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1-[1-(3-cyano-6-methylpyridin-2-yl)piperidin-4-yl]-N-cyclopropyl-1H-1,2,3-triazole-4-carboxamide
N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-2-[4-(trifluoromethyl)phenyl]-1,3-thiazole-4-carboxamide
3-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}-1-ethyl-4,6-dimethyl-1,2-dihydropyridin-2-one
4-amino-N-cyclopentyl-N-[(5-methylthiophen-2-yl)methyl]pyridine-2-carboxamide
N-({4-[(3-fluorophenyl)methoxy]phenyl}methyl)-4-methyl-N-(pyridin-2-ylmethyl)benzamide
3-{4-[(3,4-dimethylphenyl)methyl]piperazin-1-yl}-2,5-dimethylpyrazine
N-{1-[1-(1-benzofuran-2-ylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}-2-methoxy-2-phenylacetamide
4-[4-(pyridin-2-ylmethyl)-1,4-diazepane-1-carbonyl]benzene-1-sulfonamide
N3-(1-benzothiophen-2-ylmethyl)-N5-cycloheptyl-1-cyclopropyl-N3-methyl-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
N-cyclopentyl-2-[4-(morpholin-4-yl)-6-oxo-1,6-dihydropyridazin-1-yl]butanamide
3-(1-cyclopentyl-3-methyl-1H-pyrazol-5-yl)-1-[(1-methyl-1H-imidazol-2-yl)methyl]-1-propylurea
2-methyl-N-(1-methyl-3-{1-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-1,2,5,6-tetrahydropyridin-3-yl}-1H-pyrazol-5-yl)propanamide
2-{3-[(4-cyclopropyl-1H-1,2,3-triazol-1-yl)methyl]piperidine-1-carbonyl}-5-methylpyrazine
N-[4-(3-cyclopropyl-1-phenyl-1H-1,2,4-triazol-5-yl)phenyl]acetamide
N-[(1-methyl-1H-imidazol-2-yl)methyl]-N-(propan-2-yl)-5-[(5,6,7,8-tetrahydronaphthalen-2-yloxy)methyl]-1,2-oxazole-3-carboxamide
5-[1-(2,2-dimethylpropyl)-4-hydroxypiperidin-4-yl]-N-methyl-N-(quinolin-8-ylmethyl)-1-benzofuran-2-carboxamide
3-[(1H-indol-3-ylmethyl)amino]-N-(pyridin-2-ylmethyl)-5-(pyrrolidine-1-sulfonyl)benzamide
3-(1-{[2-(3-methylphenyl)pyrimidin-5-yl]methyl}piperidin-4-yl)-N-(oxolan-2-ylmethyl)propanamide
1-{[3-(2,5-dimethylthiophen-3-yl)-1-(2-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N,N-dimethylpyrrolidin-3-amine
3-[N-(2-phenylethyl)-1-(1,3,7-trimethyl-1H-indol-2-yl)formamido]propanamide
N-{2-[(6-methylpyridazin-3-yl)amino]ethyl}pyridine-3-carboxamide
1-[(2-methoxyphenyl)methyl]-6-oxo-N-[2-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)ethyl]piperidine-3-carboxamide
N-cyclopropyl-2-[4-(4-methyl-2,5-dioxoimidazolidin-4-yl)piperidin-1-yl]pyridine-4-carboxamide
N-{2-[(2-methyl-1H-imidazol-1-yl)methyl]phenyl}morpholine-2-carboxamide
N-methyl-N-[2-(pyridin-2-yl)ethyl]-3-{1-[2-(pyridin-2-ylsulfanyl)acetyl]piperidin-3-yl}propanamide
3-[2-(7-fluoro-1-methyl-1,2,3,4-tetrahydroisoquinolin-2-yl)-2-oxoethyl]-5,5-dimethyl-1,3-oxazolidine-2,4-dione
N-methyl-3-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]-N-{[3-(3-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl}propanamide
3-{1-[(1-methyl-1H-pyrazol-4-yl)methyl]piperidin-3-yl}-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
(4aS,7aR)-1-(4-fluoro-3-methylbenzoyl)-4-(3-methylbutanoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-(4-fluoro-2-methylphenyl)-2-{[1-(4-oxo-3,4-dihydroquinazolin-3-yl)propan-2-yl]amino}acetamide
9-[3-(pyridin-4-yl)propanoyl]-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
4-[(4-phenyl-1,3-thiazol-2-yl)methyl]thiomorpholine
2-(4-tert-butylphenoxymethyl)-4-hydroxy-N-[1-(pyrimidin-4-yl)ethyl]pyrimidine-5-carboxamide
[(2,3-difluoro-6-methoxyphenyl)methyl](methyl)[1-(pyridin-4-yl)ethyl]amine
N-(butan-2-yl)-5-methyl-4-{methyl[2-(pyridin-2-yl)ethyl]amino}thieno[2,3-d]pyrimidine-6-carboxamide
1-(5-methoxy-2-{[(1-phenylcyclopropyl)amino]methyl}phenoxy)-3-(pyrrolidin-1-yl)propan-2-ol
3,5-dimethyl-1-[4-(trifluoromethoxy)phenyl]-1H-1,2,4-triazole
N-{[2-(2-methoxyphenoxy)pyridin-3-yl]methyl}-2-oxo-1,3-oxazolidine-4-carboxamide
4-methyl-N-[(3S)-2-oxoazepan-3-yl]-N-({4-[3-(pyridin-3-yl)propoxy]phenyl}methyl)-1,2,5-oxadiazole-3-carboxamide
1-{2-[4-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)phenyl]acetyl}-3-propylpiperidine-3-carboxylic acid
1-[2-(4-chlorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]-3-methoxypropan-1-one
6-{1-oxa-7-azaspiro[3.5]nonan-7-yl}-N-[3-(pyridin-2-yl)propyl]pyridine-3-carboxamide
[2-ethoxy-5-({[2-(pyridin-3-yloxy)propyl]amino}methyl)phenyl]methyl acetate
5-methoxy-3-{[4-(1-methylpiperidin-4-yl)piperidin-1-yl]methyl}-1H-indazole
1-(furan-2-ylmethyl)-4-{imidazo[1,2-a]pyridine-3-carbonyl}-1,4-diazepan-6-ol
(5-{1,8-dioxa-4,11-diazaspiro[5.6]dodecan-4-ylmethyl}-2-ethoxyphenyl)methanol
4-[2-methyl-1-(3-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}piperidin-1-yl)propan-2-yl]morpholine
N-(3,4-difluorophenyl)-1-{[5-(1,2-oxazol-3-yl)thiophen-2-yl]sulfonyl}piperidin-3-amine
4-[4-methyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-[(5-methylthiophen-2-yl)methyl]piperidine
3-(2H-1,3-benzodioxol-5-yl)-5-(cyclopentylmethyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine