2-cyclopentyl-3-oxo-2,9-diazaspiro[5.5]undecan-9-yl}methyl)-N-methyl-1,2,4-oxadiazole-3-carboxamide
(4aS,8aR)-6-[(4-methyl-1,3-thiazol-5-yl)methyl]-1-[2-(thiophen-2-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
N-[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]-1-(2-ethoxyethyl)-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
2,6-dihydroxy-N-{[4-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}benzamide
N-[2-(dimethylamino)ethyl]-3-(1-{8-oxatricyclo[7.4.0.02,7]trideca-1(9),2(7),3,5,10,12-hexaen-6-ylmethyl}piperidin-4-yl)propanamide
1-[3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)propanoyl]-4-(1H-pyrazol-1-yl)piperidine-4-carboxylic acid
N-{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-N-methyl-3-(4-methyl-1,3-thiazol-5-yl)propanamide
1-(3-chloro-4-methoxyphenyl)-N-(1,2-oxazol-3-ylmethyl)-5-oxopyrrolidine-3-carboxamide
N-[1-(2,3-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3-(1-oxo-2,3-dihydro-1H-isoindol-2-yl)propanamide
2-({4-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)benzoic acid
2,3,5-trimethyl-N-[1-(1-methyl-1H-imidazol-2-yl)butyl]pyrazolo[1,5-a]pyrimidin-7-amine
1-[2-(dimethylamino)-5,6-dimethylpyrimidin-4-yl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
4-{4-[4-cyclopropyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-methylpyrimidine
(1S,5R)-6-benzyl-3-(1,4-dithiepan-6-yl)-3,6-diazabicyclo[3.2.2]nonan-7-one
8-(5-acetylthiophene-3-carbonyl)-3-(3-methylbutyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
8-(butane-1-sulfonyl)-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
7-(2,2-diphenylacetyl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
5-chloro-N-(2-oxopyrrolidin-3-yl)-3-phenyl-1H-indole-2-carboxamide
4-[(4-methoxyphenyl)methyl]-1-(4-methylbenzoyl)-1,4-diazepan-5-one
1-[(1-ethyl-1H-pyrazol-4-yl)methyl]-4-(2-methylpyridin-4-yl)-1,4-diazepane
2-(3-methylbut-2-en-1-yl)-8-(pyrazin-2-yl)-2,8-diazaspiro[4.5]decan-3-one
methyl({2-methylimidazo[1,2-a]pyridin-3-yl}methyl){[5-(oxolan-2-yl)thiophen-2-yl]methyl}amine
N-butyl-4-{[2-(4-methoxyphenyl)ethyl]amino}-N,5-dimethylthieno[2,3-d]pyrimidine-6-carboxamide
3-chloro-6-[(3R,4R)-3-hydroxy-3,4-dimethylpyrrolidin-1-yl]pyridine-2-carboxylic acid
2-[2-benzyl-5-oxo-4-(2-phenylphenyl)piperazin-1-yl]-2-oxoacetamide
1-[1-(2,2-diphenylethyl)pyrrolidin-3-yl]-4-methylpiperazine
2-(2-methoxyethyl)-9-[2-(2-methyl-1H-imidazol-1-yl)propanoyl]-2,9-diazaspiro[5.5]undecan-3-one
1-{[1-(2-hydroxyethyl)-3-methyl-1H-pyrazol-4-yl]methyl}-4-(oxan-4-yl)-1,4-diazepan-6-ol
[4-({4-[2-(5-methylfuran-2-yl)propyl]-1H-1,2,3-triazol-1-yl}methyl)phenyl]methanol
1-[4-(pyridin-2-yl)piperazin-1-yl]-3-[1-(pyrimidin-2-yl)piperidin-3-yl]propan-1-one
(3R,4S)-1-(oxane-4-carbonyl)-4-phenylpyrrolidin-3-amine