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(1S,5R)-3-[2-(3-methylphenyl)acetyl]-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
9-[(1S,6R)-3,9-diazabicyclo[4.2.1]nonan-9-yl]-3-azaspiro[5.5]undecane
dimethyl[1-(4-{1-[(4-methylphenyl)methyl]-1H-1,2,3-triazol-4-yl}phenyl)ethyl]amine
3-methyl-7-[2-(methylsulfanyl)-1,3-thiazole-4-carbonyl]-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
1-(2-methoxypyridine-3-carbonyl)-4-(2-methylquinolin-6-yl)piperidin-4-ol
{[1-(furan-2-ylmethyl)piperidin-4-yl]methyl}(methyl)[(4-methyl-1H-imidazol-2-yl)methyl]amine
1-{5-[(3aS,6aS)-octahydropyrrolo[2,3-c]pyrrole-1-carbonyl]-2-methylphenyl}imidazolidin-2-one
methyl (2S,4R)-1-{[(4S)-4-(prop-1-en-2-yl)cyclohex-1-en-1-yl]methyl}-4-[2-(1H-pyrazol-1-yl)benzamido]pyrrolidine-2-carboxylate
4-methyl-N-{[1-(2-methylpropyl)pyrrolidin-3-yl]methyl}-1H-imidazole-5-carboxamide
1-[3-(hydroxymethyl)phenyl]-4-oxo-5-phenoxy-1,4-dihydropyridine-3-carboxylic acid
4-[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]-N-{2-[methyl(phenyl)amino]propyl}butanamide
(3S,4S)-4-cyclopropyl-1-(pyridine-3-sulfonyl)pyrrolidine-3-carboxylic acid
5-(azocane-1-carbonyl)-2-benzyl-1,3-benzoxazole
3-(3-methoxyphenoxy)-1-{[1,2,4]triazolo[1,5-a]pyrimidine-2-carbonyl}azetidine
7-(1,3-benzothiazol-2-yl)-9-methoxy-4-[(2-methoxyphenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-[(1-methyl-2-oxo-1,2,3,4-tetrahydroquinolin-4-yl)methyl]-2-oxo-1H,2H,5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
2-(6-chloro-2H-1,3-benzodioxol-5-yl)-1-[2-(1-methylpyrrolidin-2-yl)ethyl]-1H-imidazole
1-(butan-2-yl)-3-(6-fluoropyridin-3-yl)-1-(pyridin-2-ylmethyl)urea
1-cyclopropyl-4-(4-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-yl}piperidine-1-carbonyl)pyrrolidin-2-one
2-(3-methoxypropyl)-8-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
1-{1-[4-(2H-1,3-benzodioxol-5-yl)pyrimidin-2-yl]-5-cyclopropyl-1H-pyrazole-4-carbonyl}azepane
6-[(1S,6R)-3,9-diazabicyclo[4.2.1]nonan-9-yl]-N-[(4-ethyl-1,3-thiazol-2-yl)methyl]pyridine-3-carboxamide
N-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-1-{[3-(trifluoromethyl)phenyl]methyl}-1H-1,2,3-triazole-4-carboxamide
2-[4-(ethoxycarbonyl)piperazin-1-yl]-2-[4-(1H-pyrazol-5-yl)phenyl]acetic acid
2-[4-(furan-3-ylmethyl)morpholin-3-yl]-N-methyl-N-[(5-methylthiophen-2-yl)methyl]acetamide
1-methyl-1'-[3-(2-methylpropyl)-1,2-oxazole-5-carbonyl]-1,2-dihydrospiro[indole-3,3'-piperidine]-2-one
N2,N2,6-trimethyl-N4-{1-[4-methyl-2-(pyridin-4-yl)pyrimidin-5-yl]ethyl}pyrimidine-2,4-diamine
3-{2-[(4-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}-N-methyl-N-[1-(thiophen-2-yl)ethyl]propanamide
2-hydroxy-5-{[2-(2-methoxyethyl)morpholin-4-yl]methyl}benzoic acid
methyl 4-(4-{[4-(3-methylphenyl)phenyl]carbamoyl}piperidin-1-yl)-4-oxobutanoate
4-(1H-imidazol-2-yl)-1-[3-(2-methyl-1H-imidazol-1-yl)-1-phenylpropyl]-1H-1,2,3-triazole
6-[(3S,4S)-3,4-dihydroxypiperidin-1-yl]-N-methyl-N-(quinolin-2-ylmethyl)pyridine-3-carboxamide
N-methyl-N-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]quinoline-2-carboxamide
2-(1-{[3-(2,5-dimethylphenyl)-1H-pyrazol-4-yl]methyl}-3-oxopiperazin-2-yl)-N-methylacetamide
N-{1-[(4-chlorophenyl)methyl]piperidin-3-yl}-2-[(5-ethyl-1,3,4-oxadiazol-2-yl)sulfanyl]acetamide
2-(3-fluorophenyl)-N-[(2-methyl-1,3-thiazol-4-yl)methyl]-1,3-benzoxazole-5-carboxamide
1-(4-{4-[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]pyrimidin-2-yl}-1,4-diazepan-1-yl)ethan-1-one
3-(2H-1,3-benzodioxol-5-ylmethyl)-1-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}-3-methylpiperidine
5-[4-(2-ethylpyrimidine-5-carbonyl)piperazin-1-yl]-2-methyl-2,3-dihydropyridazin-3-one
(3R,4R)-1-{furo[3,2-c]pyridin-4-yl}-4-(morpholin-4-yl)piperidin-3-ol
(2-methoxyethyl)({2-phenyl-1-[1-(quinoxalin-5-ylmethyl)piperidin-4-yl]ethyl})(pyridin-2-ylmethyl)amine
(3aR,6aS)-5-[(5-chloro-2-fluorophenyl)methyl]-2-methyl-octahydropyrrolo[3,4-c]pyrrole-1,3-dione
N-[(5-{[3-(2-aminoethyl)phenyl]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl)methyl]-2-methoxyacetamide
1-(5-{3-[1-(pyridin-2-ylmethyl)-1H-pyrazol-3-yl]phenyl}thiophen-2-yl)ethan-1-one
2-(4-fluorophenyl)-4-[3-(5-methylthiophen-2-yl)-1H-pyrazole-5-carbonyl]morpholine
5-cyclobutyl-N-[2-(dimethylamino)-2-(5-methylfuran-2-yl)ethyl]-1,3,4-oxadiazol-2-amine
N-[2-(1H-imidazol-4-yl)ethyl]-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
3-(2-{[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]carbamoyl}piperidine-1-carbonyl)pyridin-1-ium-1-olate
4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]-N-[(4-methylphenyl)methyl]piperidine-1-carboxamide
(4aS,7aR)-1-(3-chloro-5-methoxybenzoyl)-4-propyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione